SYNTHETIC STUDIES ON 1,3,4-OXADIAZOLES

被引：0
|
作者：
Sujatha, K. [1 ,2 ]
Khadar, A. M. A. [1 ]
Kalluraya, Balakrishna [1 ]
Babu, M. [1 ]
机构：
[1] Mangalore Univ, Dept Studies Chem, Mangalagangothri 575199, India
[2] SeQuent Sci Ltd, Ind Area, Baikampady, New Mangalore, India
来源：
INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY | 2009年 / 19卷 / 01期
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中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A new series of 5-(alpha-aryloxyethyl)-1,3,4-oxadiazole-2-thiones (4) were prepared and subjected to Mannich reaction in the presence of formaldehyde and appropriate amine. Such reactions resulted in the regioselective formation of 3-aryl aminomethyl-2-thiones (5). The structures of the new compounds have been established by spectral and analytical data. The compounds have been tested for their antimicrobial activity.
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页码：33 / 36
页数：4
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