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- [1] Design and synthesis of a series of bioavailable fatty acid synthase (FASN) KR domain inhibitors for cancer therapyBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2018, 28 (12) : 2159 - 2164Lu, Tianbao论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USASchubert, Carsten论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USACummings, Maxwell D.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USABignan, Gilles论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USAConnolly, Peter J.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USASmans, Karine论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Turnhoutseweg 30, B-2340 Beerse, Belgium Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USALudovici, Donald论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USAParker, Michael H.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USAMeyer, Christophe论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, CS10615,Campus Maigremont, F-27106 Val De Reuil, France Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USARocaboy, Christian论文数: 0 引用数: 0 h-index: 0机构: Parque Tecnol Fuente Alamo, Villapharma Res, Carretera El Estrecho Lobosillo, Murcia 30320, Spain Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USAAlexander, Richard论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USAGrasberger, Bruce论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USADe Breucker, Sabine论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Turnhoutseweg 30, B-2340 Beerse, Belgium Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USAEsser, Norbert论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Turnhoutseweg 30, B-2340 Beerse, Belgium Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USAFraiponts, Erwin论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Turnhoutseweg 30, B-2340 Beerse, Belgium Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USAGilissen, Ron论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Turnhoutseweg 30, B-2340 Beerse, Belgium Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USAJanssens, Boudewijn论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Turnhoutseweg 30, B-2340 Beerse, Belgium Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USAPeeters, Danielle论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Turnhoutseweg 30, B-2340 Beerse, Belgium Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USAVan Nuffel, Luc论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Turnhoutseweg 30, B-2340 Beerse, Belgium Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USAVermeulen, Peter论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Turnhoutseweg 30, B-2340 Beerse, Belgium Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USABischoff, James论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USAMeerpoel, Lieven论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Turnhoutseweg 30, B-2340 Beerse, Belgium Janssen Res & Dev LLC, 1400 McKean Rd, Spring House, PA 19477 USA
- [2] NOVEL INHIBITORS OF FATTY ACID SYNTHASE (FASN) WITH ANTICANCER ACTIVITYDRUGS OF THE FUTURE, 2009, 34 : 196 - 196Benhamu, Bellinda论文数: 0 引用数: 0 h-index: 0机构: Univ Complutense Madrid, Fac Ciencias Quim, Dept Quim Organ 1, E-28040 Madrid, Spain Univ Complutense Madrid, Fac Ciencias Quim, Dept Quim Organ 1, E-28040 Madrid, SpainTurrado, Carlos论文数: 0 引用数: 0 h-index: 0机构: Univ Complutense Madrid, Fac Ciencias Quim, Dept Quim Organ 1, E-28040 Madrid, Spain Univ Complutense Madrid, Fac Ciencias Quim, Dept Quim Organ 1, E-28040 Madrid, SpainOrtega-Gutierrez, Silvia论文数: 0 引用数: 0 h-index: 0机构: Univ Complutense Madrid, Fac Ciencias Quim, Dept Quim Organ 1, E-28040 Madrid, Spain Univ Complutense Madrid, Fac Ciencias Quim, Dept Quim Organ 1, E-28040 Madrid, SpainPuig, Teresa论文数: 0 引用数: 0 h-index: 0机构: Inst Catala Oncol, E-17007 Girona, Spain Inst Invest Biomed Girona, E-17007 Girona, Spain Univ Complutense Madrid, Fac Ciencias Quim, Dept Quim Organ 1, E-28040 Madrid, SpainRelat, Joana论文数: 0 引用数: 0 h-index: 0机构: Univ Barcelona, Dept Bioquim & Biol Mol, Inst Biomed, E-08028 Barcelona, Spain Univ Complutense Madrid, Fac Ciencias Quim, Dept Quim Organ 1, E-28040 Madrid, SpainCasals, Gemma论文数: 0 引用数: 0 h-index: 0机构: Inst Catala Oncol, E-17007 Girona, Spain Inst Invest Biomed Girona, E-17007 Girona, Spain Univ Complutense Madrid, Fac Ciencias Quim, Dept Quim Organ 1, E-28040 Madrid, SpainOliveras, Glorio论文数: 0 引用数: 0 h-index: 0机构: Inst Catala Oncol, E-17007 Girona, Spain Inst Invest Biomed Girona, E-17007 Girona, Spain Univ Complutense Madrid, Fac Ciencias Quim, Dept Quim Organ 1, E-28040 Madrid, SpainMarrero, Pedro F.