共 9 条
- [1] Discovery of DWP213388, a Potent ITK and BTK Selective Dual Inhibitor with Excellent Efficacy and Safety, for Treating GvhdBLOOD, 2019, 134Eom, Deokki论文数: 0 引用数: 0 h-index: 0机构: Daewoong Life Sci Res Inst, Yongin, South Korea Daewoong Life Sci Res Inst, Yongin, South KoreaJung, Jae Hun论文数: 0 引用数: 0 h-index: 0机构: Daewoong Life Sci Res Inst, Yongin, South Korea Daewoong Life Sci Res Inst, Yongin, South KoreaKim, Eun Kyung论文数: 0 引用数: 0 h-index: 0机构: Daewoong Life Sci Res Inst, Yongin, South Korea Daewoong Life Sci Res Inst, Yongin, South KoreaKim, Wolyoung论文数: 0 引用数: 0 h-index: 0机构: Daewoong Life Sci Res Inst, Yongin, South Korea Daewoong Life Sci Res Inst, Yongin, South KoreaLi, Qingri论文数: 0 引用数: 0 h-index: 0机构: Daewoong Life Sci Res Inst, Yongin, South Korea Daewoong Life Sci Res Inst, Yongin, South KoreaJung, Jaehyun论文数: 0 引用数: 0 h-index: 0机构: Daewoong Life Sci Res Inst, Yongin, South Korea Daewoong Life Sci Res Inst, Yongin, South KoreaIm, Sohee论文数: 0 引用数: 0 h-index: 0机构: Daewoong Life Sci Res Inst, Yongin, South Korea Daewoong Life Sci Res Inst, Yongin, South KoreaShin, Yong Dae论文数: 0 引用数: 0 h-index: 0机构: Daewoong Life Sci Res Inst, Yongin, South Korea Daewoong Life Sci Res Inst, Yongin, South KoreaHyun, Hyaejung论文数: 0 引用数: 0 h-index: 0机构: Daewoong Life Sci Res Inst, Yongin, South Korea Daewoong Life Sci Res Inst, Yongin, South KoreaPark, Joon Seok论文数: 0 引用数: 0 h-index: 0机构: Daewoong Life Sci Res Inst, Yongin, South Korea Daewoong Life Sci Res Inst, Yongin, South Korea
- [2] Discovery of DWP212525, a Potent JAK3 and BTK Dual Target Inhibitor for the Treatment of Autoimmune DiseasesARTHRITIS & RHEUMATOLOGY, 2019, 71Shin, Yong Dae论文数: 0 引用数: 0 h-index: 0机构: Daewoong Life Sci Res Inst, Yongin, South Korea Daewoong Life Sci Res Inst, Yongin, South KoreaJung, Jae-Hun论文数: 0 引用数: 0 h-index: 0机构: Daewoong Life Sci Res Inst, Yongin, South Korea Daewoong Life Sci Res Inst, Yongin, South KoreaKim, Eun Kyung论文数: 0 引用数: 0 h-index: 0机构: Daewoong Life Sci Res Inst, Yongin, South Korea Daewoong Life Sci Res Inst, Yongin, South KoreaIm, Sohee论文数: 0 引用数: 0 h-index: 0机构: Daewoong Life Sci Res Inst, Yongin, South Korea Daewoong Life Sci Res Inst, Yongin, South KoreaJun, Sunah论文数: 0 引用数: 0 h-index: 0机构: Daewoong Life Sci Res Inst, Yongin, South Korea Daewoong Life Sci Res Inst, Yongin, South KoreaKim, NamYoun论文数: 0 引用数: 0 h-index: 0机构: Daewoong Life Sci Res Inst, Yongin, South Korea Daewoong Life Sci Res Inst, Yongin, South KoreaJeong, SeungHwarn论文数: 0 引用数: 0 h-index: 0机构: Daewoong Life Sci Res Inst, Yongin, South Korea Daewoong Life Sci Res Inst, Yongin, South KoreaHyun, Hyaejung论文数: 0 引用数: 0 h-index: 0机构: Daewoong Life Sci Res Inst, Yongin, South Korea Daewoong Life Sci Res Inst, Yongin, South KoreaPark, Joon Seok论文数: 0 引用数: 0 h-index: 0机构: Daewoong Life Sci Res Inst, Yongin, South Korea Daewoong Life Sci Res Inst, Yongin, South Korea
- [3] Discovery of M2951: A selective, covalent inhibitor of BTK for the treatment of autoimmune diseasesABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2017, 254Goutopoulos, Andreas论文数: 0 引用数: 0 h-index: 0机构: EMD Serono, Boston, MA USA EMD Serono, Boston, MA USA
- [4] Discovery of Evobrutinib: An Oral, Potent, and Highly Selective, Covalent Bruton's Tyrosine Kinase (BTK) Inhibitor for the Treatment of Immunological DiseasesJOURNAL OF MEDICINAL CHEMISTRY, 2019, 62 (17) : 7643 - 7655Caldwell, Richard D.论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USAQiu, Hui论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USAAskew, Ben C.论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA Breakthrough Chem Advisors, 266 Arrowhead Rd, Marshfield, MA 02050 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USABender, Andrew T.论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USABrugger, Nadia论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USACamps, Montserrat论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA 45 Chemin Cazers Bas, F-81100 Castres, France EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USADhanabal, Mohanraj论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USADutt, Vikram论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USAEichhorn, Thomas论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USAGardberg, Anna S.论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA Constellat Pharmaceut, 215 First St,Suite 200, Cambridge, MA 02142 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USAGoutopoulos, Andreas论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USAGrenningloh, Roland论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USAHead, Jared论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USAHealey, Brian论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA UMass Boston, Venture Dev Ctr, 100 Morrissey Blvd, Boston, MA 02125 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USAHodous, Brian L.