共 25 条
- [1] BT8009, a Bicycle Toxin Conjugate targeting Nectin-4, shows target selectivity, and efficacy in preclinical large and small tumor modelsMOLECULAR CANCER THERAPEUTICS, 2019, 18 (12)Rigby, Michael论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, MA USA Bicycle TX Ltd, Cambridge, MA USABennett, Gavin论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, MA USA Bicycle TX Ltd, Cambridge, MA USAChen, Liuhong论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, MA USA Bicycle TX Ltd, Cambridge, MA USAMudd, Gemma论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, MA USA Bicycle TX Ltd, Cambridge, MA USABeswick, Paul论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, MA USA Bicycle TX Ltd, Cambridge, MA USAHarrison, Helen论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, MA USA Bicycle TX Ltd, Cambridge, MA USAWatcham, Sophie论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, MA USA Bicycle TX Ltd, Cambridge, MA USAAllen, Heather论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, MA USA Bicycle TX Ltd, Cambridge, MA USABrown, Amy论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, MA USA Bicycle TX Ltd, Cambridge, MA USAVan Rietschoten, Katerine论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, MA USA Bicycle TX Ltd, Cambridge, MA USAJeffrey, Philip论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, MA USA Bicycle TX Ltd, Cambridge, MA USAPark, Peter U.论文数: 0 引用数: 0 h-index: 0机构: Orum Therapeut, Cambridge, MA USA Bicycle TX Ltd, Cambridge, MA USAHaines, Eric论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Inc, Lexington, MA USA Bicycle TX Ltd, Cambridge, MA USAKeen, Nicholas论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Inc, Lexington, MA USA Bicycle TX Ltd, Cambridge, MA USALahdenranta, Johanna论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Inc, Lexington, MA USA Bicycle TX Ltd, Cambridge, MA USA
- [2] BT8009; A Nectin-4 Targeting Bicycle Toxin Conjugate for Treatment of Solid TumorsMOLECULAR CANCER THERAPEUTICS, 2022, 21 (12) : 1747 - 1756Rigby, Michael论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, England Bicycle TX Ltd, Blocks A&B,Portway Bldg,Granta Pk, Cambridge CB21 6GP, England Bicycle TX Ltd, Cambridge, EnglandBennett, Gavin论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, England Bicycle TX Ltd, Cambridge, EnglandChen, Liuhong论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, England Bicycle TX Ltd, Cambridge, EnglandMudd, Gemma E.论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, England Bicycle TX Ltd, Cambridge, EnglandHarrison, Helen论文数: 0 引用数: 0 h-index: 0机构: Amphista Therapeut, Cori Bldg, Cambridge, England Bicycle TX Ltd, Cambridge, EnglandBeswick, Paul J.论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, England Bicycle TX Ltd, Cambridge, EnglandVan Rietschoten, Katerine论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, England Bicycle TX Ltd, Cambridge, EnglandWatcham, Sophie M.论文数: 0 引用数: 0 h-index: 0机构: Kymab Ltd, Bennet Bldg,Babraham Res Campus, Cambridge, England Bicycle TX Ltd, Cambridge, EnglandScott, Heather S.论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, England Bicycle TX Ltd, Cambridge, EnglandBrown, Amy N.