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- [1] Bcl-2/Bcl-xl inhibitor APG-1252-M1 is a promising therapeutic strategy for gastric carcinomaCANCER MEDICINE, 2020, 9 (12): : 4197 - 4206Yi, Hanjie论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Dept Expt Res, State Key Lab Oncol South China,Canc Ctr, 651 Dongfeng Rd East, Guangzhou 510060, Peoples R China Nanchang Univ, Affiliated Hosp 2, Dept Med Oncol, Nanchang, Jiangxi, Peoples R China Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Dept Expt Res, State Key Lab Oncol South China,Canc Ctr, 651 Dongfeng Rd East, Guangzhou 510060, Peoples R ChinaQiu, Miao-Zhen论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Dept Med Oncol, State Key Lab Oncol South China,Canc Ctr, 651 Dongfeng Rd East, Guangzhou 510060, Peoples R China Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Dept Expt Res, State Key Lab Oncol South China,Canc Ctr, 651 Dongfeng Rd East, Guangzhou 510060, Peoples R ChinaYuan, Luping论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Dept Expt Res, State Key Lab Oncol South China,Canc Ctr, 651 Dongfeng Rd East, Guangzhou 510060, Peoples R China Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Dept Expt Res, State Key Lab Oncol South China,Canc Ctr, 651 Dongfeng Rd East, Guangzhou 510060, Peoples R ChinaLuo, Qiuyun论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Dept Expt Res, State Key Lab Oncol South China,Canc Ctr, 651 Dongfeng Rd East, Guangzhou 510060, Peoples R China Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Dept Expt Res, State Key Lab Oncol South China,Canc Ctr, 651 Dongfeng Rd East, Guangzhou 510060, Peoples R ChinaPan, Wentao论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Dept Expt Res, State Key Lab Oncol South China,Canc Ctr, 651 Dongfeng Rd East, Guangzhou 510060, Peoples R China Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Dept Expt Res, State Key Lab Oncol South China,Canc Ctr, 651 Dongfeng Rd East, Guangzhou 510060, Peoples R ChinaZhou, Suna论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Dept Expt Res, State Key Lab Oncol South China,Canc Ctr, 651 Dongfeng Rd East, Guangzhou 510060, Peoples R China Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Dept Expt Res, State Key Lab Oncol South China,Canc Ctr, 651 Dongfeng Rd East, Guangzhou 510060, Peoples R ChinaZhang, Lin论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Dept Clin Lab Med, Canc Ctr, Guangzhou, Peoples R China Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Dept Expt Res, State Key Lab Oncol South China,Canc Ctr, 651 Dongfeng Rd East, Guangzhou 510060, Peoples R ChinaYan, Xianglei论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Dept Expt Res, State Key Lab Oncol South China,Canc Ctr, 651 Dongfeng Rd East, Guangzhou 510060, Peoples R China Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Dept Expt Res, State Key Lab Oncol South China,Canc Ctr, 651 Dongfeng Rd East, Guangzhou 510060, Peoples R ChinaYang, Da-Jun论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Dept Expt Res, State Key Lab Oncol South China,Canc Ctr, 651 Dongfeng Rd East, Guangzhou 510060, Peoples R China Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Dept Expt Res, State Key Lab Oncol South China,Canc Ctr, 651 Dongfeng Rd East, Guangzhou 510060, Peoples R China
- [2] Therapeutic potential of the novel Bcl-2/Bcl-XL dual inhibitor, APG1252, alone or in combination against non-small cell lung cancerMOLECULAR CARCINOGENESIS, 2022, 61 (11) : 1031 - 1042Qian, Luxi论文数: 0 引用数: 0 h-index: 0机构: Nanjing Med Univ, Dept Radiat Oncol, Jiangsu Canc Hosp, Jiangsu Inst Canc Res, Nanjing, Jiangsu, Peoples R China Nanjing Med Univ, Affiliated Canc Hosp, Nanjing, Jiangsu, Peoples R China Emory Univ, Sch Med, Dept Hematol & Med Oncol, 1365-C Clifton Rd,C3088, Atlanta, GA 30322 USA Winship Canc Inst, 1365-C Clifton Rd,C3088, Atlanta, GA 30322 USA Nanjing Med Univ, Dept Radiat Oncol, Jiangsu Canc Hosp, Jiangsu Inst Canc Res, Nanjing, Jiangsu, Peoples R ChinaVallega, Karin A.