论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA Accent Therapeut, 65 Hayden Ave, Cambridge, MA 02421 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USAHuck, Bayard R.论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USAJohnson, Theresa L.论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USAJones, Christopher论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USAJones, Reinaldo C.论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USAMochalkin, Igor论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA Vertex Pharmaceut, 3215 Merryfield Row, San Diego, CA 92121 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USAMorandi, Federica论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA Hoffmann La Roche AG, Roche Innovat Ctr Basel, Pharma Res & Early Dev, Basel, Switzerland EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USANgan Nguyen论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA Adv Instruments LLC, Two Technol Way, Norwood, MA 02062 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USAMeyring, Michael论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA Nuvisan GmbH, Site Grafing,Feld 32, D-85567 Grafing, Germany EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USAPotnick, Justin R.论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USASantos, Dusica Cvetinovic论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USASchmidt, Ralf论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USASherer, Brian论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USAShutes, Adam论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA Boston Cheese Cellar, 8 Birch St, Roslindale, MA 02131 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USAUrbahns, Klaus论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USAFollis, Ariele Viacava论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USAWegener, Ansgar A.论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USAZimmerli, Simone C.论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USALiu-Bujalski, Lesley论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst Inc, 45 A Middlesex Turnpike, Billerica, MA 01821 USA
- [5] Discovery of VX-509 (Decernotinib): A Potent and Selective Janus Kinase 3 Inhibitor for the Treatment of Autoimmune DiseasesJOURNAL OF MEDICINAL CHEMISTRY, 2015, 58 (18) : 7195 - 7216Farmer, Luc J.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Canada Inc, Laval, PQ H7V 4A7, Canada Vertex Pharmaceut Inc, Boston, MA 02210 USALedeboer, Mark W.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAHoock, Thomas论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAArnost, Michael J.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USABethiel, Randy S.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USABennani, Youssef L.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Canada Inc, Laval, PQ H7V 4A7, Canada Vertex Pharmaceut Inc, Boston, MA 02210 USABlack, James J.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USABrummel, Christopher L.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAChakilam, Ananthsrinivas论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USADorsch, Warren A.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAFan, Bin论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USACochran, John E.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAHalas, Summer论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAHarrington, Edmund M.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAHogan, James K.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAHowe, David论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAHuang, Hui论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAJacobs, Dylan H.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USALaitinen, Leena M.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USALiao, Shengkai论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAMahajan, Sudipta论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAMarone, Valerie论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAMartinez-Botella, Gabriel论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAMcCarthy, Pamela论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAMessersmith, David论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USANamchuk, Mark论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAOh, Luke论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAPenney, Marina S.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAPierce, Albert C.