论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, England Bicycle TX Ltd, Cambridge, EnglandPark, Peter U.论文数: 0 引用数: 0 h-index: 0机构: Orum Therapeut, Cambridge, MA USA Bicycle TX Ltd, Cambridge, EnglandCampbell, Carly论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Inc, Boston, MA USA Bicycle TX Ltd, Cambridge, EnglandHaines, Eric论文数: 0 引用数: 0 h-index: 0机构: Ikena Oncol, Boston, MA USA Bicycle TX Ltd, Cambridge, EnglandLahdenranta, Johanna论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Inc, Boston, MA USA Bicycle TX Ltd, Cambridge, EnglandSkynner, Michael J.论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, England Bicycle TX Ltd, Cambridge, EnglandJeffrey, Phil论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, England Bicycle TX Ltd, Cambridge, EnglandKeen, Nicholas论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Inc, Boston, MA USA Bicycle TX Ltd, Cambridge, EnglandLee, Kevin论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, England Bicycle TX Ltd, Cambridge, England
- [3] Discovery of BT8009: A Nectin-4 Targeting Bicycle Toxin Conjugate for the Treatment of CancerJOURNAL OF MEDICINAL CHEMISTRY, 2022, 65 (21) : 14337 - 14347Mudd, Gemma E.论文数: 0 引用数: 0 h-index: 0机构: BicycleTx Ltd, Cambridge CB22 3AT, England BicycleTx Ltd, Cambridge CB22 3AT, EnglandScott, Heather论文数: 0 引用数: 0 h-index: 0机构: BicycleTx Ltd, Cambridge CB22 3AT, England BicycleTx Ltd, Cambridge CB22 3AT, EnglandChen, Liuhong论文数: 0 引用数: 0 h-index: 0机构: BicycleTx Ltd, Cambridge CB22 3AT, England BicycleTx Ltd, Cambridge CB22 3AT, Englandvan Rietschoten, Katerine论文数: 0 引用数: 0 h-index: 0机构: BicycleTx Ltd, Cambridge CB22 3AT, England BicycleTx Ltd, Cambridge CB22 3AT, EnglandIvanova-Berndt, Gabriela论文数: 0 引用数: 0 h-index: 0机构: BicycleTx Ltd, Cambridge CB22 3AT, England BicycleTx Ltd, Cambridge CB22 3AT, EnglandDzionek, Katarzyna论文数: 0 引用数: 0 h-index: 0机构: BicycleTx Ltd, Cambridge CB22 3AT, England BicycleTx Ltd, Cambridge CB22 3AT, EnglandBrown, Amy论文数: 0 引用数: 0 h-index: 0机构: BicycleTx Ltd, Cambridge CB22 3AT, England BicycleTx Ltd, Cambridge CB22 3AT, EnglandWatcham, Sophie论文数: 0 引用数: 0 h-index: 0机构: BicycleTx Ltd, Cambridge CB22 3AT, England BicycleTx Ltd, Cambridge CB22 3AT, EnglandWhite, Lewi论文数: 0 引用数: 0 h-index: 0机构: BicycleTx Ltd, Cambridge CB22 3AT, England BicycleTx Ltd, Cambridge CB22 3AT, EnglandPark, Peter U.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Inc, Lexington, MA 02421 USA BicycleTx Ltd, Cambridge CB22 3AT, EnglandJeffrey, Phil论文数: 0 引用数: 0 h-index: 0机构: BicycleTx Ltd, Cambridge CB22 3AT, England BicycleTx Ltd, Cambridge CB22 3AT, EnglandRigby, Mike论文数: 0 引用数: 0 h-index: 0机构: BicycleTx Ltd, Cambridge CB22 3AT, England BicycleTx Ltd, Cambridge CB22 3AT, EnglandBeswick, Paul论文数: 0 引用数: 0 h-index: 0机构: BicycleTx Ltd, Cambridge CB22 3AT, England BicycleTx Ltd, Cambridge CB22 3AT, England
