AURORA AND POLO-LIKE KINASE INHIBITORS: A CLINICAL PERSPECTIVE

被引:0
|
作者
Awada, A. [1 ]
Metzger, O. [1 ]
机构
[1] Inst Jules Bordet, B-1000 Brussels, Belgium
关键词
D O I
暂无
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
引用
收藏
页码:27 / 27
页数:1
相关论文
共 50 条
  • [1] Synthetic Strategies of Pyrimidine-Based Scaffolds as Aurora Kinase and Polo-like Kinase Inhibitors
    Jadhav, Mrunal
    Sankhe, Kaksha
    Bhandare, Richie R.
    Edis, Zehra
    Bloukh, Samir Haj
    Khan, Tabassum Asif
    MOLECULES, 2021, 26 (17):
  • [2] Discovery of thiophene inhibitors of polo-like kinase
    Emmitte, Kyle A.
    Andrews, C. Webb
    Badiang, Jennifer G.
    Davis-Ward, Ronda G.
    Dickson, Hamilton D.
    Drewry, David H.
    Emerson, Holly K.
    Epperly, Andrea H.
    Hassler, Daniel F.
    Knick, Victoria B.
    Kuntz, Kevin W.
    Lansing, Timothy J.
    Linn, James A.
    Mook, Robert A., Jr.
    Nailor, Kristen E.
    Salovich, James M.
    Spehar, Glenn M.
    Cheung, Mui
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009, 19 (03) : 1018 - 1021
  • [3] Developing polo-like kinase 1 inhibitors
    Huang, Xufeng
    Xie, Zhouling
    Liao, Chenzhong
    FUTURE MEDICINAL CHEMISTRY, 2020, 12 (10) : 869 - 871
  • [4] Human Polo-like Kinase Inhibitors as Antiplasmodials
    Bohmer, Monica J.
    Wang, Jinhua
    Istvan, Eva S.
    Luth, Madeline R.
    Collins, Jennifer E.
    Huttlin, Edward L.
    Wang, Lushun
    Mittal, Nimisha
    Hao, Mingfeng
    Kwiatkowski, Nicholas P.
    Gygi, Steven P.
    Chakrabarti, Ratna
    Deng, Xianming
    Goldberg, Daniel E.
    Winzeler, Elizabeth A.
    Gray, Nathanael S.
    Chakrabarti, Debopam
    ACS INFECTIOUS DISEASES, 2023, 9 (04): : 1004 - 1021
  • [5] Polo-like kinase inhibitors in hematologic malignancies
    Talati, Chetasi
    Griffiths, Elizabeth A.
    Wetzler, Meir
    Wang, Eunice S.
    CRITICAL REVIEWS IN ONCOLOGY HEMATOLOGY, 2016, 98 : 200 - 210
  • [6] Progress in the discovery of polo-like kinase inhibitors
    McInnes, C
    Mezna, M
    Fischer, PM
    CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2005, 5 (02) : 181 - 197
  • [7] Inhibitors of the Polo-Box Domain of Polo-Like Kinase 1
    Berg, Angela
    Berg, Thorsten
    CHEMBIOCHEM, 2016, 17 (08) : 650 - 656
  • [8] Polo-Like Kinase (PLK) Inhibitors in Preclinical and Early Clinical Development in Oncology
    Schoffski, Patrick
    ONCOLOGIST, 2009, 14 (06): : 559 - 570
  • [9] Current clinical trials with polo-like kinase 1 inhibitors in solid tumors
    Yim, Hyungshin
    ANTI-CANCER DRUGS, 2013, 24 (10) : 999 - 1006
  • [10] Application of a Fluorescence Recovery-Based Polo-Like Kinase 1 Binding Assay to Polo-Like Kinase 2 and Polo-Like Kinase 3
    Tsuji, Kohei
    Tamamura, Hirokazu
    Burke Jr, Terrence R.
    BIOLOGICAL & PHARMACEUTICAL BULLETIN, 2024, 47 (07) : 1282 - 1287