One-Pot Synthesis of 3-Aryltetramic Acids

被引：12

作者：

Mallinger, Aurelie ^{[1
]}

Nadal, Brice ^{[1
]}

Chopin, Nicolas ^{[1
]}

Le Gall, Thierry ^{[1
]}

机构：

[1] CEA Saclay, iBiTecS, Serv Chim Bioorgan & Marquage, F-91191 Gif Sur Yvette, France

来源：

EUROPEAN JOURNAL OF ORGANIC CHEMISTRY | 2010年 / 2010卷 / 06期

关键词：

Tetramic acid; Nitrogen heterocycles; Amides; Ring closure; Dieckinann condensation; Synthetic methods; TETRAMIC ACIDS; INSECTICIDAL ACTIVITY; TETRONIC ACIDS; DERIVATIVES; PRECURSORS;

D O I：

10.1002/ejoc.200901092

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Tetramic acids Substituted in the 3-position by various aryl groups were prepared in one-pot from amino esters and methyl arylacetates, by treatment with potassium tert-butoxide. A tandem process, involving the formation of an amide and a condensation reaction, is likely to occur. N-Unsubstituted tetramic acids were obtained from adducts containing a N-(2,4-dimethoxybenzyl) group.

引用

页码：1142 / 1148

页数：7

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