共 50 条
- [1] Discovery of novel pyrimidinetrione derivatives as DprE1 inhibitors with potent antimycobacterial activitiesEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 289Liang, Jing论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Wuya Coll Innovat, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Wuya Coll Innovat, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R ChinaLiu, Yang论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Wuya Coll Innovat, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Wuya Coll Innovat, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R ChinaGuan, Qing论文数: 0 引用数: 0 h-index: 0机构: Wuhan Univ, Taikang Med Sch, Frontier Sci Ctr Immunol & Metab, Sch Basic Med Sci,Hubei Prov Key Lab Allergy & Imm, Wuhan 430071, Peoples R China Shenyang Pharmaceut Univ, Wuya Coll Innovat, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R ChinaLi, Yan论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Wuya Coll Innovat, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Wuya Coll Innovat, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R ChinaZheng, Meng-Zhu论文数: 0 引用数: 0 h-index: 0机构: Huazhong Univ Sci & Technol, Tongji Med Coll, Sch Pharm, Hubei Key Lab Nat Med Chem & Resource Evaluat, Wuhan 430071, Peoples R China Shenyang Pharmaceut Univ, Wuya Coll Innovat, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R ChinaZhang, Xiao-Lian论文数: 0 引用数: 0 h-index: 0机构: Wuhan Univ, Taikang Med Sch, Frontier Sci Ctr Immunol & Metab, Sch Basic Med Sci,Hubei Prov Key Lab Allergy & Imm, Wuhan 430071, Peoples R China Wuhan Univ, Zhongnan Hosp, Dept Allergy, Wuhan 430071, Peoples R China Shenyang Pharmaceut Univ, Wuya Coll Innovat, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R ChinaChen, Li-Xia论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Wuya Coll Innovat, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Wuya Coll Innovat, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R ChinaLi, Hua论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Wuya Coll Innovat, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Fujian Univ Tradit Chinese Med, Inst Struct Pharmacol & TCM Chem Biol, Coll Pharm, Fujian Key Lab Chinese Mat Med, Fuzhou 350122, Peoples R China Shenyang Pharmaceut Univ, Wuya Coll Innovat, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China
- [2] Identification and Profiling of Hydantoins-A Novel Class of Potent Antimycobacterial DprE1 InhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2018, 61 (24) : 11221 - 11249Rogacki, Maciej K.论文数: 0 引用数: 0 h-index: 0机构: Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, Univ Pl 1, B-2610 Antwerp, Belgium GlaxoSmithKline, DDW, Tres Cantos Medicines Dev Campus,Severo Ochoa 2, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, Univ Pl 1, B-2610 Antwerp, BelgiumPitta, Eleni论文数: 0 引用数: 0 h-index: 0机构: Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, Univ Pl 1, B-2610 Antwerp, Belgium GlaxoSmithKline, DDW, Tres Cantos Medicines Dev Campus,Severo Ochoa 2, Madrid 28760, Spain Frederick Univ, Sch Hlth Sci, Dept Pharm, Y Freiderickou 7, CY-1036 Nicosia, Cyprus Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, Univ Pl 1, B-2610 Antwerp, BelgiumBalabon, Olga论文数: 0 引用数: 0 h-index: 0机构: Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, Univ Pl 1, B-2610 Antwerp, Belgium GlaxoSmithKline, DDW, Tres Cantos Medicines Dev Campus,Severo Ochoa 2, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, Univ Pl 1, B-2610 Antwerp, BelgiumHuss, Sophie论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, DDW, Tres Cantos Medicines Dev Campus,Severo Ochoa 2, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, Univ Pl 1, B-2610 Antwerp, BelgiumLopez-Roman, Eva Maria论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, DDW, Tres Cantos Medicines Dev Campus,Severo Ochoa 2, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, Univ Pl 1, B-2610 Antwerp, BelgiumArgyrou, Argyrides论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Platform Technol & Sci, Stevenage SG1 2NY, Herts, England AstraZeneca UK Ltd, Discovery Sci, Discovery Biol, IMED Biotech Unit, Darwin Bldg,310 Cambridge Sci Pk, Cambridge CB4 0FZ, England Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, Univ Pl 1, B-2610 Antwerp, BelgiumBlanco-Ruano, Delia论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, DDW, Tres Cantos Medicines Dev Campus,Severo Ochoa 2, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, Univ Pl 1, B-2610 Antwerp, BelgiumCacho, Monica论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, DDW, Tres Cantos Medicines Dev Campus,Severo Ochoa 2, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, Univ Pl 1, B-2610 Antwerp, BelgiumVande Velde, Christophe M. L.论文数: 0 引用数: 0 h-index: 0机构: Univ Antwerp, Fac Appl Engn, Adv Reactor Technol, Groenenborgerlaan 171, B-2020 Antwerp, Belgium Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, Univ Pl 1, B-2610 Antwerp, BelgiumAugustyns, Koen论文数: 0 引用数: 0 h-index: 0机构: Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, Univ Pl 1, B-2610 Antwerp, Belgium Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, Univ Pl 1, B-2610 Antwerp, BelgiumBallell, Lluis论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, DDW, Tres Cantos Medicines Dev Campus,Severo Ochoa 2, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, Univ Pl 1, B-2610 Antwerp, BelgiumBarros, David论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, DDW, Tres Cantos Medicines Dev Campus,Severo Ochoa 2, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, Univ Pl 1, B-2610 Antwerp, BelgiumBates, Robert H.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, DDW, Tres Cantos Medicines Dev Campus,Severo Ochoa 2, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, Univ Pl 1, B-2610 Antwerp, BelgiumCunningham, Fraser论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, DDW, Tres Cantos Medicines Dev Campus,Severo Ochoa 2, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, Univ Pl 1, B-2610 Antwerp, Belgium论文数: 引用数: h-index:机构:
- [3] Scaffold Morphing To Identify Novel DprE1 Inhibitors with Antimycobacterial ActivityACS MEDICINAL CHEMISTRY LETTERS, 2019, 10 (10): : 1480 - 1485Manjunatha, M. R.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, India AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, IndiaShandil, Radha论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, DMPK & Anim Sci, IMED Infect, Bangalore 560024, Karnataka, India Fdn Neglected Dis Res, 20A KIADB Ind Area, Bengaluru 561203, India AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, IndiaPanda, Manoranjan论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, India AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, IndiaSadler, Claire论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Safety Assessment, IMED, Alderly Pk, Mereside, England AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, IndiaAmbady, Anisha论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, IMED Infect, Dept Biosci, Bangalore 560024, Karnataka, India AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, IndiaPanduga, Vijender论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, DMPK & Anim Sci, IMED Infect, Bangalore 560024, Karnataka, India AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, IndiaKumar, Naveen论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, DMPK & Anim Sci, IMED Infect, Bangalore 560024, Karnataka, India AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, IndiaMahadevaswamy, Jyothi论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, IMED Infect, Dept Biosci, Bangalore 560024, Karnataka, India AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, IndiaSreenivasaiah, M.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, India AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, IndiaNarayan, Ashwini论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, IMED Infect, Dept Biosci, Bangalore 560024, Karnataka, India AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, IndiaGuptha, Supreeth论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, IMED Infect, Dept Biosci, Bangalore 560024, Karnataka, India AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, IndiaSharma, Sreevalli论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, IMED Infect, Dept Biosci, Bangalore 560024, Karnataka, India AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, IndiaSambandamurthy, Vasan K.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, IMED Infect, Dept Biosci, Bangalore 560024, Karnataka, India AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, IndiaRamachandran, Vasanthi论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, IMED Infect, Dept Biosci, Bangalore 560024, Karnataka, India AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, IndiaMallya, Meenakshi论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, India AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, IndiaCooper, Christopher论文数: 0 引用数: 0 h-index: 0机构: Global Alliance TB, New York, NY 10005 USA AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, IndiaMdluli, Khisi论文数: 0 引用数: 0 h-index: 0机构: Global Alliance TB, New York, NY 10005 USA AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, IndiaButler, Scott论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, GHP, Infect IMED, Waltham, MA 02451 USA AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, IndiaTommasi, Ruben论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, GHP, Infect IMED, Waltham, MA 02451 USA AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, IndiaIyer, Pravin S.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, India AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, IndiaNarayanan, Shridhar论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, IMED Infect, Dept Biosci, Bangalore 560024, Karnataka, India Fdn Neglected Dis Res, 20A KIADB Ind Area, Bengaluru 561203, India AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, IndiaChatterji, Monalisa论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, IMED Infect, Dept Biosci, Bangalore 560024, Karnataka, India AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, IndiaShirude, Pravin S.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, India Biocon Bristol Myers Squibb Res & Dev Ctr, Bommasandra Jigani Link Rd, Bangalore 560099, Karnataka, India AstraZeneca India, Dept Med Chem, IMED Infect, Bellary Rd, Bangalore 560024, Karnataka, India
