Pharmacological characterization of GV191869X: A novel, potent and selective CCK-B receptor antagonist

被引:0
|
作者
Corsi, M [1 ]
Oliosi, B [1 ]
van Amsterdam, FTM [1 ]
Antolini, M [1 ]
Melotto, S [1 ]
Gerrard, P [1 ]
Maraia, G [1 ]
Reggiani, A [1 ]
Ursini, A [1 ]
Donati, D [1 ]
Gaviraghi, G [1 ]
Ratti, E [1 ]
Trist, DG [1 ]
机构
[1] GlaxoWellcome SpA, Med Res Ctr, I-37135 Verona, Italy
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
249P
引用
收藏
页码:U144 / U144
页数:1
相关论文
共 50 条
  • [1] THE CHARACTERIZATION IN FUNCTIONAL ASSAYS OF GV-150013 - A NOVEL CCK-B RECEPTOR ANTAGONIST
    CORSI, M
    DALFORNO, G
    VANAMSTERDAM, FTM
    FERIANI, A
    URSINI, A
    RATTI, E
    GAVIRAGHI, G
    TRIST, DG
    BRITISH JOURNAL OF PHARMACOLOGY, 1995, 114 : P91 - P91
  • [2] RECEPTOR-BINDING CHARACTERISTICS OF THE SELECTIVE CCK-B ANTAGONIST GV-150013
    VANAMSTERDAM, FTM
    OLIOSI, B
    CORSI, M
    RATTI, EA
    GAVIRAGHI, G
    TRIST, DG
    BRITISH JOURNAL OF PHARMACOLOGY, 1995, 116 : P240 - P240
  • [3] ANXIOLYTIC ACTIVITY OF GV-150013, A NEW POTENT AND SELECTIVE CHOLECYSTOKININ-B (CCK-B) ANTAGONIST
    REGGIANI, A
    GERRARD, PA
    MARAIA, G
    MELOTTO, S
    RATTI, E
    GAVIRAGHI, G
    TRIST, DG
    BRITISH JOURNAL OF PHARMACOLOGY, 1995, 114 : P92 - P92
  • [4] SYNTHESIS AND CCK-B BINDING AFFINITIES OF CYCLIC ANALOGS OF THE POTENT AND SELECTIVE CCK-B RECEPTOR ANTAGONIST CIL-988
    DIDIER, E
    HORWELL, DC
    PRITCHARD, MC
    TETRAHEDRON, 1992, 48 (39) : 8471 - 8490
  • [5] SYNTHESIS OF A POTENT AND SELECTIVE NONPEPTIDE CCK-B GASTRIN RECEPTOR ANTAGONIST TRITIATED LIGAND
    HILL, D
    HORWELL, DC
    HUNTER, JC
    KNEEN, CO
    PRITCHARD, MC
    SUMANCHAUHAN, N
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1993, 3 (05) : 885 - 888
  • [6] PHARMACOLOGICAL PROFILES OF AG-341R, A NOVEL SELECTIVE GASTRIN CCK-B ANTAGONIST
    BABA, A
    HOSHINO, E
    ONOMA, M
    ESAKI, T
    TAKEDA, K
    GASTROENTEROLOGY, 1995, 108 (04) : A950 - A950
  • [7] RATIONALLY DESIGNED DIPEPTOID ANALOGS OF CCK - ACID MIMICS OF THE POTENT AND SELECTIVE NONPEPTIDE CCK-B RECEPTOR ANTAGONIST CI-988
    DRYSDALE, MJ
    PRITCHARD, MC
    HORWELL, DC
    JOURNAL OF MEDICINAL CHEMISTRY, 1992, 35 (14) : 2573 - 2581
  • [8] THE SYNTHESIS AND CCK RECEPTOR AFFINITIES OF SELECTED CARBOXYLIC-ACID MIMICS OF CL-988 - A POTENT AND SELECTIVE CCK-B ANTAGONIST
    DRYSDALE, MJ
    PRITCHARD, MC
    HORWELL, DC
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1992, 2 (01) : 45 - 48
  • [9] Novel nonpeptide CCK-B antagonists: Design and development of quinazolinone derivatives as potent, selective, and orally active CCK-B antagonists
    Padia, JK
    Field, M
    Hinton, J
    Meecham, K
    Pablo, J
    Pinnock, R
    Roth, BD
    Singh, L
    Suman-Chauhan, N
    Trivedi, BK
    Webdale, L
    JOURNAL OF MEDICINAL CHEMISTRY, 1998, 41 (07) : 1042 - 1049
  • [10] STIMULATION OF FEEDING BY THE SELECTIVE CCK-A RECEPTOR ANTAGONIST DEVAZEPIDE IS NOT MEDIATED THROUGH THE CCK-B RECEPTOR IN RATS
    CASTELLANOS, DA
    REIDELBERGER, RD
    APPETITE, 1994, 23 (03) : 296 - 296