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- [1] Structure-based design of Trifarotene (CD5789), a potent and selective RARγ agonist for the treatment of acne[J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2018, 28 (10) : 1736 - 1741Thoreau, Etienne论文数: 0 引用数: 0 h-index: 0机构: Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, France Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, FranceArlabosse, Jean-Marie论文数: 0 引用数: 0 h-index: 0机构: Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, France Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, FranceBouix-Peter, Claire论文数: 0 引用数: 0 h-index: 0机构: Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, France Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, FranceChambon, Sandrine论文数: 0 引用数: 0 h-index: 0机构: Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, France Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, FranceChantalat, Laurent论文数: 0 引用数: 0 h-index: 0机构: Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, France Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, FranceDaver, Sebastien论文数: 0 引用数: 0 h-index: 0机构: Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, France Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, FranceDumais, Laurence论文数: 0 引用数: 0 h-index: 0机构: Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, France Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, FranceDuvert, Gwenaelle论文数: 0 引用数: 0 h-index: 0机构: Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, France Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, FranceFeret, Angelique论文数: 0 引用数: 0 h-index: 0机构: Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, France Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, FranceOuvry, Gilles论文数: 0 引用数: 0 h-index: 0机构: Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, France Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, FrancePascau, Jonathan论文数: 0 引用数: 0 h-index: 0机构: Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, France Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, FranceRaffin, Catherine论文数: 0 引用数: 0 h-index: 0机构: Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, France Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, FranceRodeville, Nicolas论文数: 0 引用数: 0 h-index: 0机构: Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, France Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, FranceSoulet, Catherine论文数: 0 引用数: 0 h-index: 0机构: Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, France Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, FranceTabet, Samuel论文数: 0 引用数: 0 h-index: 0机构: Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, France Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, FranceTalano, Sandrine论文数: 0 引用数: 0 h-index: 0机构: Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, France Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, FrancePortal, Thibaud论文数: 0 引用数: 0 h-index: 0机构: Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, France Nestle Skin Hlth, Les Templiers 2400 Route Colles, F-06410 Biot, France