- [4] Optimization of Hydantoins as Potent Antimycobacterial Decaprenylphosphoryl-β-D-Ribose Oxidase (DprE1) InhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2020, 63 (10) : 5367 - 5386Balabon, Olga论文数: 0 引用数: 0 h-index: 0机构: Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, B-2610 Antwerp, Belgium GlaxoSmithKline, Global Hlth R&D, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, B-2610 Antwerp, BelgiumPitta, Eleni论文数: 0 引用数: 0 h-index: 0机构: Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, B-2610 Antwerp, Belgium GlaxoSmithKline, Global Hlth R&D, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, B-2610 Antwerp, BelgiumRogacki, Maciej K.论文数: 0 引用数: 0 h-index: 0机构: Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, B-2610 Antwerp, Belgium GlaxoSmithKline, Global Hlth R&D, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, B-2610 Antwerp, BelgiumMeiler, Eugenia论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Global Hlth R&D, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, B-2610 Antwerp, BelgiumCasanueva, Ruth论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Global Hlth R&D, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, B-2610 Antwerp, BelgiumGuijarro, Laura论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Global Hlth R&D, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, B-2610 Antwerp, BelgiumHuss, Sophie论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Global Hlth R&D, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, B-2610 Antwerp, BelgiumMaria Lopez-Roman, Eva论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Global Hlth R&D, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, B-2610 Antwerp, BelgiumSantos-Villarejo, Angel论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Global Hlth R&D, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, B-2610 Antwerp, BelgiumAugustyns, Koen论文数: 0 引用数: 0 h-index: 0机构: Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, B-2610 Antwerp, Belgium Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, B-2610 Antwerp, BelgiumBallell, Lluis论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Global Hlth R&D, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, B-2610 Antwerp, BelgiumBarros Aguirre, David论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Global Hlth R&D, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, B-2610 Antwerp, BelgiumBates, Robert H.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Global Hlth R&D, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, B-2610 Antwerp, BelgiumCunningham, Fraser论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Global Hlth R&D, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, B-2610 Antwerp, BelgiumCacho, Monica论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Global Hlth R&D, Madrid 28760, Spain Univ Antwerp, Dept Pharmaceut Sci, Lab Med Chem, B-2610 Antwerp, Belgium论文数: 引用数: h-index:机构:
- [5] Design, Synthesis, and Molecular Docking of Novel Benzothiazinone Derivatives as DprE1 Inhibitors with Potential Antitubercular ActivitiesRUSSIAN JOURNAL OF BIOORGANIC CHEMISTRY, 2025, 51 (01) : 65 - 78Raghu, M. S.论文数: 0 引用数: 0 h-index: 0机构: New Horizon Coll Engn, Dept Chem, Bengaluru 560103, Karnataka, India New Horizon Coll Engn, Dept Chem, Bengaluru 560103, Karnataka, IndiaJassim, Amar Yasser论文数: 0 引用数: 0 h-index: 0机构: Univ Basrah, Marine Sci Ctr, Dept Marine Vertebrate, Basra, Iraq New Horizon Coll Engn, Dept Chem, Bengaluru 560103, Karnataka, IndiaKumar, K. Yogesh论文数: 0 引用数: 0 h-index: 0机构: Jain Univ, Fac Engn & Technol, Dept Chem, Ramanagara 562112, India New Horizon Coll Engn, Dept Chem, Bengaluru 560103, Karnataka, IndiaAlharethy, Fahd论文数: 0 引用数: 0 h-index: 0机构: King Saud Univ, Coll Sci, Dept Chem, Riyadh 11451, Saudi Arabia New Horizon Coll Engn, Dept Chem, Bengaluru 560103, Karnataka, IndiaPrashanth, M. K.论文数: 0 引用数: 0 h-index: 0机构: BNM Inst Technol, Dept Chem, Bengaluru 560070, India New Horizon Coll Engn, Dept Chem, Bengaluru 560103, Karnataka, IndiaJeon, Byong-Hun论文数: 0 引用数: 0 h-index: 0机构: Hanyang Univ, Dept Earth Resources & Environm Engn, 222 Wangsimni Ro, Seoul 04763, South Korea New Horizon Coll Engn, Dept Chem, Bengaluru 560103, Karnataka, India
- [6] Identification of novel DprE1 inhibitors for the treatment of tuberculosisABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2013, 245Franco, Jimmy论文数: 0 引用数: 0 h-index: 0机构: Merrimack Coll, Dept Chem, N Andover, MA 01845 USA Merrimack Coll, Dept Chem, N Andover, MA 01845 USALaverty, Daniel论文数: 0 引用数: 0 h-index: 0机构: Merrimack Coll, Dept Chem, N Andover, MA 01845 USA Merrimack Coll, Dept Chem, N Andover, MA 01845 USADaniels, Dave论文数: 0 引用数: 0 h-index: 0机构: Merrimack Coll, Dept Chem, N Andover, MA 01845 USA Merrimack Coll, Dept Chem, N Andover, MA 01845 USAWilsey, Claire论文数: 0 引用数: 0 h-index: 0机构: Merrimack Coll, Dept Chem, N Andover, MA 01845 USA Merrimack Coll, Dept Chem, N Andover, MA 01845 USAGolijanin, Petar论文数: 0 引用数: 0 h-index: 0机构: Merrimack Coll, Dept Chem, N Andover, MA 01845 USA Merrimack Coll, Dept Chem, N Andover, MA 01845 USAGurka, Jessica论文数: 0 引用数: 0 h-index: 0机构: Merrimack Coll, Dept Chem, N Andover, MA 01845 USA Merrimack Coll, Dept Chem, N Andover, MA 01845 USA
