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- [1] Discovery of CCT251921: A potent, selective and orally bioavailable small molecule modulator of the mediator complex-associated kinases CDK8 and CDK19ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2016, 251Mallinger, Aurelie论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, England Inst Canc Res, London, EnglandSchiemann, Kai论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, Merck Serono, Darmstadt, Germany Inst Canc Res, London, EnglandRink, Christian论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, England Inst Canc Res, London, EnglandStieber, Frank论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, Merck Serono, Darmstadt, Germany Inst Canc Res, London, EnglandCalderini, Michel论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, Merck Serono, Darmstadt, Germany Inst Canc Res, London, EnglandStubbs, Mark论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, England Inst Canc Res, London, EnglandPoeschke, Oliver论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, Merck Serono, Darmstadt, Germany Inst Canc Res, London, EnglandBusch, Michael论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, Merck Serono, Darmstadt, Germany Inst Canc Res, London, EnglandCzodrowski, Paul论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, Merck Serono, Darmstadt, Germany Inst Canc Res, London, EnglandMusil, Djordje论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, Merck Serono, Darmstadt, Germany Inst Canc Res, London, EnglandSchwarz, Daniel论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, Merck Serono, Darmstadt, Germany Inst Canc Res, London, EnglandOrtiz-Ruiz, Maria-Jesus论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, England Inst Canc Res, London, EnglandSchneider, Richard论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, Merck Serono, Darmstadt, Germany Inst Canc Res, London, EnglandValenti, Melanie论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, England Inst Canc Res, London, EnglandBrandon, Alexis de Haven论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, England Inst Canc Res, London, EnglandWorkman, Paul论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, England Inst Canc Res, London, EnglandDale, Trevor论文数: 0 引用数: 0 h-index: 0机构: Cardiff Univ, Sch Biosci, Cardiff, S Glam, Wales Inst Canc Res, London, EnglandWienke, Dirk论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, Merck Serono, Darmstadt, Germany Inst Canc Res, London, EnglandClarke, Paul论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, England Inst Canc Res, London, EnglandEsdar, Christina论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, Merck Serono, Darmstadt, Germany Inst Canc Res, London, EnglandRaynaud, Florence论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, England Inst Canc Res, London, EnglandEccles, Suzanne论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, England Inst Canc Res, London, EnglandRohdich, Felix论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, Merck Serono, Darmstadt, Germany Inst Canc Res, London, EnglandBlagg, Julian论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, Merck Serono, Darmstadt, Germany Inst Canc Res, London, England
- [2] CDK8/CDK19 inhibition as therapeutic target of metastatic prostate cancerVIRCHOWS ARCHIV, 2017, 471 : S269 - S269Offermann, A.论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp UKSH, Inst Pathol, Lubeck, Germany Univ Hosp UKSH, Inst Pathol, Lubeck, GermanyBecker, F.论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp UKSH, Inst Pathol, Lubeck, Germany Univ Hosp UKSH, Inst Pathol, Lubeck, GermanyKluemper, N.论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp UKSH, Inst Pathol, Lubeck, Germany Univ Hosp UKSH, Inst Pathol, Lubeck, GermanyVogel, W.论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp UKSH, Inst Pathol, Lubeck, Germany Univ Hosp UKSH, Inst Pathol, Lubeck, GermanyBraegelmann, J.论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp UKSH, Inst Pathol, Lubeck, Germany Univ Hosp UKSH, Inst Pathol, Lubeck, GermanyPerner, S.论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp UKSH, Inst Pathol, Lubeck, Germany Univ Hosp UKSH, Inst Pathol, Lubeck, Germany
- [3] Preventing adaptive therapeutic resistance to CDK4/6 inhibition with CDK8/19 inhibitorsCANCER RESEARCH, 2022, 82 (04)Mack, Zachary论文数: 0 引用数: 0 h-index: 0Yastrebova, Margarita论文数: 0 引用数: 0 h-index: 0Khamidullina, Alvina论文数: 0 引用数: 0 h-index: 0Sharko, Amanda论文数: 0 引用数: 0 h-index: 0Ding, Xiaokai论文数: 0 引用数: 0 h-index: 0Bowe, Stephan论文数: 0 引用数: 0 h-index: 0Sashi, Nikitha论文数: 0 引用数: 0 h-index: 0Safa, Samantha论文数: 0 引用数: 0 h-index: 0Digsby, Kaitlyn论文数: 0 引用数: 0 h-index: 0Eckstrom, Amanda论文数: 0 引用数: 0 h-index: 0Sikirzhitski, Vitali论文数: 0 引用数: 0 h-index: 0Lim, Chang-Uk论文数: 0 引用数: 0 h-index: 0Tatarskiy, Victor论文数: 0 引用数: 0 h-index: 0Roninson, Igor论文数: 0 引用数: 0 h-index: 0Broude, Eugenia论文数: 0 引用数: 0 h-index: 0
- [4] Studies of CDK 8/19 inhibitors: Discovery of novel and selective CDK8/19 dual inhibitors and elimination of their CYP3A4 time-dependent inhibition potentialBIOORGANIC & MEDICINAL CHEMISTRY, 2017, 25 (12) : 3018 - 3033Fujimoto, Jun论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Shonan Res Ctr, Pharmaceut Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Shonan Res Ctr, Pharmaceut Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, JapanHirayama, Takaharu论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Shonan Res Ctr, Pharmaceut Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Shonan Res Ctr, Pharmaceut Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, JapanHirata, Yasuhiro论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Shonan Res Ctr, Pharmaceut Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Shonan Res Ctr, Pharmaceut Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, JapanHikichi, Yukiko论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Prod Informat Grp Japan Oncol Business, Chuo Ku, 12-10,Nihonbashi 2 Chome, Tokyo 1038686, Japan Takeda Pharmaceut Co Ltd, Shonan Res Ctr, Pharmaceut Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, JapanMurai, Saomi论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Shonan Res Ctr, Pharmaceut Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Shonan Res Ctr, Pharmaceut Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, JapanHasegawa, Maki论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Shonan Res Ctr, Pharmaceut Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Shonan Res Ctr, Pharmaceut Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, JapanHasegawa, Yuka论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Shonan Res Ctr, Pharmaceut Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Shonan Res Ctr, Pharmaceut Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, JapanYonemori, Kazuko论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Shonan Res Ctr, Pharmaceut Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Shonan Res Ctr, Pharmaceut Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, JapanHata, Akito论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Shonan Res Ctr, Pharmaceut Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Shonan Res Ctr, Pharmaceut Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, JapanAoyama, Kazunobu论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Shonan Res Ctr, Pharmaceut Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Shonan Res Ctr, Pharmaceut Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, JapanCary, Douglas R.论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Shonan Res Ctr, Pharmaceut Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, Japan Peptidream Inc, Tokyo, Japan Takeda Pharmaceut Co Ltd, Shonan Res Ctr, Pharmaceut Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, Japan