- [4] A multi tumor survey of Nectin-4 expression to guide BT8009 indication selection.CANCER RESEARCH, 2021, 81 (13)Campbell, Carly T.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Lexington, MA USA Bicycle Therapeut, Lexington, MA USASmale, Robert论文数: 0 引用数: 0 h-index: 0机构: NeoGenomics, Aliso Viejo, CA USA Bicycle Therapeut, Lexington, MA USARigby, Michael论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Cambridge, England Bicycle Therapeut, Lexington, MA USAWatson, Shawn论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Lexington, MA USA Bicycle Therapeut, Lexington, MA USADickson, Amy论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Lexington, MA USA Bicycle Therapeut, Lexington, MA USAGelb, Tara论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Lexington, MA USA Bicycle Therapeut, Lexington, MA USACohen, Heather论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Lexington, MA USA Bicycle Therapeut, Lexington, MA USALee, Pierre论文数: 0 引用数: 0 h-index: 0机构: Abcam, Burlingame, CA USA Bicycle Therapeut, Lexington, MA USARagheb, Josette William论文数: 0 引用数: 0 h-index: 0机构: NeoGenomics, Aliso Viejo, CA USA Bicycle Therapeut, Lexington, MA USABlakemore, Stephen J.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Lexington, MA USA Bicycle Therapeut, Lexington, MA USA
- [5] Association of combined phase I/II study of a novel bicyclic peptide and MMAE conjugate BT8009 in patients with advanced malignancies with Nectin-4 expression.JOURNAL OF CLINICAL ONCOLOGY, 2021, 39 (15)McKean, Meredith论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USAFalchook, Gerald Steven论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USABendell, Johanna C.论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USABashir, Babar论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USAPalmisiano, Neil论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USAWatson, Roshawn论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USAMcKenna, Mary-Anne论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USACampbell, Carly论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USASmethurst, Dominic Paul论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USAJeffrey, Phil论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USAKirui, Julius论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USAArkenau, Hendrik-Tobias论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USAFontana, Elisa论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USA
- [6] Effects of Nectin-4 targeted Bicycle Toxin Conjugate, zelenectide pevedotin (BT8009), and enfortumab vedotin on a human corneal tissue modelEUROPEAN JOURNAL OF CANCER, 2024, 211 : S115 - S115Kristensson, J.论文数: 0 引用数: 0 h-index: 0机构: BicycleTx, Biol, Cambridge, England BicycleTx, Biol, Cambridge, EnglandCampbell, C.论文数: 0 引用数: 0 h-index: 0机构: BicycleTx, Translat, Boston, MA USA BicycleTx, Biol, Cambridge, EnglandLudbrook, S.论文数: 0 引用数: 0 h-index: 0机构: BicycleTx, Biol, Cambridge, England BicycleTx, Biol, Cambridge, EnglandHirschberg, S.论文数: 0 引用数: 0 h-index: 0机构: BicycleTx, Clin, Cambridge, England BicycleTx, Biol, Cambridge, EnglandRigby, M.论文数: 0 引用数: 0 h-index: 0机构: BicycleTx, Biol, Cambridge, England BicycleTx, Biol, Cambridge, England
- [7] The Tumor-Associated Marker, PVRL4 (Nectin-4), Is the Epithelial Receptor for MorbillivirusesVIRUSES-BASEL, 2014, 6 (06): : 2268 - 2286Delpeut, Sebastien论文数: 0 引用数: 0 h-index: 0机构: Dalhousie Univ, Dept Microbiol & Immunol, Halifax, NS B3H 1X5, Canada Canadian Ctr Vaccinol, IWK Hlth Ctr, Halifax, NS B3H 1X5, Canada Dalhousie Univ, Dept Microbiol & Immunol, Halifax, NS B3H 1X5, CanadaNoyce, Ryan S.论文数: 0 引用数: 0 h-index: 0机构: Dalhousie Univ, Dept Microbiol & Immunol, Halifax, NS B3H 1X5, Canada Canadian Ctr Vaccinol, IWK Hlth Ctr, Halifax, NS B3H 1X5, Canada Dalhousie Univ, Dept Microbiol & Immunol, Halifax, NS B3H 1X5, CanadaRichardson, Christopher D.论文数: 0 引用数: 0 h-index: 0机构: Dalhousie Univ, Dept Microbiol & Immunol, Halifax, NS B3H 1X5, Canada Canadian Ctr Vaccinol, IWK Hlth Ctr, Halifax, NS B3H 1X5, Canada Dalhousie Univ, Dept Pediat, Halifax, NS B3K 6R8, Canada Dalhousie Univ, Dept Microbiol & Immunol, Halifax, NS B3H 1X5, Canada
