Stereocontrolled synthesis of tricyclic fused oxazolidinone as antibacterial agent

被引：11

作者：

Cui, Yingjie ^{[1
]}

Dang, Yaxian ^{[1
]}

Yang, Yushe ^{[1
]}

Ji, Ruyun ^{[1
]}

机构：

[1] Chinese Acad Sci, Shanghai Inst Biol Sci, Shanghai Inst Mat Med, Shanghai 201203, Peoples R China

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 2006年 / 43卷 / 04期

关键词：

D O I：

10.1002/jhet.5570430438

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Tricyclic fused oxazolidinone 3a and 3b have been synthesized as antibacterial agents in 12 and 11 steps respectively. The key intermediates 10a and 10b have been developed via opening of epoxide 9a and 9b and cyclization by the resulting oxygen anion attack.

引用

页码：1071 / 1075

页数：5

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