One-pot synthesis of pyridine derivatives via diels-alder reactions of 2,4-dimethyl-5-methoxyoxazole

被引:14
|
作者
Bondock, S [1 ]
机构
[1] Mansoura Univ, Fac Sci, Dept Chem, Mansoura, Egypt
关键词
D O I
10.1002/hc.20064
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
A novel series of pyridine derivatives with anticipated biological activity have been synthesized via Diels-Alder reactions of 2,4-dimethyl-5-methoxyoxazole with different types of dienophiles. The regioselectivity of the cycloaddition was inverted from methylacrylate to tert-butylacrylate. The structural elucidation of the new compounds was carried on the basis of spectral and X-ray analyses. (C) 2005 Wiley Periodicals, Inc.
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收藏
页码:49 / 55
页数:7
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