- [8] BT8009-100: A phase I/II study of novel bicyclic peptide and MMAE conjugate BT8009 in patients (pts) with advanced malignancies associated with nectin-4 expression, including urothelial cancer (UC).JOURNAL OF CLINICAL ONCOLOGY, 2023, 41Baldini, Capucine论文数: 0 引用数: 0 h-index: 0机构: Gustave Roussy, Drug Dev Dept DITEP, Villejuif, FranceGoldschmidt, Vincent论文数: 0 引用数: 0 h-index: 0机构: Gustave Roussy, Drug Dev Dept DITEP, Villejuif, FranceBrana, Irene论文数: 0 引用数: 0 h-index: 0机构: Gustave Roussy, Drug Dev Dept DITEP, Villejuif, FranceDoger, Bernard论文数: 0 引用数: 0 h-index: 0机构: Gustave Roussy, Drug Dev Dept DITEP, Villejuif, FranceItaliano, Antoine论文数: 0 引用数: 0 h-index: 0机构: Gustave Roussy, Drug Dev Dept DITEP, Villejuif, FranceCousin, Sophie论文数: 0 引用数: 0 h-index: 0机构: Gustave Roussy, Drug Dev Dept DITEP, Villejuif, FranceFalchook, Gerald Steven论文数: 0 引用数: 0 h-index: 0机构: Gustave Roussy, Drug Dev Dept DITEP, Villejuif, FranceNecchi, Andrea论文数: 0 引用数: 0 h-index: 0机构: Gustave Roussy, Drug Dev Dept DITEP, Villejuif, FranceReig, Oscar论文数: 0 引用数: 0 h-index: 0机构: Gustave Roussy, Drug Dev Dept DITEP, Villejuif, FranceCarter, Louise论文数: 0 引用数: 0 h-index: 0机构: Gustave Roussy, Drug Dev Dept DITEP, Villejuif, FranceFontana, Elisa论文数: 0 引用数: 0 h-index: 0机构: Gustave Roussy, Drug Dev Dept DITEP, Villejuif, FranceVerlingue, Loic论文数: 0 引用数: 0 h-index: 0机构: Gustave Roussy, Drug Dev Dept DITEP, Villejuif, FranceHazard, Sebastien论文数: 0 引用数: 0 h-index: 0机构: Gustave Roussy, Drug Dev Dept DITEP, Villejuif, FranceDickson, Amy论文数: 0 引用数: 0 h-index: 0机构: Gustave Roussy, Drug Dev Dept DITEP, Villejuif, FranceXu, Cong论文数: 0 引用数: 0 h-index: 0机构: Gustave Roussy, Drug Dev Dept DITEP, Villejuif, FranceXu, Hongmei论文数: 0 引用数: 0 h-index: 0机构: Gustave Roussy, Drug Dev Dept DITEP, Villejuif, FranceSharma, Rajiv论文数: 0 引用数: 0 h-index: 0机构: Gustave Roussy, Drug Dev Dept DITEP, Villejuif, FranceSmethurst, Dominic论文数: 0 引用数: 0 h-index: 0机构: Gustave Roussy, Drug Dev Dept DITEP, Villejuif, FranceMcKean, Meredith论文数: 0 引用数: 0 h-index: 0机构: Gustave Roussy, Drug Dev Dept DITEP, Villejuif, France
- [9] BT8009-100 phase I/II study of novel bi-cyclic peptide and MMAE conjugate BT8009 in patients with advanced malignancies associated with nectin-4 expressionCANCER RESEARCH, 2022, 82 (12)McKean, Meredith论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst Tennessee Oncol, Nashville, TN USA Sarah Cannon Res Inst Tennessee Oncol, Nashville, TN USABaldini, Capucine论文数: 0 引用数: 0 h-index: 0机构: Inst Gustave Roussy, Villejuif, France Sarah Cannon Res Inst Tennessee Oncol, Nashville, TN USAVerlingue, Loic论文数: 0 引用数: 0 h-index: 0机构: Inst Gustave Roussy, Villejuif, France Sarah Cannon Res Inst Tennessee Oncol, Nashville, TN USADoger, Bernard论文数: 0 引用数: 0 h-index: 0机构: START Madrid FJD, Madrid, Spain