论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Sch Med, Dept Hematol & Med Oncol, 1365-C Clifton Rd,C3088, Atlanta, GA 30322 USA Winship Canc Inst, 1365-C Clifton Rd,C3088, Atlanta, GA 30322 USA Nanjing Med Univ, Dept Radiat Oncol, Jiangsu Canc Hosp, Jiangsu Inst Canc Res, Nanjing, Jiangsu, Peoples R ChinaYao, Weilong论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Sch Med, Dept Hematol & Med Oncol, 1365-C Clifton Rd,C3088, Atlanta, GA 30322 USA Winship Canc Inst, 1365-C Clifton Rd,C3088, Atlanta, GA 30322 USA Capital Med Univ, Beijing Friendship Hosp, Dept Gastroenterol, Beijing, Peoples R China Nanjing Med Univ, Dept Radiat Oncol, Jiangsu Canc Hosp, Jiangsu Inst Canc Res, Nanjing, Jiangsu, Peoples R ChinaWang, Dongsheng论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Sch Med, Dept Hematol & Med Oncol, 1365-C Clifton Rd,C3088, Atlanta, GA 30322 USA Winship Canc Inst, 1365-C Clifton Rd,C3088, Atlanta, GA 30322 USA Nanjing Med Univ, Dept Radiat Oncol, Jiangsu Canc Hosp, Jiangsu Inst Canc Res, Nanjing, Jiangsu, Peoples R ChinaZhai, Yifan论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma Suzhou Co Ltd, Suzhou, Jiangsu, Peoples R China Nanjing Med Univ, Dept Radiat Oncol, Jiangsu Canc Hosp, Jiangsu Inst Canc Res, Nanjing, Jiangsu, Peoples R ChinaHe, Xia论文数: 0 引用数: 0 h-index: 0机构: Nanjing Med Univ, Dept Radiat Oncol, Jiangsu Canc Hosp, Jiangsu Inst Canc Res, Nanjing, Jiangsu, Peoples R China Nanjing Med Univ, Affiliated Canc Hosp, Nanjing, Jiangsu, Peoples R China Nanjing Med Univ, Dept Radiat Oncol, Jiangsu Canc Hosp, Jiangsu Inst Canc Res, Nanjing, Jiangsu, Peoples R ChinaSun, Shi-Yong论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Sch Med, Dept Hematol & Med Oncol, 1365-C Clifton Rd,C3088, Atlanta, GA 30322 USA Winship Canc Inst, 1365-C Clifton Rd,C3088, Atlanta, GA 30322 USA Nanjing Med Univ, Dept Radiat Oncol, Jiangsu Canc Hosp, Jiangsu Inst Canc Res, Nanjing, Jiangsu, Peoples R China
- [3] APG-1252-12A induces mitochondria-dependent apoptosis through inhibiting the antiapoptotic proteins Bcl-2/Bcl-xl in HL-60 cellsINTERNATIONAL JOURNAL OF ONCOLOGY, 2017, 51 (02) : 563 - 572Wang, Jing论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Affiliated Hosp 1, Dept Pharm, 58 2nd Zhongshan Rd, Guangzhou 510080, Guangdong, Peoples R China Sun Yat Sen Univ, Affiliated Hosp 1, Dept Pharm, 58 2nd Zhongshan Rd, Guangzhou 510080, Guangdong, Peoples R ChinaYang, Dajun论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Canc Ctr, Collaborat Innovat Ctr Canc Med, State Key Lab Oncol South China, Guangzhou 510060, Guangdong, Peoples R China Ascentage Pharma Grp Inc, Taizhou 225309, Jiangsu, Peoples R China Sun Yat Sen Univ, Affiliated Hosp 1, Dept Pharm, 58 2nd Zhongshan Rd, Guangzhou 510080, Guangdong, Peoples R ChinaLuo, Qiuyun论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Canc Ctr, Collaborat Innovat Ctr Canc Med, State Key Lab Oncol South China, Guangzhou 510060, Guangdong, Peoples R China Sun Yat Sen Univ, Affiliated Hosp 1, Dept Pharm, 58 2nd Zhongshan Rd, Guangzhou 510080, Guangdong, Peoples R ChinaQiu, Miaozhen论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Canc Ctr, Collaborat Innovat Ctr Canc Med, State Key Lab Oncol South China, Guangzhou 510060, Guangdong, Peoples R China Sun Yat Sen Univ, Affiliated Hosp 1, Dept Pharm, 58 2nd Zhongshan Rd, Guangzhou 510080, Guangdong, Peoples R ChinaZhang, Lin论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Canc Ctr, Collaborat Innovat Ctr Canc Med, State Key Lab Oncol South China, Guangzhou 510060, Guangdong, Peoples R China Sun Yat Sen Univ, Affiliated Hosp 1, Dept Pharm, 58 2nd Zhongshan Rd, Guangzhou 510080, Guangdong, Peoples R ChinaLi, Baoxia论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Canc Ctr, Collaborat Innovat Ctr Canc Med, State Key Lab Oncol South China, Guangzhou 510060, Guangdong, Peoples R China Sun Yat Sen Univ, Affiliated Hosp 1, Dept Pharm, 58 2nd Zhongshan Rd, Guangzhou 510080, Guangdong, Peoples R