8-Halo-1,3-dimethyl-7-(thiiran-2-ylmethyl)-3,7-dihydro-1H-purine-2,6-diones, Model Thiiranes for Investigating Reactions with Nucleophiles

被引：1
|
作者：
Khaliullin, F. A. [1 ]
Klen, E. E. [1 ]
机构：
[1] Bashkir State Med Univ, Ufa 450000, Russia
来源：
RUSSIAN JOURNAL OF ORGANIC CHEMISTRY | 2009年 / 45卷 / 11期
关键词：
Benzimidazole; Ethyl Cyanoacetate; Methylsulfanyl; Sodium Methylate; Thiiranes;
D O I：
10.1134/S1070428009110207
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
For the study of thiirane reactions with nucleophiles 8-halo-1,3-dimethyl-7-(thiiran-2-ylmethyl)-3,7dihydro-1H-purine-2,6-diones that did not form polymeric products through intramolecular heterocyclization into dihydrothiazolopurine derivatives were selected as model compounds. The possibility to employ the model thiiranes for the study of reactions with various nucleophiles was demonstrated.
引用
收藏
页码：1697 / 1699
页数：3
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