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- [1] Mutant-Selective Irreversible EGFR Inhibitor, Naquotinib, Inhibits Tumor Growth in NSCLC Models with EGFR-Activating Mutations, T790M Mutation, and AXL OverexpressionMOLECULAR CANCER THERAPEUTICS, 2019, 18 (08) : 1366 - 1373Tanaka, Hiroaki论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanSakagami, Hideki论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanKaneko, Naoki论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanKonagai, Satoshi论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanYamamoto, Hiroko论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanMatsuya, Takahiro论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanYuri, Masatoshi论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanYamanaka, Yosuke论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanMori, Masamichi论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanTakeuchi, Masahiro论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanKoshio, Hiroyuki论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanHirano, Masaaki论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanKuromitsu, Sadao论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan
- [2] Discovery of a Mutant-Selective Covalent Inhibitor of EGFR that Overcomes T790M-Mediated Resistance in NSCLCCANCER DISCOVERY, 2013, 3 (12) : 1404 - 1415Walter, Annette O.论文数: 0 引用数: 0 h-index: 0机构: Clovis Oncol Inc, San Francisco, CA 94158 USA Clovis Oncol Inc, San Francisco, CA 94158 USASjin, Robert Tjin Tham论文数: 0 引用数: 0 h-index: 0机构: Celgene Avil Res, Bedford, MA USA Clovis Oncol Inc, San Francisco, CA 94158 USAHaringsma, Henry J.论文数: 0 引用数: 0 h-index: 0机构: Clovis Oncol Inc, San Francisco, CA 94158 USA Clovis Oncol Inc, San Francisco, CA 94158 USAOhashi, Kadoaki论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Med, Div Hematol Oncol, Nashville, TN 37212 USA Clovis Oncol Inc, San Francisco, CA 94158 USASun, Jing论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Med, Div Hematol Oncol, Nashville, TN 37212 USA Clovis Oncol Inc, San Francisco, CA 94158 USALee, Kwangho论文数: 0 引用数: 0 h-index: 0机构: Celgene Avil Res, Bedford, MA USA Clovis Oncol Inc, San Francisco, CA 94158 USADubrovskiy, Aleksandr论文数: 0 引用数: 0 h-index: 0机构: Celgene Avil Res, Bedford, MA USA Clovis Oncol Inc, San Francisco, CA 94158 USALabenski, Matthew论文数: 0 引用数: 0 h-index: 0机构: Celgene Avil Res, Bedford, MA USA Clovis Oncol Inc, San Francisco, CA 94158 USAZhu, Zhendong论文数: 0 引用数: 0 h-index: 0机构: Celgene Avil Res, Bedford, MA USA Clovis Oncol Inc, San Francisco, CA 94158 USAWang, Zhigang论文数: 0 引用数: 0 h-index: 0机构: Celgene Avil Res, Bedford, MA USA Clovis Oncol Inc, San Francisco, CA 94158 USASheets, Michael论文数: 0 引用数: 0 h-index: 0机构: Celgene Avil Res, Bedford, MA USA Clovis Oncol Inc, San Francisco, CA 94158 USASt Martin, Thia论文数: 0 引用数: 0 h-index: 0机构: Celgene Avil Res, Bedford, MA USA Clovis Oncol Inc, San Francisco, CA 94158 USAKarp, Russell论文数: 0 引用数: 0 h-index: 0机构: Celgene Avil Res, Bedford, MA USA Clovis Oncol Inc, San Francisco, CA 94158 USAvan Kalken, Dan论文数: 0 引用数: 0 h-index: 0机构: Celgene Avil Res, Bedford, MA USA Clovis Oncol Inc, San Francisco, CA 94158 USAChaturvedi, Prasoon论文数: 0 引用数: 0 h-index: 0机构: Celgene Avil Res, Bedford, MA USA Clovis Oncol Inc, San Francisco, CA 94158 USANiu, Deqiang论文数: 0 引用数: 0 h-index: 0机构: Celgene Avil Res, Bedford, MA USA Clovis Oncol Inc, San Francisco, CA 94158 USANacht, Mariana论文数: 0 引用数: 0 h-index: 0机构: Celgene Avil Res, Bedford, MA USA Clovis Oncol Inc, San Francisco, CA 94158 USAPetter, Russell C.