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USARaybuck, Scott A.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USARugg, Arthur论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USASalituro, Francesco G.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USASaxena, Kumkum论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAShannon, Dean论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAShlyakter, Dina论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USASwenson, Lora论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USATian, Shi-Kai论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USATown, Christopher论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAWang, Jian论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAWang, Tiansheng论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAWannamaker, M. Woods论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAWinquist, Raymond J.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAZuccola, Harmon J.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USA
- [6] Discovery of Clinical Candidate GLPG3970: A Potent and Selective Dual SIK2/SIK3 Inhibitor for the Treatment of Autoimmune and Inflammatory DiseasesJOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (07) : 5233 - 5258Peixoto, Christophe论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceJoncour, Agnes论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceTemal-Laib, Taoues论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceTirera, Amynata论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceDos Santos, Aurelie论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceJary, Helene论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceBucher, Denis论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceLaenen, Wendy论文数: 0 引用数: 0 h-index: 0机构: Galapagos NV, B-2800 Mechelen, Belgium Galapagos SASU, F-93230 Romainville, FranceFernandes, Anna Pereira论文数: 0 引用数: 0 h-index: 0机构: Galapagos NV, B-2800 Mechelen, Belgium Galapagos SASU, F-93230 Romainville, FranceLavazais, Stephanie论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceDelachaume, Carole论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceMerciris, Didier论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceSaccomani, Corinne论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceDrennan, Michael论文数: 0 引用数: 0 h-index: 0机构: Galapagos NV, B-2800 Mechelen, Belgium Galapagos SASU, F-93230 Romainville, FranceLopez-Ramos, Miriam论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceWakselman, Emanuelle论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceDupont, Sonia论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceBorgonovi, Monica论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceMagadan, Carlos Roca论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceMonjardet, Alain论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceBrys, Reginald论文数: 0 引用数: 0 h-index: 0机构: Galapagos NV, B-2800 Mechelen, Belgium Galapagos SASU, F-93230 Romainville, FranceDe Vos, Steve论文数: 0 引用数: 0 h-index: 0机构: Galapagos NV, B-2800 Mechelen, Belgium Galapagos SASU, F-93230 Romainville, FranceAndrews, Martin论文数: 0 引用数: 0 h-index: 0机构: Galapagos NV, B-2800 Mechelen, Belgium Galapagos SASU, F-93230 Romainville, FranceJimenez, Juan-Miguel论文数: 0 引用数: 0 h-index: 0机构: Galapagos NV, B-2800 Mechelen, Belgium Galapagos SASU, F-93230 Romainville, FranceAmantini, David论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, FranceDesroy, Nicolas论文数: 0 引用数: 0 h-index: 0机构: Galapagos SASU, F-93230 Romainville, France Galapagos SASU, F-93230 Romainville, France
- [7] Discovery of the First-in-Class Dual-Target ROCK/HDAC Inhibitor with Potent Antitumor Efficacy in Vivo That Trigger Antitumor ImmunityJOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (22) : 20619 - 20638Mao, Churu论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Inst Marine Biol & Pharmacol, Ocean Coll, Zhoushan 316021, Peoples R China Zhejiang Univ, Inst Marine Biol & Pharmacol, Ocean Coll, Zhoushan 316021, Peoples R ChinaFang, Jiebin论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Hainan Inst, Sanya 572025, Peoples R China Zhejiang Univ, Inst Marine Biol & Pharmacol, Ocean Coll, Zhoushan 316021, Peoples R ChinaZou, Shijie论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Inst Marine Biol & Pharmacol, Ocean Coll, Zhoushan 316021, Peoples R China Zhejiang Univ, Inst Marine Biol & Pharmacol, Ocean Coll, Zhoushan 316021, Peoples R ChinaHuang, Yun论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Inst Marine Biol & Pharmacol, Ocean Coll, Zhoushan 316021, Peoples R China Zhejiang Univ, Inst Marine