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- [1] In vitro characterization of TAS-121, a novel, highly potent, and mutant-specific EGFR-TKI.[J]. MOLECULAR CANCER THERAPEUTICS, 2013, 12 (11)Ito, Kimihiro论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Tsukuba, Ibaraki, JapanMiyadera, Kazutaka论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Tsukuba, Ibaraki, JapanAoyagi, Yoshimi论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Tsukuba, Ibaraki, JapanKato, Masanori论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Tsukuba, Ibaraki, JapanYonekura, Kazuhiko论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Tsukuba, Ibaraki, JapanIwasawa, Yoshikazu论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Tsukuba, Ibaraki, JapanUtsugi, Teruhiro论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Tsukuba, Ibaraki, Japan
- [2] Characterization of TAS-121, a novel mutant-specific EGFR-TKI, on pharmacokinetics, pharmacodynamics, and antitumor activity.[J]. MOLECULAR CANCER THERAPEUTICS, 2013, 12 (11)Kato, Masanori论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Ibaraki, JapanMiyadera, Kazutaka论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Ibaraki, JapanShibata, Yoshihiro论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Ibaraki, JapanIto, Kimihiro论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Ibaraki, JapanAoyagi, Yoshimi论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Ibaraki, JapanChiba, Masato论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Ibaraki, JapanYonekura, Kazuhiko论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Ibaraki, JapanIwasawa, Yoshikazu论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Ibaraki, JapanUtsugi, Teruhiro论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Ibaraki, Japan
- [3] Hsp90 inhibition suppresses mutant EGFR-T790M signaling and overcomes kinase inhibitor resistance[J]. CANCER RESEARCH, 2008, 68 (14) : 5827 - 5838Shimamura, Takeshi论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Brigham & Womens Hosp, Dept Med, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USALi, Danan论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Harvard Univ, Ctr Canc, Ludwig Ctr Dana Farber, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAJi, Hongbin论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Harvard Univ, Ctr Canc, Ludwig Ctr Dana Farber, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAHaringsma, Henry J.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USALiniker, Elizabeth论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USABorgman, Christa L.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USALowell, April M.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAMinami, Yuko论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Dana Farber Canc Inst, Ctr Canc Genome Discovery, Boston, MA 02215 USA Brigham & Womens Hosp, Dept Med, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAMcNamara, Kate论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAPerera, Samanthi A.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Harvard Univ, Ctr Canc, Ludwig Ctr Dana Farber, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAZaghlul, Sara论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAThomas, Roman K.论文数: 0 引用数: 0 h-index: 0机构: Univ Cologne, Ctr Integrated Oncol, Cologne, Germany Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAGreulich, Heidi论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Dana Farber Canc Inst, Ctr Canc Genome Discovery, Boston, MA 02215 USA Harvard Univ, Broad Inst, Cambridge, MA 02138 USA MIT, Cambridge, MA 02139 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAKobayashi, Susumu论文数: 0 引用数: 0 h-index: 0机构: Beth Israel Deaconess Med Ctr, Dept Med, Boston, MA 02215 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAChirieac, Lucian R.论文数: 0 引用数: 0 h-index: 0机构: Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAPadera, Robert F.