A general palladium-catalyzed coupling of aryl bromides/triflates and thiols

被引：467
|
作者：
Itoh, T [1 ]
Mase, T [1 ]
机构：
[1] Banyu Pharmaceut Co Ltd, Proc Res, Proc R&D, Okazaki, Aichi 4440858, Japan
来源：
ORGANIC LETTERS | 2004年 / 6卷 / 24期
关键词：
D O I：
10.1021/ol047996t
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
[GRAPHICS] We have developed an efficient palladium-catalyzed carbon-sulfur bond formation reaction of aryl bromides, triflates, and activated aryl chloride, Using this protocol, we have shown tolerance to a wide variety of aryl thiols and alkyl thiols that can also be used as sulfide equivalents.
引用
收藏
页码：4587 / 4590
页数：4
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