A one-pot synthesis of tetrahydroisoquinolonic acids from aldehydes and amines in trimethylorthoformate

被引：0
|
作者：
Yu, NF
Poulain, R
Gesquiere, JC
机构：
[1] Fac Pharm, Chim Organ Lab, UMR CNRS 8525, F-59006 Lille, France
[2] CEREP, F-59000 Lille, France
来源：
SYNLETT | 2000年 / 03期
关键词：
cyclization; amines; aldehydes; solvent effect; orthoformate;
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Tetrahydroisoquinolonic acids are synthesized in the presence of excess trimethyl orthoformate by a one-pot procedure directly from the corresponding amines, aldehydes and homophthalic anhydride.
引用
收藏
页码：355 / 356
页数：2
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