One-pot synthesis of 3-(2-cyanophenyl)-quinazolin-4(3H)-one

被引：0
|
作者：
Szczepankiewicz, W [1 ]
Suwinski, J [1 ]
机构：
[1] Silesian Tech Univ, Inst Organ Chem & Technol, PL-44100 Gliwice, Poland
来源：
KHIMIYA GETEROTSIKLICHESKIKH SOEDINENII | 2000年 / 07期
关键词：
anthranilonitrile; 3-(2-cyanophenyl)quinazolin-4(3H)-one; N-formylation;
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Anthranilonitrile reacting with formic acid at room temperature for three days gave 64 % of 3-(2-cyanophenyl)quinazolin-4(3H)-one. Under similar conditions anthranilic acid, 4-nitroaniline and 2,5-dichloroaniline were N-formylated in good yields.
引用
收藏
页码：922 / 924
页数：3
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