- [2] Non-clinical and human pharmacology of the potent and selective topical RARγ agonist trifarotene[J]. JOURNAL OF INVESTIGATIVE DERMATOLOGY, 2018, 138 (09) : B17 - B17Aubert, J.论文数: 0 引用数: 0 h-index: 0机构: Galderma R&D, Biot, Provence Alpes, France Galderma R&D, Biot, Provence Alpes, FranceBertino, B.论文数: 0 引用数: 0 h-index: 0机构: Galderma R&D, Biot, Provence Alpes, France Galderma R&D, Biot, Provence Alpes, FranceBlanchet-Rethore, S.论文数: 0 引用数: 0 h-index: 0机构: Galderma R&D, Biot, Provence Alpes, France Galderma R&D, Biot, Provence Alpes, FranceCarlavan, I.论文数: 0 引用数: 0 h-index: 0机构: Galderma R&D, Biot, Provence Alpes, France Galderma R&D, Biot, Provence Alpes, FranceDeret, S.论文数: 0 引用数: 0 h-index: 0机构: Galderma R&D, Nestle Skin Hlth, Biot, Provence Alpes, France Galderma R&D, Biot, Provence Alpes, FranceDreno, B.论文数: 0 引用数: 0 h-index: 0机构: Univ Nantes, CRCINA, CHU Nantes, CIC 1413, Nantes, Pays De La Loir, France Galderma R&D, Biot, Provence Alpes, FranceLuzy, A.论文数: 0 引用数: 0 h-index: 0机构: Galderma R&D, Biot, Provence Alpes, France Galderma R&D, Biot, Provence Alpes, FranceMounier, C.论文数: 0 引用数: 0 h-index: 0机构: Galderma R&D, Biot, Provence Alpes, France Galderma R&D, Biot, Provence Alpes, FrancePascau, J.论文数: 0 引用数: 0 h-index: 0机构: Galderma R&D, Nestle Skin Hlth, Biot, Provence Alpes, France Galderma R&D, Biot, Provence Alpes, FrancePelisson, I.论文数: 0 引用数: 0 h-index: 0机构: Galderma R&D, Biot, Provence Alpes, France Galderma R&D, Biot, Provence Alpes, FrancePortal, T.论文数: 0 引用数: 0 h-index: 0机构: Galderma SA, Lausanne, Vaud, Switzerland Galderma R&D, Biot, Provence Alpes, FranceRivier, M.论文数: 0 引用数: 0 h-index: 0机构: Galderma R&D, Biot, Provence Alpes, France Galderma R&D, Biot, Provence Alpes, FranceRosso, P.论文数: 0 引用数: 0 h-index: 0机构: Galderma R&D, Biot, Provence Alpes, France Galderma R&D, Biot, Provence Alpes, FranceThoreau, E.论文数: 0 引用数: 0 h-index: 0机构: Nestle Skin Hlth, Biot, Provence Alpes, France Galderma R&D, Biot, Provence Alpes, FranceVial, E.论文数: 0 引用数: 0 h-index: 0机构: Galderma R&D, Nestle Skin Hlth, Biot, Provence Alpes, France Galderma R&D, Biot, Provence Alpes, FranceVoegel, J. J.论文数: 0 引用数: 0 h-index: 0机构: Galderma R&D, Biot, Provence Alpes, France Galderma R&D, Biot, Provence Alpes, France
- [3] Structure-based design of potent and selective CGRP receptor antagonists for the treatment of migraine[J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2019, 258Bell, Ian论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Discovery Chem, West Point, PA USA Merck & Co Inc, Discovery Chem, West Point, PA USA
- [4] Structure-Based Design of Potent and Selective Inhibitors of Pyruvate Carboxylase[J]. PROTEIN SCIENCE, 2021, 30 : 141 - 141Schneider, Nicholas论文数: 0 引用数: 0 h-index: 0机构: Marquette Univ, Dept Biol Sci, Milwaukee, WI 53233 USA Marquette Univ, Dept Biol Sci, Milwaukee, WI 53233 USABurkett, Daniel论文数: 0 引用数: 0 h-index: 0机构: Marquette Univ, Dept Chem, Milwaukee, WI 53233 USA Marquette Univ, Dept Biol Sci, Milwaukee, WI 53233 USAWyatt, Brittney论文数: 0 引用数: 0 h-index: 0机构: Marquette Univ, Dept Biol Sci, Milwaukee, WI 53233 USA Marquette Univ, Dept Biol Sci, Milwaukee, WI 53233 USAMews, Mallory论文数: 0 引用数: 0 h-index: 0机构: Marquette Univ, Dept Biol Sci, Milwaukee, WI 53233 USA Marquette Univ, Dept Biol Sci, Milwaukee, WI 53233 USABautista, Anson论文数: 0 引用数: 0 h-index: 0机构: Marquette Univ, Dept Chem, Milwaukee, WI 53233 USA Marquette Univ, Dept Biol Sci, Milwaukee, WI 53233 USAEngel, Ryan论文数: 0 引用数: 0 h-index: 0机构: Marquette Univ, Dept Chem, Milwaukee, WI 53233 USA Marquette Univ, Dept Biol Sci, Milwaukee, WI 53233 USADockendorff, Chris论文数: 0 引用数: 0 h-index: 0机构: Marquette Univ, Dept Chem, Milwaukee, WI 53233 USA Marquette Univ, Dept Biol Sci, Milwaukee, WI 53233 USADonaldson, William论文数: 0 引用数: 0 h-index: 0机构: Marquette Univ, Dept Chem, Milwaukee, WI 53233 USA Marquette Univ, Dept Biol Sci, Milwaukee, WI 53233 USASt Maurice, Martin论文数: 0 引用数: 0 h-index: 0机构: Marquette Univ, Dept Biol Sci, Milwaukee, WI 53233 USA Marquette Univ, Dept Biol Sci, Milwaukee, WI 53233 USA
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