ChinaChen, Haibo论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Canc Ctr, Collaborat Innovat Ctr Canc Med, State Key Lab Oncol South China, Guangzhou 510060, Guangdong, Peoples R China Sun Yat Sen Univ, Sun Yat Sen Mem Hosp, Guangzhou 510120, Guangdong, Peoples R China Sun Yat Sen Univ, Affiliated Hosp 1, Dept Pharm, 58 2nd Zhongshan Rd, Guangzhou 510080, Guangdong, Peoples R ChinaYi, Hanjie论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Canc Ctr, Collaborat Innovat Ctr Canc Med, State Key Lab Oncol South China, Guangzhou 510060, Guangdong, Peoples R China Sun Yat Sen Univ, Affiliated Hosp 1, Dept Pharm, 58 2nd Zhongshan Rd, Guangzhou 510080, Guangdong, Peoples R ChinaYan, Xianglei论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Canc Ctr, Collaborat Innovat Ctr Canc Med, State Key Lab Oncol South China, Guangzhou 510060, Guangdong, Peoples R China Sun Yat Sen Univ, Affiliated Hosp 1, Dept Pharm, 58 2nd Zhongshan Rd, Guangzhou 510080, Guangdong, Peoples R ChinaLi, Shuxia论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Affiliated Hosp 1, Dept Pharm, 58 2nd Zhongshan Rd, Guangzhou 510080, Guangdong, Peoples R China Sun Yat Sen Univ, Affiliated Hosp 1, Dept Pharm, 58 2nd Zhongshan Rd, Guangzhou 510080, Guangdong, Peoples R ChinaSun, Jian论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Canc Ctr, Collaborat Innovat Ctr Canc Med, State Key Lab Oncol South China, Guangzhou 510060, Guangdong, Peoples R China Sun Yat Sen Univ, Affiliated Hosp 1, Dept Pharm, 58 2nd Zhongshan Rd, Guangzhou 510080, Guangdong, Peoples R China
- [4] A Phase I Study of Novel Bcl-2/Bcl-xL Inhibitor APG-1252 in Patients with Advanced SCLC or Other Solid TumorJOURNAL OF THORACIC ONCOLOGY, 2018, 13 (12) : S1048 - S1049Wu, Y.论文数: 0 引用数: 0 h-index: 0机构: Guangdong Lung Canc Inst, Guangzhou, Guangdong, Peoples R China Guangdong Lung Canc Inst, Guangzhou, Guangdong, Peoples R ChinaLakhani, N. J.论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USA Guangdong Lung Canc Inst, Guangzhou, Guangdong, Peoples R ChinaBoyer, M.论文数: 0 引用数: 0 h-index: 0机构: Chris OBrien Lifehouse, Sydney, NSW, Australia Guangdong Lung Canc Inst, Guangzhou, Guangdong, Peoples R ChinaZhou, Q.论文数: 0 引用数: 0 h-index: 0机构: Guangdong Lung Canc Inst, Guangzhou, Guangdong, Peoples R China Guangdong Lung Canc Inst, Guangzhou, Guangdong, Peoples R ChinaRasco, D. W.论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut, San Antonio, AL USA Guangdong Lung Canc Inst, Guangzhou, Guangdong, Peoples R ChinaHuang, Y.论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma Grp Inc, Rockville, MD USA Guangdong Lung Canc Inst, Guangzhou, Guangdong, Peoples R ChinaMen, L.论文数: 0 引用数: 0 h-index: 0机构: Suzhou Ascentage Pharma Inc, Suzhou, Peoples R China Guangdong Lung Canc Inst, Guangzhou, Guangdong, Peoples R ChinaLi, Y.论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma Grp Inc, Rockville, MD USA Guangdong Lung Canc Inst, Guangzhou, Guangdong, Peoples R ChinaXia, Z.论文数: 0 引用数: 0 h-index: 0机构: Suzhou Ascentage Pharma Inc, Suzhou, Peoples R China Guangdong Lung Canc Inst, Guangzhou, Guangdong, Peoples R ChinaWang, H.论文数: 0 引用数: 0 h-index: 0机构: Suzhou Ascentage Pharma Inc, Suzhou, Peoples R China Guangdong Lung Canc Inst, Guangzhou, Guangdong, Peoples R ChinaJi, J.论文数: 0 引用数: 0 h-index: 0机构: Suzhou Ascentage Pharma Inc, Suzhou, Peoples R China Guangdong Lung Canc Inst, Guangzhou, Guangdong, Peoples R ChinaLu, B.论文数: 0 引用数: 0 h-index: 0机构: Suzhou Ascentage Pharma Inc, Suzhou, Peoples R China Guangdong Lung Canc Inst, Guangzhou, Guangdong, Peoples R ChinaHe, Z.论文数: 0 引用数: 0 h-index: 0机构: Suzhou Ascentage Pharma Inc, Suzhou, Peoples R China Guangdong Lung Canc Inst, Guangzhou, Guangdong, Peoples R ChinaDong, Q.论文数: 0 引用数: 0 h-index: 0机构: Suzhou Ascentage Pharma Inc, Suzhou, Peoples R China Guangdong Lung Canc Inst, Guangzhou, Guangdong, Peoples R ChinaYang, D.论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma Grp Inc, Rockville, MD USA Guangdong Lung Canc Inst, Guangzhou, Guangdong, Peoples R ChinaZhai, Y.论文数: 0 引用数: 0 h-index: 0机构: Suzhou Ascentage Pharma Inc, Suzhou, Peoples R China Guangdong Lung Canc Inst, Guangzhou, Guangdong, Peoples R China