- [7] Discovery of novel thiophene derivatives as potent neuraminidase inhibitorsEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 225Zhong, Zhi Jian论文数: 0 引用数: 0 h-index: 0机构: Shanghai Inst Technol, Sch Chem & Environm Engn, Shanghai 201418, Peoples R China Shanghai Inst Technol, Sch Chem & Environm Engn, Shanghai 201418, Peoples R ChinaHu, Xiao Tong论文数: 0 引用数: 0 h-index: 0机构: Huazhong Agr Univ, Coll Vet Med, Unit Anim Infect Dis, State Key Lab Agr Microbiol, Wuhan 430070, Hubei, Peoples R China Shanghai Inst Technol, Sch Chem & Environm Engn, Shanghai 201418, Peoples R ChinaCheng, Li Ping论文数: 0 引用数: 0 h-index: 0机构: Shanghai Inst Technol, Sch Chem & Environm Engn, Shanghai 201418, Peoples R China Shanghai Inst Technol, Sch Chem & Environm Engn, Shanghai 201418, Peoples R ChinaZhang, Xing Yong论文数: 0 引用数: 0 h-index: 0机构: Shanghai Inst Technol, Sch Chem & Environm Engn, Shanghai 201418, Peoples R China Shanghai Inst Technol, Sch Chem & Environm Engn, Shanghai 201418, Peoples R ChinaZhang, Qiang论文数: 0 引用数: 0 h-index: 0机构: Huazhong Agr Univ, Coll Biomed & Hlth, Wuhan 430070, Hubei, Peoples R China Shanghai Inst Technol, Sch Chem & Environm Engn, Shanghai 201418, Peoples R ChinaZhang, Ju论文数: 0 引用数: 0 h-index: 0机构: Huazhong Agr Univ, Wuhan Yangene Biol Technol Co LTD, Yuechuang Ctr, Wuhan 430070, Hubei, Peoples R China Shanghai Inst Technol, Sch Chem & Environm Engn, Shanghai 201418, Peoples R China
- [8] 4-Aminoquinolone Piperidine Amides: Noncovalent Inhibitors of DprE1 with Long Residence Time and Potent Antimycobacterial ActivityJOURNAL OF MEDICINAL CHEMISTRY, 2014, 57 (12) : 5419 - 5434Naik, Maruti论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, IndiaHumnabadkar, Vaishali论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, Dept Biosci, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, IndiaTantry, Subramanyam J.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, IndiaPanda, Manoranjan论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, IndiaNarayan, Ashwini论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, Dept Biosci, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, IndiaGuptha, Supreeth论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, Dept Biosci, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, IndiaPanduga, Vijender论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, DMPK Drug Metab & Pharmacokinet & Anim Sci, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, IndiaManjrekar, Praveena论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, IndiaJena, Lalit Kumar论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, IndiaKoushik, Krishna论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, IndiaShanbhag, Gajanan论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, IndiaJatheendranath, Sandesh论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, IndiaManjunatha, M. 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- [10] Discovery of Pyrazolopyridones as a Novel Class of Noncovalent DprE1 Inhibitor with Potent Anti-Mycobacterial ActivityJOURNAL OF MEDICINAL CHEMISTRY, 2014, 57 (11) : 4761 - 4771Panda, Manoranjan论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, IndiaRamachandran, Sreekanth论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, IndiaRamachandran, Vasanthi论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, IMED Infect, Dept Biosci, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, IndiaShirude, Pravin S.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, IndiaHumnabadkar, Vaishali论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, IMED Infect, Dept Biosci, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, IndiaNagalapur, Kavitha论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, IndiaSharma, Sreevalli论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, IMED Infect, Dept Biosci, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, IndiaKaur, Parvinder论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, IMED Infect, Dept Biosci, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, IndiaGuptha, Supreeth论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, IMED Infect, Dept Biosci, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, IndiaNarayan, Ashwini论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, IMED Infect, Dept Biosci, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, IndiaMahadevaswamy, Jyothi论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, IMED Infect, Dept Biosci, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, IndiaAmbady, Anisha论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, IMED Infect, Dept Biosci, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, IndiaHegde, Naina论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, IMED Infect, Dept Biosci, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, IndiaRudrapatna, Suresh S.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, IndiaHosagrahara, Vinayak P.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, IMED Infect, Dept Biosci, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, IndiaSambandamurthy, Vasan K.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, IMED Infect, Dept Biosci, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, IndiaRaichurkar, Anandkumar论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, IMED Infect, Dept Chem, Bangalore 560024, Karnataka, India