Synthesis and evaluation of quinoline carboxyguanidines as antidiabetic agents

被引：146
|
作者：
Edmont, D [1 ]
Rocher, R [1 ]
Plisson, C [1 ]
Chenault, J [1 ]
机构：
[1] Univ Orleans, Inst Chim Organ & Analyt, F-45067 Orleans 2, France
来源：
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 2000年 / 10卷 / 16期
关键词：
D O I：
10.1016/S0960-894X(00)00354-1
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
The synthesis and in vivo activities of a series of substituted quinoline carboxyguanidines as a possible novel class of antidiabetic agents is described. (C) 2000 Elsevier Science Ltd. All rights reserved.
引用
收藏
页码：1831 / 1834
页数：4
相关论文
共 50 条
  • [1] Synthesis,Antidiabetic and Antitubercular Evaluation of Quinoline-pyrazolopyrimidine hybrids and Quinoline-4-Arylamines
    Cele, Nosipho
    Awolade, Paul
    Seboletswe, Pule
    Khubone, Lungisani
    Olofinsan, Kolawole
    Islam, Md. Shahidul
    Jordaan, Audrey
    Warner, Digby F.
    Singh, Parvesh
    CHEMISTRYOPEN, 2024, 13 (09):
  • [2] Synthesis and biological evaluation of β-lactams as potent antidiabetic agents
    Shaheen, Salma
    Arshad, Jahan Zaib
    Haider, Mansoor
    Ashraf, Adnan
    Ahmad, Muhammad Mahboob
    Ashfaq, Muhammad
    Ismail, Mostafa A.
    Najam, Tayyaba
    Shah, Syed Shoaib Ahmad
    NEW JOURNAL OF CHEMISTRY, 2024, 48 (46) : 19427 - 19440
  • [3] Synthesis and biological evaluation of esculetin derivatives as antidiabetic agents
    Han, Mengjie
    Feng, Jingmei
    Wang, Xiaoyu
    Wang, Jigang
    Liu, Yuxin
    Zhao, Ritong
    Mu, Yajuan
    JOURNAL OF MOLECULAR STRUCTURE, 2025, 1324
  • [4] SYNTHESIS AND EVALUATION OF SOME SUBSTITUTED THIADIAZOLES AS ANTIDIABETIC AGENTS
    Pattan, Shashikant R.
    Kekare, Prajact
    Pranesh
    Raveendra, L. H.
    Hariprasad, C. K.
    INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY, 2009, 18 (03) : 317 - 318
  • [5] Quinoline Based thiazolidinediones: Design, Synthesis, In Silico, In Vitro, Antioxidant and Antidiabetic Evaluation
    Mohd, Sharfuddin
    Bidye, Durgesh Paresh
    Dixit, Sheshagiri R.
    Revanasiddappa, B. C.
    Harish, Vancha
    Kumar, Rakesh
    Sharma, Vikas
    CHEMISTRYSELECT, 2024, 9 (41):
  • [6] Synthesis, Antidiabetic Evaluation and Bioisosteric Modification of Quinoline Incorporated 2-pyrazoline Derivatives
    Kumar, Abhishek
    Kumar, Pankaj
    Shetty, Chaithra Raju
    James, Jainey Puthenveettil
    Shetty, Honey Chandrashekhar
    INDIAN JOURNAL OF PHARMACEUTICAL EDUCATION AND RESEARCH, 2021, 55 (02) : 574 - 580
  • [7] Synthesis, Characterization and Biological Evaluation of Thiazolidinedione Derivative as Novel Antidiabetic Agents
    Patel, Shivkant
    Sen, Ashim Kumar
    Dash, Dillip Kumar
    Sadhu, Piyushkumar
    Kumari, Mamta
    Baile, Sunil Bhaurao
    JOURNAL OF PHARMACEUTICAL RESEARCH INTERNATIONAL, 2021, 33 (35A) : 123 - 133
  • [8] Design, synthesis, docking and biological evaluation of chalcones as promising antidiabetic agents
    Rammohan, Aluru
    Bhaskar, Baki Vijaya
    Venkateswarlu, Nagam
    Gu, Wei
    Zyryanov, Grigory V.
    BIOORGANIC CHEMISTRY, 2020, 95
  • [9] Synthesis and Evaluation of Novel Oleanolic Acid Derivatives as Potential Antidiabetic Agents
    Zhang, Liying
    Jia, Xiaojian
    Dong, Jizhe
    Chen, Dongyin
    Liu, Jun
    Zhang, Luyong
    Wen, Xiaoan
    CHEMICAL BIOLOGY & DRUG DESIGN, 2014, 83 (03) : 297 - 305
  • [10] Synthesis and biological evaluation of novel neoflavonoid derivatives as potential antidiabetic agents
    Wang, Bing
    Li, Na
    Liu, Teng
    Sun, Jie
    Wang, Xiaojing
    RSC ADVANCES, 2017, 7 (55): : 34448 - 34460
12345