SYNTHESIS AND ANTIMICROBIAL ACTIVITY OF PYRAZOLYL 1,3,4-OXADIAZOLES

被引：8
|
作者：
Padmavathi, Venkatapuram [1 ]
Reddy, Gali Sudhakar [1 ]
Reddy, Guda Dinneswara [1 ]
Payani, Thalari [1 ]
机构：
[1] Sri Venkateswara Univ, Dept Chem, Tirupati 517502, Andhra Pradesh, India
来源：
SYNTHETIC COMMUNICATIONS | 2010年 / 40卷 / 04期
关键词：
Antimicrobial activity; 1,3-dipolar cycloaddition; 1,3,4-oxadiazoles; pyrazolines; DERIVATIVES; AGENTS; 1,2,4-TRIAZOLES; OXADIAZOLES; ACIDS;
D O I：
10.1080/00397910902985531
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The pyrazolyl oxadiazoles are synthesized from arylsulfonylacetic acid methyl ester and benzylsulfonylacetic acid methyl ester. Preliminary antimicrobial screening of the compounds showed that bis heterocycles with a chloro-substituted benzyl moiety exhibited high activity.
引用
收藏
页码：482 / 493
页数：12
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