论文数: 0 引用数: 0 h-index: 0机构: Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAKubo, Shigeto论文数: 0 引用数: 0 h-index: 0机构: Beth Israel Deaconess Med Ctr, Dept Radiol, Boston, MA 02215 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USATakahashi, Masaya论文数: 0 引用数: 0 h-index: 0机构: Beth Israel Deaconess Med Ctr, Dept Radiol, Boston, MA 02215 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USATenen, Daniel G.论文数: 0 引用数: 0 h-index: 0机构: Beth Israel Deaconess Med Ctr, Dept Med, Boston, MA 02215 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA论文数: 引用数: h-index:机构:Wong, Kwok-Kin论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Harvard Univ, Ctr Canc, Ludwig Ctr Dana Farber, Boston, MA 02115 USA Brigham & Womens Hosp, Dept Med, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAShapiro, Geoffrey I.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Brigham & Womens Hosp, Dept Med, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA
- [4] TAS-121, A Selective Mutant EGFR Inhibitor, Shows Activity Against Tumors Expressing Various EGFR Mutations Including T790M and Uncommon Mutations G719X[J]. MOLECULAR CANCER THERAPEUTICS, 2019, 18 (05) : 920 - 928Ito, Kimihiro论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, JapanNishio, Makoto论文数: 0 引用数: 0 h-index: 0机构: Japanese Fdn Canc Res, Canc Inst Hosp, Dept Thorac Med Oncol, Tokyo, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, JapanKato, Masanori论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, JapanMurakami, Haruyasu论文数: 0 引用数: 0 h-index: 0机构: Shizuoka Canc Ctr, Div Thorac Oncol, Shizuoka, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, JapanAoyagi, Yoshimi论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, JapanOhe, Yuichiro论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr, Dept Thorac Oncol, Tokyo, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, JapanOkayama, Takashige论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, JapanHashimoto, Akihiro论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, JapanOhsawa, Hirokazu论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, JapanTanaka, Gotaro论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, JapanNonoshita, Katsumasa论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, JapanIto, Satoru论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, JapanMatsuo, Kenichi论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, JapanMiyadera, Kazutaka论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, Ibaraki, Japan
- [5] Discovery of a Potent and Mutant-Selective EGFR Inhibitor that Overcomes T790M-Mediated Resistance in Lung Cancer[J]. Targeted Oncology, 2018, 13 : 389 - 398Dong Ha Kim论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Pulmonology and Critical Care Medicine, Asan Medical CenterYun Jung Choi论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Pulmonology and Critical Care Medicine, Asan Medical CenterSeon Ye Kim论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Pulmonology and Critical Care Medicine, Asan Medical CenterJung-Eun Lee论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Pulmonology and Critical Care Medicine, Asan Medical CenterKi Jung Sung论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Pulmonology and Critical Care Medicine, Asan Medical CenterYoung Hoon Sung论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Pulmonology and Critical Care Medicine, Asan Medical CenterWoo Sung Kim论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Pulmonology and Critical Care Medicine, Asan Medical CenterSung-Eun Kim论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Pulmonology and Critical Care Medicine, Asan Medical CenterHyung Chul Ryu论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Pulmonology and Critical Care Medicine, Asan Medical CenterJae Sun Kim论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Pulmonology and Critical Care Medicine, Asan Medical CenterLu Guangying论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Pulmonology and Critical Care Medicine, Asan Medical CenterChang-Min Choi论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Pulmonology and Critical Care Medicine, Asan Medical CenterJin Kyung Rho论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Pulmonology and Critical Care Medicine, Asan Medical CenterJae Cheol Lee论文数: 0 引用数: 0 h-index: 0机构: University of Ulsan,Department of Pulmonology and Critical Care Medicine, Asan Medical Center
