Uncommon intramolecular palladium-catalyzed cyclization of indole derivatives

被引：47
|
作者：
Beccalli, EM
Broggini, G
机构：
[1] Univ Milan, Ist Chim Organ, I-20133 Milan, Italy
[2] Univ Insubria, Dipartimento Sci Chim Fis & Matemat, I-22100 Como, Italy
来源：
TETRAHEDRON LETTERS | 2003年 / 44卷 / 09期
关键词：
Pd catalyst; intramolecular cyclization; indoles; carbolinones;
D O I：
10.1016/S0040-4039(03)00116-3
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A novel synthetic strategy based on the intramolecular palladium-catalyzed oxidative cyclization reaction, allows the formation of C-C bond and the synthesis of beta-carbolinones. The reaction has been performed in the presence of catalytic amount of PdCl2(CH3CN)(2) and benzoquinone as a reoxidant. (C) 2003 Elsevier Science Ltd. All rights reserved.
引用
收藏
页码：1919 / 1921
页数：3
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