Potent and isoform-selective ATAD2 bromodomain inhibitor with unprecedented chemical structure and mode of action

被引：0
|
作者：
Fernandez-Montalvan, Amaury E.
Berger, Markus
Kuropka, Benno
Koo, Seong Joo
Badock, Volker
Weiske, Joerg
Holton, Simon J.
Chaikuad, Apirat
Diaz-Saez, Laura
Bennett, James
Federov, Oleg
Huber, Kilian
Centrella, Paolo
Clark, Matthew A.
Dumelin, Christoph E.
Sigel, Eric A.
Soutter, Holly S.
Troast, Dawn M.
Zhang, Ying
Cuozzo, John W.
Keefe, Anthony D.
Roche, Didier
Rodeschini, Vincent
Huebner, Jan
Weinmann, Hilmar
Hartung, Ingo V.
Gorjanacz, Matyas
机构：
来源：
CANCER RESEARCH | 2017年 / 77卷
关键词：
D O I：
10.1158/1538-7445.AM2017-5084
中图分类号：
R73 [肿瘤学];
学科分类号：
100214 ;
摘要：
5084
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收藏
页数：2
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