Biol & Pharmacol, Ocean Coll, Zhoushan 316021, Peoples R ChinaChen, Xiaoming论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Inst Marine Biol & Pharmacol, Ocean Coll, Zhoushan 316021, Peoples R China Zhejiang Univ, Inst Marine Biol & Pharmacol, Ocean Coll, Zhoushan 316021, Peoples R ChinaDing, Xia论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Inst Marine Biol & Pharmacol, Ocean Coll, Zhoushan 316021, Peoples R China Zhejiang Univ, Inst Marine Biol & Pharmacol, Ocean Coll, Zhoushan 316021, Peoples R ChinaFang, Zhangyun论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Inst Marine Biol & Pharmacol, Ocean Coll, Zhoushan 316021, Peoples R China Zhejiang Univ, Inst Marine Biol & Pharmacol, Ocean Coll, Zhoushan 316021, Peoples R ChinaZhang, Ningjing论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Inst Marine Biol & Pharmacol, Ocean Coll, Zhoushan 316021, Peoples R China Zhejiang Univ, Inst Marine Biol & Pharmacol, Ocean Coll, Zhoushan 316021, Peoples R ChinaLou, Yijie论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Chinese Med Univ, Affiliated Hosp Zhejiang Chinese Med 1, Key Lab Digest Pathophysiol Zhejiang Prov, Hangzhou 310053, Peoples R China Zhejiang Univ, Inst Marine Biol & Pharmacol, Ocean Coll, Zhoushan 316021, Peoples R ChinaChen, Zhe论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Chinese Med Univ, Affiliated Hosp Zhejiang Chinese Med 1, Key Lab Digest Pathophysiol Zhejiang Prov, Hangzhou 310053, Peoples R China Zhejiang Univ, Inst Marine Biol & Pharmacol, Ocean Coll, Zhoushan 316021, Peoples R ChinaDing, Wanjing论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Inst Marine Biol & Pharmacol, Ocean Coll, Zhoushan 316021, Peoples R China Zhejiang Univ, Hainan Inst, Sanya 572025, Peoples R China Zhejiang Univ, Inst Marine Biol & Pharmacol, Ocean Coll, Zhoushan 316021, Peoples R ChinaMa, Zhongjun论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Inst Marine Biol & Pharmacol, Ocean Coll, Zhoushan 316021, Peoples R China Zhejiang Univ, Hainan Inst, Sanya 572025, Peoples R China Zhejiang Univ, Inst Marine Biol & Pharmacol, Ocean Coll, Zhoushan 316021, Peoples R China
- [8] Discovery of CP-690,550: A Potent and Selective Janus Kinase (JAK) Inhibitor for the Treatment of Autoimmune Diseases and Organ Transplant RejectionJOURNAL OF MEDICINAL CHEMISTRY, 2010, 53 (24) : 8468 - 8484Flanagan, Mark E.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USABlumenkopf, Todd A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, New London, CT 06320 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USABrissette, William H.论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, New Haven, CT 06520 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USABrown, Matthew F.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USACasavant, Jeffrey M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAShang-Poa, Chang论文数: 0 引用数: 0 h-index: 0机构: Univ Connecticut, Dept Stat, Storrs, CT 06269 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USADoty, Jonathan L.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAElliott, Eileen A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAFisher, Michael B.论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Ridgefield, CT 06877 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAHines, Michael论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAKent, Craig论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAKudlacz, Elizabeth M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, New London, CT 06320 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USALillie, Brett M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAMagnuson, Kelly S.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, New London, CT 06320 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAMcCurdy, Sandra P.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAMunchhof, Michael J.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAPerry, Bret D.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USASawyer, Perry S.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAStrelevitz, Timothy J.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USASubramanyam, Chakrapani论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USASun, Jianmin论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAWhipple, David A.论文数: 0 引用数: 0 h-index: 0机构: Univ Kansas, Del Shankel Struct Biol Ctr, Lawrence, KS 66047 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USAChangelian, Paul S.论文数: 0 引用数: 0 h-index: 0机构: Lycera Corp, Plymouth, MI 48170 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA
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