- [6] Discovery of a Potent and Mutant-Selective EGFR Inhibitor that Overcomes T790M-Mediated Resistance in Lung Cancer[J]. TARGETED ONCOLOGY, 2018, 13 (03) : 389 - 398Kim, Dong Ha论文数: 0 引用数: 0 h-index: 0机构: Univ Ulsan, Dept Pulmonol & Crit Care Med, Coll Med, Asan Med Ctr, Seoul 05505, South Korea Univ Ulsan, Asan Inst Life Sci, Coll Med, Asan Med Ctr, Seoul 05505, South Korea Univ Ulsan, Dept Pulmonol & Crit Care Med, Coll Med, Asan Med Ctr, Seoul 05505, South KoreaChoi, Yun Jung论文数: 0 引用数: 0 h-index: 0机构: Univ Ulsan, Dept Pulmonol & Crit Care Med, Coll Med, Asan Med Ctr, Seoul 05505, South Korea Univ Ulsan, Asan Inst Life Sci, Coll Med, Asan Med Ctr, Seoul 05505, South Korea Univ Ulsan, Dept Pulmonol & Crit Care Med, Coll Med, Asan Med Ctr, Seoul 05505, South KoreaKim, Seon Ye论文数: 0 引用数: 0 h-index: 0机构: Univ Ulsan, Dept Pulmonol & Crit Care Med, Coll Med, Asan Med Ctr, Seoul 05505, South Korea Univ Ulsan, Asan Inst Life Sci, Coll Med, Asan Med Ctr, Seoul 05505, South Korea Univ Ulsan, Dept Pulmonol & Crit Care Med, Coll Med, Asan Med Ctr, Seoul 05505, South KoreaLee, Jung-Eun论文数: 0 引用数: 0 h-index: 0机构: Univ Ulsan, Dept Pulmonol & Crit Care Med, Coll Med, Asan Med Ctr, Seoul 05505, South Korea Univ Ulsan, Asan Inst Life Sci, Coll Med, Asan Med Ctr, Seoul 05505, South Korea Univ Ulsan, Dept Pulmonol & Crit Care Med, Coll Med, Asan Med Ctr, Seoul 05505, South KoreaSung, Ki Jung论文数: 0 引用数: 0 h-index: 0机构: Univ Ulsan, Dept Pulmonol & Crit Care Med, Coll Med, Asan Med Ctr, Seoul 05505, South Korea Univ Ulsan, Asan Inst Life Sci, Coll Med, Asan Med Ctr, Seoul 05505, South Korea Univ Ulsan, Dept Pulmonol & Crit Care Med, Coll Med, Asan Med Ctr, Seoul 05505, South KoreaSung, Young Hoon论文数: 0 引用数: 0 h-index: 0机构: Univ Ulsan, Asan Inst Life Sci, Coll Med, Asan Med Ctr, Seoul 05505, South Korea Univ Ulsan, Dept Convergence Med, Coll Med, Asan Med Ctr, Seoul 05505, South Korea Univ Ulsan, Dept Pulmonol & Crit Care Med, Coll Med, Asan Med Ctr, Seoul 05505, South KoreaKim, Woo Sung论文数: 0 引用数: 0 h-index: 0机构: Univ Ulsan, Dept Pulmonol & Crit Care Med, Coll Med, Asan Med Ctr, Seoul 05505, South Korea Univ Ulsan, Dept Pulmonol & Crit Care Med, Coll Med, Asan Med Ctr, Seoul 05505, South KoreaKim, Sung-Eun论文数: 0 引用数: 0 h-index: 0机构: Oncobix, Yongin 16950, South Korea Univ Ulsan, Dept Pulmonol & Crit Care Med, Coll Med, Asan Med Ctr, Seoul 05505, South KoreaRyu, Hyung Chul论文数: 0 引用数: 0 h-index: 0机构: J2H Biotech, Ansan 16648, South Korea Univ Ulsan, Dept Pulmonol & Crit Care Med, Coll Med, Asan Med Ctr, Seoul 05505, South KoreaKim, Jae Sun论文数: 0 引用数: 0 h-index: 0机构: J2H Biotech, Ansan 16648, South Korea Univ Ulsan, Dept Pulmonol & Crit Care Med, Coll Med, Asan Med Ctr, Seoul 05505, South KoreaLu Guangying论文数: 0 引用数: 0 h-index: 0机构: East China Univ Sci & Technol, Coll Pharm, Shanghai 200237, Peoples R China Univ Ulsan, Dept Pulmonol & Crit Care Med, Coll Med, Asan Med Ctr, Seoul 05505, South KoreaChoi, Chang-Min论文数: 0 引用数: 0 h-index: 0机构: Univ Ulsan, Dept Pulmonol & Crit Care Med, Coll Med, Asan Med Ctr, Seoul 05505, South Korea Univ Ulsan, Dept Oncol, Coll Med, Asan Med Ctr, Seoul 05505, South Korea Univ Ulsan, Dept Pulmonol & Crit Care Med, Coll Med, Asan Med Ctr, Seoul 05505, South KoreaRho, Jin Kyung论文数: 0 引用数: 0 h-index: 0机构: Univ Ulsan, Dept Convergence Med, Coll Med, Asan Med Ctr, Seoul 05505, South Korea Univ Ulsan, Dept Asan Inst Life Sci, Coll Med, 86 Asanbyeoungwon Gil, Seoul 138736, South Korea Univ Ulsan, Dept Pulmonol & Crit Care Med, Coll Med, Asan Med Ctr, Seoul 05505, South KoreaLee, Jae Cheol论文数: 0 引用数: 0 h-index: 0机构: Univ Ulsan, Dept Oncol, Coll Med, Asan Med Ctr, Seoul 05505, South Korea Univ Ulsan, Dept Oncol, Asan Med Ctr, Coll Med, Olymp Ro 43 Gil, Seoul 138736, South Korea Univ Ulsan, Dept Pulmonol & Crit Care Med, Coll Med, Asan Med Ctr, Seoul 05505, South Korea
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