Higher blood brain barrier penetration of [14C]apalutamide and [14C]enzalutamide compared to [14C]darolutamide in rats using whole-body autoradiography.

被引:34
|
作者
Zurth, Christian
Sandman, Steffen
Trummel, Dagmar
Seidel, Dietrich
Nubbemeyer, Reinhard
Gieschen, Hille
机构
[1] Bayer AG, Berlin, Germany
[2] Bayer AG, Wuppertal, Germany
关键词
D O I
10.1200/JCO.2019.37.7_suppl.156
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
156
引用
收藏
页数:1
相关论文
共 50 条
  • [1] Blood-brain barrier penetration of [14C]darolutamide compared with [14C]enzalutamide in rats using whole body autoradiography.
    Zurth, Christian
    Sandmann, Steffen
    Trummel, Dagmar
    Seidel, Dietrich
    Gieschen, Hille
    JOURNAL OF CLINICAL ONCOLOGY, 2018, 36 (06)
  • [2] Orally administered [14C]DPA and [14C]DHA are metabolised differently to [14C]EPA in rats
    Kaur, Gunveen
    Molero, Juan C.
    Weisinger, Harrison S.
    Sinclair, Andrew J.
    BRITISH JOURNAL OF NUTRITION, 2013, 109 (03) : 441 - 448
  • [3] [14C]-testosterone, [14C]-benzoic acid, and [14C]-caffeine: Comparative in vitro dermal penetration studies
    Dummer, Karen
    Ford, Gill
    McEwen, Andrew B.
    Wood, Stuart G.
    DRUG METABOLISM REVIEWS, 2006, 38 : 179 - 179
  • [4] UPTAKE OF [14C]GLUTAMINE IN TISSUES OF MOUSE STUDIED BY WHOLE-BODY AUTORADIOGRAPHY
    CASSANO, GB
    HANSSON, E
    JOURNAL OF NEUROCHEMISTRY, 1965, 12 (9-10) : 851 - &
  • [5] Natural 14C in Saccoglossus bromophenolosus compared to 14C in surrounding sediments
    Teuten, Emma L.
    King, Gary M.
    Reddy, Christopher M.
    MARINE ECOLOGY PROGRESS SERIES, 2006, 324 : 167 - 172
  • [6] ABSORPTION OF 14C OLEIC ACID AND 14C TRIOLEIN IN BILE FISTULA RATS
    GALLAGHE.N
    WEBB, J
    DAWSON, AM
    CLINICAL SCIENCE, 1965, 29 (01) : 73 - &
  • [7] Covalent binding of radioactivity from [14C]rofecoxib, but not [14C]celecoxib or [14C]CS-706, to the arterial elastin of rats
    Oitate, Masataka
    Hirota, Takashi
    Koyama, Kumiko
    Inoue, Shin-ichi
    Kawai, Kenji
    Ikeda, Toshihiko
    DRUG METABOLISM AND DISPOSITION, 2006, 34 (08) : 1417 - 1422
  • [8] Microchannel plate detectors for 14C autoradiography
    Lees, JE
    Fraser, GW
    Carthew, P
    IEEE TRANSACTIONS ON NUCLEAR SCIENCE, 1998, 45 (03) : 1288 - 1292
  • [9] Microchannel plate detectors for 14C autoradiography
    Lees, JE
    Fraser, GW
    Carthew, P
    1997 IEEE NUCLEAR SCIENCE SYMPOSIUM - CONFERENCE RECORD, VOLS 1 & 2, 1998, : 1610 - 1614
  • [10] Tissue distribution of [14C]-EDP-420 in the rat by quantitative whole-body autoradiography
    Jiang, L. J.
    Takeuchi, M.
    Lewsley, R.
    Sonderfan, A.
    Baba, T.
    Or, Y. S.
    INTERNATIONAL JOURNAL OF ANTIMICROBIAL AGENTS, 2007, 29 : S605 - S605