Synthesis of Hexahydropyrimidines and 1,2,3,4-Tetrahydropyridines by Reaction of Ethyl Benzoylacetate with Formaldehyde and Primary Amines

被引：4
|
作者：
Kireeva, D. R. [1 ]
Kamalova, A. I. [1 ]
机构：
[1] Russian Acad Sci, Ufa Inst Chem, Ufa Fed Res Ctr, Ufa 450054, Russia
来源：
RUSSIAN JOURNAL OF ORGANIC CHEMISTRY | 2020年 / 56卷 / 10期
关键词：
ethyl benzoylacetate; hexahydropyrimidine; tetrahydropyridine; diethyl; 2; 4-dibenzoylpentanedioate; debenzoylation; one-pot synthesis; multicomponent reactions; ACETOACETATE;
D O I：
10.1134/S1070428020100103
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The reaction of ethyl benzoylacetate with formaldehyde and primary amines in boiling pyridine or methanol afforded new 1,2,3,4-tetrahydropyridine derivatives and substituted hexahydropyrimidines.
引用
收藏
页码：1733 / 1737
页数：5
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