Suzuki-Miyaura cross-coupling reaction in the functionalization of the C ring of morphinans

被引:1
|
作者
Sipos, Attila [1 ]
Berenyi, Sandor [1 ]
机构
[1] Univ Debrecen, Dept Organ Chem, H-4010 Debrecen, Hungary
关键词
Suzuki-Miyaura cross-coupling of tosylates and mesylates; spatially hindered position; 14-arylmorphinan; opioid receptor binding affinity; microwave activation;
D O I
10.2174/157017807780414145
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
New methods have been developed for the functionalization of the non-aromatic C ring of morphinans with Suzuki-Miyaura cross-coupling of sulfonates and bromides.
引用
收藏
页码:146 / 150
页数:5
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