Discovery of the first known small-molecule inhibitors of heme-regulated eukaryotic initiation factor 2α (HRI) kinase (vol 19, 6548, 2009)

被引：0
|
作者：
Rosen, Mark D. [1 ]
Woods, Craig R. [1 ]
Goldberg, Steven D. [1 ]
Hack, Michael D. [1 ]
Bounds, A. Dawn [1 ]
Yang, Young [1 ]
Wagaman, Pamela C. [1 ]
Phuong, Victor K. [1 ]
Ameriks, Angela P. [1 ]
Barrett, Terrance D. [1 ]
Kanelakis, Kimon C. [1 ]
Chuang, Jui Chang [1 ]
Shankley, Nigel P. [1 ]
Rabinowitz, Michael H. [1 ]
机构：
[1] Johnson & Johnson Pharmaceut Res & Dev LLC, San Diego, CA 92121 USA
来源：
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 2010年 / 20卷 / 12期
关键词：
D O I：
10.1016/j.bmcl.2010.04.107
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
引用
收藏
页码：3834 / 3834
页数：1
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    Rosen, Mark D.
    Woods, Craig R.
    Goldberg, Steven D.
    Hack, Michael D.
    Bounds, A. Dawn
    Yang, Young
    Wagaman, Pamela C.
    Phuong, Victor K.
    Ameriks, Angela P.
    Barrett, Terrance D.
    Kanelakis, Kimon C.
    Chang, Jui
    Shankley, Nigel P.
    Rabinowitz, Michael H.
    [J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009, 19 (23) : 6548 - 6551
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    Suresh, C. G.
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    Kumar, Avinash
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    [J]. JOURNAL OF FLUORESCENCE, 2012, 22 (01) : 431 - 441
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  • [10] NO-induced catalytic activation and heme-induced catalytic suppression of human heme-regulated eukaryotic initiation factor 2α kinase, HRI, associated with lung cancer
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    Yamamura, Ayano
    Igarashi, Jotaro
    Shimizu, Toru
    [J]. NITRIC OXIDE-BIOLOGY AND CHEMISTRY, 2010, 22 : S46 - S47
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