论文数: 0 引用数: 0 h-index: 0机构: Celgene Avil Res, Bedford, MA USA Clovis Oncol Inc, San Francisco, CA 94158 USAWestlin, William论文数: 0 引用数: 0 h-index: 0机构: Celgene Avil Res, Bedford, MA USA Clovis Oncol Inc, San Francisco, CA 94158 USALin, Kevin论文数: 0 引用数: 0 h-index: 0机构: Clovis Oncol Inc, San Francisco, CA 94158 USA Clovis Oncol Inc, San Francisco, CA 94158 USAJaw-Tsai, Sarah论文数: 0 引用数: 0 h-index: 0机构: Clovis Oncol Inc, San Francisco, CA 94158 USA Clovis Oncol Inc, San Francisco, CA 94158 USARaponi, Mitch论文数: 0 引用数: 0 h-index: 0机构: Clovis Oncol Inc, San Francisco, CA 94158 USA Clovis Oncol Inc, San Francisco, CA 94158 USAVan Dyke, Terry论文数: 0 引用数: 0 h-index: 0机构: NCI, Mouse Canc Genet Program, Frederick, MD 21701 USA NCI, Ctr Adv Preclin Res, Sci Applicat Int Corp Frederick Inc, Frederick, MD 21701 USA Clovis Oncol Inc, San Francisco, CA 94158 USAEtter, Jeff论文数: 0 引用数: 0 h-index: 0机构: Clovis Oncol Inc, San Francisco, CA 94158 USA Clovis Oncol Inc, San Francisco, CA 94158 USAWeaver, Zoe论文数: 0 引用数: 0 h-index: 0机构: NCI, Ctr Adv Preclin Res, Sci Applicat Int Corp Frederick Inc, Frederick, MD 21701 USA Clovis Oncol Inc, San Francisco, CA 94158 USAPao, William论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Med, Div Hematol Oncol, Nashville, TN 37212 USA Clovis Oncol Inc, San Francisco, CA 94158 USASingh, Juswinder论文数: 0 引用数: 0 h-index: 0机构: Celgene Avil Res, Bedford, MA USA Clovis Oncol Inc, San Francisco, CA 94158 USASimmons, Andrew D.论文数: 0 引用数: 0 h-index: 0机构: Clovis Oncol Inc, San Francisco, CA 94158 USA Clovis Oncol Inc, San Francisco, CA 94158 USAHarding, Thomas C.论文数: 0 引用数: 0 h-index: 0机构: Clovis Oncol Inc, San Francisco, CA 94158 USA Clovis Oncol Inc, San Francisco, CA 94158 USAAllen, Andrew论文数: 0 引用数: 0 h-index: 0机构: Clovis Oncol Inc, San Francisco, CA 94158 USA Clovis Oncol Inc, San Francisco, CA 94158 USA
- [3] Novel mutant-selective EGFR kinase inhibitors against EGFR T790MNATURE, 2009, 462 (7276) : 1070 - 1074Zhou, Wenjun论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAErcan, Dalia论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAChen, Liang论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAYun, Cai-Hong论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USALi, Danan论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA论文数: 引用数: h-index:机构:Cortot, Alexis B.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAChirieac, Lucian论文数: 0 引用数: 0 h-index: 0机构: Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAIacob, Roxana E.论文数: 0 引用数: 0 h-index: 0机构: Northeastern Univ, Barnett Inst Chem & Biol Anal, Boston, MA 02115 USA Northeastern Univ, Dept Chem & Biol Chem, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAPadera, Robert论文数: 0 引用数: 0 h-index: 0机构: Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAEngen, John R.