- [5] Dual BCL-2/BCL-XL Inhibitor Pelcitoclax (APG-1252) Overcomes Intrinsic and Acquired Resistance to Venetoclax in Multiple Myeloma CellsBLOOD, 2021, 138Yamamoto, Leona论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USADerebail, Sanika论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USAAktas-Samur, Anil论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USAHideshima, Teru论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USAChyra, Zuzana论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Jerome Lipper Multiple Myeloma Ctr, DanaFarber Canc Inst, Boston, MA USA Harvard Med Sch, LeBow Inst Myeloma Therapeut, Dept Med Oncol, Boston, MA USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USAChakraborty, Chandraditya论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USAYao, Yao论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USAGramegna, Doriana论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USA论文数: 引用数: h-index:机构:Samur, Mehmet K.论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USADeng, Jing论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma Grp Inc, Rockville, MD USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USAZhai, Yifan论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma Grp Inc, Rockville, MD USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USA论文数: 引用数: h-index:机构:Fulciniti, Mariateresa论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USAAnderson, Kenneth C.论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USAMunshi, Nikhil C.论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dana Farber Canc Inst, Boston, MA USA VA Boston Healthcare Syst, Boston, MA USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA USA
- [6] BM-1252 (APG-1252): a potent dual specific Bcl-2/Bcl-xL inhibitor that achieves complete tumor regression with minimal platelet toxicityEUROPEAN JOURNAL OF CANCER, 2014, 50 : 109 - 110Bai, L.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAChen, J.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USALiu, L.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAMcEachern, D.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAAguilar, A.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAZhou, H.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAYang, C. Y.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAWang, H.论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma Grp, Taizhou, Jiangsu, Peoples R China Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAWen, J.论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma Grp, Taizhou, Jiangsu, Peoples R China Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAWang, G.论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma Grp, Taizhou, Jiangsu, Peoples R China Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAZhai, Y.论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma Grp, Taizhou, Jiangsu, Peoples R China Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAGuo, M.论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma Grp, Taizhou, Jiangsu, Peoples R China Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAYang, D.论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma Grp, Taizhou, Jiangsu, Peoples R China Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAWang, S.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA
- [7] Combination of BCL-2/BCL-xL dual inhibitor APG-1252 and chemotherapeutics overcomes resistance to osimertinib in EGFR mutant NSCLC in preclinical modelsCANCER RESEARCH, 2020, 80 (16)Tao, Ran论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma Suzhou Co Ltd, Suzhou, Peoples R China Ascentage Pharma Suzhou Co Ltd, Suzhou, Peoples R ChinaWang, Guangfeng论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma Suzhou Co Ltd, Suzhou, Peoples R China Ascentage Pharma Suzhou Co Ltd, Suzhou, Peoples R ChinaFang, Douglas D.论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma Suzhou Co Ltd, Suzhou, Peoples R China Ascentage Pharma Suzhou Co Ltd, Suzhou, Peoples R ChinaZhai, Guoqin论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma Suzhou Co Ltd, Suzhou, Peoples R China Ascentage Pharma Suzhou Co Ltd, Suzhou, Peoples R ChinaLi, Yuanbao论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma Suzhou Co Ltd, Suzhou, Peoples R China Ascentage Pharma Suzhou Co Ltd, Suzhou, Peoples R ChinaLv, Jing论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma Suzhou Co Ltd, Suzhou, Peoples R China Ascentage Pharma Suzhou Co Ltd, Suzhou, Peoples R ChinaWu, Miaoyi论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma Suzhou Co Ltd, Suzhou, Peoples R China Ascentage Pharma Suzhou Co Ltd, Suzhou, Peoples R ChinaGe, Yangfeng论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma Suzhou Co Ltd, Suzhou, Peoples R China Ascentage Pharma Suzhou Co Ltd, Suzhou, Peoples R ChinaZhang, Feifei论文数: 0 引用数: 0 h-index: 0机构: Shanghai LIDE Biotech Co Ltd, Shanghai, Peoples R China Ascentage Pharma Suzhou Co Ltd, Suzhou, Peoples R ChinaWen, Danyi论文数: 0 引用数: 0 h-index: 0机构: Shanghai LIDE Biotech Co Ltd, Shanghai, Peoples R China Ascentage Pharma Suzhou Co Ltd, Suzhou, Peoples R ChinaYang, Dajun论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Canc Ctr, Guangzhou, Peoples R China Ascentage Pharma Suzhou Co Ltd, Suzhou, Peoples R ChinaZhai, Yifan论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma Suzhou Co Ltd, Suzhou, Peoples R China Ascentage Pharma Suzhou Co Ltd, Suzhou, Peoples R China
- [8] The novel BCL-2/BCL-XL inhibitor APG-1252-mediated cleavage of GSDME enhances the antitumor efficacy of HER2-targeted therapy in HER2-positive gastric cancerACTA PHARMACOLOGICA SINICA, 2024, : 1082 - 1096Luo, Qiu-yun论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Canc Ctr, State Key Lab Oncol South China, Guangzhou 510060, Peoples R China Sun Yat Sen Univ, Affiliated Hosp 3, Dept Clin Res Ctr, Guangzhou 510060, Peoples R China Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Canc Ctr, State Key Lab Oncol South China, Guangzhou 510060, Peoples R ChinaYang, Jing论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Canc Ctr, State Key Lab Oncol South China, Guangzhou 510060, Peoples R China Sun Yat Sen Univ, Canc Ctr, Dept Med Oncol, Guangzhou 510060, Peoples R China Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Canc Ctr, State Key Lab Oncol South China, Guangzhou 510060, Peoples R ChinaDi, Tian论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Canc Ctr, State Key Lab Oncol South China, Guangzhou 510060, Peoples R China Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Canc Ctr, State Key Lab Oncol South China, Guangzhou 510060, Peoples R ChinaXia, Zeng-fei论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Canc Ctr, State Key Lab Oncol South China, Guangzhou 510060, Peoples R China Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Canc Ctr, State Key Lab Oncol South China, Guangzhou 510060, Peoples R ChinaZhang, Lin论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Canc Ctr, State Key Lab Oncol South China, Guangzhou 510060, Peoples R China Sun Yat Sen Univ, Dept Clin Lab, Canc Ctr, Guangzhou 510060, Peoples R China Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Canc Ctr, State Key Lab Oncol South China, Guangzhou 510060, Peoples R ChinaPan, Wen-tao论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Canc Ctr, State Key Lab Oncol South China, Guangzhou 510060, Peoples R China Ascentage Pharm Suzhou Co Ltd, Suzhou 215000, Peoples R China Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Canc Ctr, State Key Lab Oncol South China, Guangzhou 510060, Peoples R ChinaShi, Shan论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Canc Ctr, State Key Lab Oncol South China, Guangzhou 510060, Peoples R China Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Canc Ctr, State Key Lab Oncol South China, Guangzhou 510060, Peoples R