Sarah Cannon Res Inst Tennessee Oncol, Nashville, TN USAFalchook, Gerald论文数: 0 引用数: 0 h-index: 0机构: HealthONE, Sarah Cannon Res Inst, Denver, CO USA Sarah Cannon Res Inst Tennessee Oncol, Nashville, TN USAItaliano, Antoine论文数: 0 引用数: 0 h-index: 0机构: Inst Bergonie, Bordeaux, France Sarah Cannon Res Inst Tennessee Oncol, Nashville, TN USALostes, Julia论文数: 0 引用数: 0 h-index: 0机构: Vall dHebron Inst Oncol, Barcelona, Spain Sarah Cannon Res Inst Tennessee Oncol, Nashville, TN USAReig, Oscar论文数: 0 引用数: 0 h-index: 0机构: Hosp Clin Barcelona, Barcelona, Spain Sarah Cannon Res Inst Tennessee Oncol, Nashville, TN USAWatson, Roshawn论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Lexington, MA USA Sarah Cannon Res Inst Tennessee Oncol, Nashville, TN USAHazard, Sebastien论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Lexington, MA USA Sarah Cannon Res Inst Tennessee Oncol, Nashville, TN USASmethurst, Dominic论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Cambridge, England Sarah Cannon Res Inst Tennessee Oncol, Nashville, TN USAFulci, Giulia论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Lexington, MA USA Sarah Cannon Res Inst Tennessee Oncol, Nashville, TN USAXu, Hongmei论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Lexington, MA USA Sarah Cannon Res Inst Tennessee Oncol, Nashville, TN USAJeffery, Phil论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Lexington, MA USA Sarah Cannon Res Inst Tennessee Oncol, Nashville, TN USALee, Kevin论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Cambridge, England Sarah Cannon Res Inst Tennessee Oncol, Nashville, TN USABrana, Irene论文数: 0 引用数: 0 h-index: 0机构: Vall dHebron Inst Oncol, Barcelona, Spain Sarah Cannon Res Inst Tennessee Oncol, Nashville, TN USACousin, Sophie论文数: 0 引用数: 0 h-index: 0机构: Inst Bergonie, Bordeaux, France Sarah Cannon Res Inst Tennessee Oncol, Nashville, TN USAFontana, Elisa论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst UK, London, England Sarah Cannon Res Inst Tennessee Oncol, Nashville, TN USAArkenau, Hendrik-Tobias论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst UK, London, England Sarah Cannon Res Inst Tennessee Oncol, Nashville, TN USA
- [10] Molecular-based enrichment strategy for Nectin-4 targeted Bicycle toxin conjugate BT8009.CANCER RESEARCH, 2021, 81 (13)Gelb, Tara论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Lexington, MA USA Bicycle Therapeut, Lexington, MA USASantos, Sean论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Lexington, MA USA Bicycle Therapeut, Lexington, MA USADickson, Amy论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Lexington, MA USA Bicycle Therapeut, Lexington, MA USACampbell, Carly论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Lexington, MA USA Bicycle Therapeut, Lexington, MA USARigby, Mike论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Cambridge, England Bicycle Therapeut, Lexington, MA USAMckenzie, Andrew J.论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USA Bicycle Therapeut, Lexington, MA USARozelle, Dan论文数: 0 引用数: 0 h-index: 0机构: Rancho Bio Sci, San Diego, CA USA Bicycle Therapeut, Lexington, MA USABlakemore, Stephen J.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Lexington, MA USA Bicycle Therapeut, Lexington, MA USA