论文数: 0 引用数: 0 h-index: 0机构: Northeastern Univ, Barnett Inst Chem & Biol Anal, Boston, MA 02115 USA Northeastern Univ, Dept Chem & Biol Chem, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAWong, Kwok-Kin论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA Brigham & Womens Hosp, Dept Med, Boston, MA 02115 USA Harvard Univ, Sch Med, Boston, MA 02115 USA Dana Farber Harvard Canc Ctr, Ludwig Ctr, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAEck, Michael J.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAGray, Nathanael S.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAJaenne, Pasi A.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA Brigham & Womens Hosp, Dept Med, Boston, MA 02115 USA Harvard Univ, Sch Med, Boston, MA 02115 USA Dana Farber Harvard Canc Ctr, Ludwig Ctr, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA
- [4] Novel mutant-selective EGFR kinase inhibitors against EGFR T790MNature, 2009, 462 : 1070 - 1074Wenjun Zhou论文数: 0 引用数: 0 h-index: 0机构: Department of Cancer Biology,Department of Medical OncologyDalia Ercan论文数: 0 引用数: 0 h-index: 0机构: Department of Cancer Biology,Department of Medical OncologyLiang Chen论文数: 0 引用数: 0 h-index: 0机构: Department of Cancer Biology,Department of Medical OncologyCai-Hong Yun论文数: 0 引用数: 0 h-index: 0机构: Department of Cancer Biology,Department of Medical OncologyDanan Li论文数: 0 引用数: 0 h-index: 0机构: Department of Cancer Biology,Department of Medical OncologyMarzia Capelletti论文数: 0 引用数: 0 h-index: 0机构: Department of Cancer Biology,Department of Medical OncologyAlexis B. Cortot论文数: 0 引用数: 0 h-index: 0机构: Department of Cancer Biology,Department of Medical OncologyLucian Chirieac论文数: 0 引用数: 0 h-index: 0机构: Department of Cancer Biology,Department of Medical OncologyRoxana E. Iacob论文数: 0 引用数: 0 h-index: 0机构: Department of Cancer Biology,Department of Medical OncologyRobert Padera论文数: 0 引用数: 0 h-index: 0机构: Department of Cancer Biology,Department of Medical OncologyJohn R. Engen论文数: 0 引用数: 0 h-index: 0机构: Department of Cancer Biology,Department of Medical OncologyKwok-Kin Wong论文数: 0 引用数: 0 h-index: 0机构: Department of Cancer Biology,Department of Medical OncologyMichael J. Eck论文数: 0 引用数: 0 h-index: 0机构: Department of Cancer Biology,Department of Medical OncologyNathanael S. Gray论文数: 0 引用数: 0 h-index: 0机构: Department of Cancer Biology,Department of Medical OncologyPasi A. Jänne论文数: 0 引用数: 0 h-index: 0机构: Department of Cancer Biology,Department of Medical Oncology
- [5] Preclinical assessment of a mutant-selective covalent inhibitor of EGFR that overcomes T790M-mediated resistance in NSCLC.MOLECULAR CANCER THERAPEUTICS, 2013, 12 (11)Simmons, Andrew D.论文数: 0 引用数: 0 h-index: 0机构: Clovis Oncol, San Francisco, CA USA Clovis Oncol, San Francisco, CA USAHaringsma, Henry J.论文数: 0 引用数: 0 h-index: 0机构: Clovis Oncol, San Francisco, CA USA Clovis Oncol, San Francisco, CA USAWalter, Annette O.论文数: 0 引用数: 0 h-index: 0机构: Clovis Oncol, San Francisco, CA USA Clovis Oncol, San Francisco, CA USASjin, Robert Tjin Tham论文数: 0 引用数: 0 h-index: 0机构: Celgene Avil Res, Bedford, ME USA Clovis Oncol, San Francisco, CA USAWeaver, Zoe论文数: 0 引用数: 0 h-index: 0机构: NCI Frederick, SAIC Frederick, Ctr Adv Preclin Res, Frederick, MD USA Clovis Oncol, San Francisco, CA USAAllen, Andrew论文数: 0 引用数: 0 h-index: 0机构: Clovis Oncol, San Francisco, CA USA Clovis Oncol, San Francisco, CA USAHarding, Thomas C.论文数: 0 引用数: 0 h-index: 0机构: Clovis Oncol, San Francisco, CA USA Clovis Oncol, San Francisco, CA USA
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