ChinaYang, Li-qiong论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Canc Ctr, State Key Lab Oncol South China, Guangzhou 510060, Peoples R China Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Canc Ctr, State Key Lab Oncol South China, Guangzhou 510060, Peoples R ChinaSun, Jian论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Affiliated Hosp 3, Dept Clin Res Ctr, Guangzhou 510060, Peoples R China Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Canc Ctr, State Key Lab Oncol South China, Guangzhou 510060, Peoples R ChinaQiu, Miao-zhen论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Canc Ctr, State Key Lab Oncol South China, Guangzhou 510060, Peoples R China Sun Yat Sen Univ, Canc Ctr, Dept Med Oncol, Guangzhou 510060, Peoples R China Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Canc Ctr, State Key Lab Oncol South China, Guangzhou 510060, Peoples R ChinaYang, Da-jun论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Canc Ctr, State Key Lab Oncol South China, Guangzhou 510060, Peoples R China Ascentage Pharm Suzhou Co Ltd, Suzhou 215000, Peoples R China Sun Yat Sen Univ, Collaborat Innovat Ctr Canc Med, Canc Ctr, State Key Lab Oncol South China, Guangzhou 510060, Peoples R China
- [9] A Potent and Highly Efficacious Bcl-2/Bcl-xL InhibitorJOURNAL OF MEDICINAL CHEMISTRY, 2013, 56 (07) : 3048 - 3067Aguilar, Angelo论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAZhou, Haibin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAChen, Jianfang论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USALiu, Liu论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USABai, Longchuan论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAMcEachern, Donna论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAYang, Chao-Yie论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAMeagher, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Inst Life Sci, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAStuckey, Jeanne论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Inst Life Sci, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAWang, Shaomeng论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA
- [10] Targeting BCL-2 and BCL-xL with a novel dual inhibitor APG-1252 triggers cell death and inhibits tumor growth in small cell lung cancer modelsCANCER RESEARCH, 2018, 78 (13)Wang, GuangFeng论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma, Shanghai, Peoples R China Ascentage Pharma, Shanghai, Peoples R ChinaMin, Ping论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma, Shanghai, Peoples R China Ascentage Pharma, Shanghai, Peoples R ChinaWu, MiaoYi论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma, Shanghai, Peoples R China Ascentage Pharma, Shanghai, Peoples R ChinaDang, Shuo论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma, Shanghai, Peoples R China Ascentage Pharma, Shanghai, Peoples R ChinaTang, ChuanYan论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma, Shanghai, Peoples R China Ascentage Pharma, Shanghai, Peoples R ChinaZhang, Fei论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma, Shanghai, Peoples R China Ascentage Pharma, Shanghai, Peoples R ChinaGuo, Ming论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma, Shanghai, Peoples R China Ascentage Pharma, Shanghai, Peoples R ChinaWang, Shaomeng论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Sch Med, Ann Arbor, MI USA Ascentage Pharma, Shanghai, Peoples R ChinaDeng, Jing论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma, Shanghai, Peoples R China Ascentage Pharma, Shanghai, Peoples R ChinaFang, Douglas D.论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma, Shanghai, Peoples R China Ascentage Pharma, Shanghai, Peoples R ChinaYang, DaJun论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Ctr Canc, Guangzhou, Guangdong, Peoples R China Ascentage Pharma, Shanghai, Peoples R ChinaZhai, YiFan论文数: 0 引用数: 0 h-index: 0机构: Ascentage Pharma, Shanghai, Peoples R China Ascentage Pharma, Shanghai, Peoples R China