论文数: 0 引用数: 0 h-index: 0机构: Univ Barcelona, Dept Bioquim & Biol Mol, Inst Biomed, E-08028 Barcelona, Spain Univ Complutense Madrid, Fac Ciencias Quim, Dept Quim Organ 1, E-28040 Madrid, SpainHaro, Diego论文数: 0 引用数: 0 h-index: 0机构: Univ Barcelona, Dept Bioquim & Biol Mol, Inst Biomed, E-08028 Barcelona, Spain Univ Complutense Madrid, Fac Ciencias Quim, Dept Quim Organ 1, E-28040 Madrid, SpainCufi, Silvia论文数: 0 引用数: 0 h-index: 0机构: Hosp Duran & Reynals, Lab Translac, Inst Catala Oncol, E-08907 Barcelona, Spain Univ Complutense Madrid, Fac Ciencias Quim, Dept Quim Organ 1, E-28040 Madrid, SpainAguilar, Helena论文数: 0 引用数: 0 h-index: 0机构: Hosp Duran & Reynals, Lab Translac, Inst Catala Oncol, E-08907 Barcelona, Spain Univ Complutense Madrid, Fac Ciencias Quim, Dept Quim Organ 1, E-28040 Madrid, SpainUrruticoechea, Ander论文数: 0 引用数: 0 h-index: 0机构: Hosp Duran & Reynals, Lab Translac, Inst Catala Oncol, E-08907 Barcelona, Spain Univ Complutense Madrid, Fac Ciencias Quim, Dept Quim Organ 1, E-28040 Madrid, SpainColomer, Ramon论文数: 0 引用数: 0 h-index: 0机构: Inst Catala Oncol, E-17007 Girona, Spain Inst Invest Biomed Girona, E-17007 Girona, Spain Ctr Oncol MD Anderson Espana, E-28033 Madrid, Spain Univ Complutense Madrid, Fac Ciencias Quim, Dept Quim Organ 1, E-28040 Madrid, SpainLopez-Rodriguez, Maria L.论文数: 0 引用数: 0 h-index: 0机构: Univ Complutense Madrid, Fac Ciencias Quim, Dept Quim Organ 1, E-28040 Madrid, Spain Univ Complutense Madrid, Fac Ciencias Quim, Dept Quim Organ 1, E-28040 Madrid, Spain
- [3] Structure-Based Discovery of Lipoteichoic Acid Synthase InhibitorsJOURNAL OF CHEMICAL INFORMATION AND MODELING, 2022, 62 (10) : 2586 - 2599Wezen, Xavier Chee论文数: 0 引用数: 0 h-index: 0机构: Swinburne Univ Technol Sarawak, Fac Engn Comp & Sci, Sch Chem Engn & Sci, Sci Program, Kuching 93350, Malaysia Swinburne Univ Technol Sarawak, Fac Engn Comp & Sci, Sch Chem Engn & Sci, Sci Program, Kuching 93350, MalaysiaChandran, Aneesh论文数: 0 引用数: 0 h-index: 0机构: Kannur Univ, Dept Biotechnol & Microbiol, Kannur 670661, Kerala, India Swinburne Univ Technol Sarawak, Fac Engn Comp & Sci, Sch Chem Engn & Sci, Sci Program, Kuching 93350, MalaysiaEapen, Rohan Sakariah论文数: 0 引用数: 0 h-index: 0机构: Univ Cambridge, Dept Pharmacol, Cambridge CB2 1PD, England Swinburne Univ Technol Sarawak, Fac Engn Comp & Sci, Sch Chem Engn & Sci, Sci Program, Kuching 93350, MalaysiaWaters, Elaine论文数: 0 引用数: 0 h-index: 0机构: Univ Liverpool, Inst Infect & Global Hlth, Dept Clin Infect Microbiol & Immunol, Liverpool L69 7BE, Merseyside, England Swinburne Univ Technol Sarawak, Fac Engn Comp & Sci, Sch Chem Engn & Sci, Sci Program, Kuching 93350, MalaysiaBricio-Moreno, Laura论文数: 0 引用数: 0 h-index: 0机构: Univ Liverpool, Inst Infect & Global Hlth, Dept Clin Infect Microbiol & Immunol, Liverpool L69 7BE, Merseyside, England Swinburne Univ Technol Sarawak, Fac Engn Comp & Sci, Sch Chem Engn & Sci, Sci Program, Kuching 93350, MalaysiaTosi, Tommaso论文数: 0 引用数: 0 h-index: 0机构: Imperial Coll London, Sect Mol Microbiol, London SW7 2AZ, England Imperial Coll London, MRC Ctr Mol Bacteriol & Infect, London SW7 2AZ, England Swinburne Univ Technol Sarawak, Fac Engn Comp & Sci, Sch Chem Engn & Sci, Sci Program, Kuching 93350, MalaysiaDolan, Stephen论文数: 0 引用数: 0 h-index: 0机构: Univ Cambridge, Dept Biochem, Cambridge CB2 1QW, England Swinburne Univ Technol Sarawak, Fac Engn Comp & Sci, Sch Chem Engn & Sci, Sci Program, Kuching 93350, MalaysiaMillership, Charlotte论文数: 0 引用数: 0 h-index: 0机构: Imperial Coll London, Sect Mol Microbiol, London SW7 2AZ, England Imperial Coll London, MRC Ctr Mol Bacteriol & Infect, London SW7 2AZ, England Swinburne Univ Technol Sarawak, Fac Engn Comp & Sci, Sch Chem Engn & Sci, Sci Program, Kuching 93350, MalaysiaKadioglu, Aras论文数: 0 引用数: 0 h-index: 0机构: Univ Liverpool, Inst Infect & Global Hlth, Dept Clin Infect Microbiol & Immunol, Liverpool L69 7BE, Merseyside, England Swinburne Univ Technol Sarawak, Fac Engn Comp & Sci, Sch Chem Engn & Sci, Sci Program, Kuching 93350, MalaysiaGrundling, Angelika论文数: 0 引用数: 0 h-index: 0机构: Imperial Coll London, Sect Mol Microbiol, London SW7 2AZ, England Imperial Coll London, MRC Ctr Mol Bacteriol & Infect, London SW7 2AZ, England Swinburne Univ Technol Sarawak, Fac Engn Comp & Sci, Sch Chem Engn & Sci, Sci Program, Kuching 93350, MalaysiaItzhaki, Laura S.论文数: 0 引用数: 0 h-index: 0机构: Univ Cambridge, Dept Pharmacol, Cambridge CB2 1PD, England Swinburne Univ Technol Sarawak, Fac Engn Comp & Sci, Sch Chem Engn & Sci, Sci Program, Kuching 93350, MalaysiaWelch, Martin论文数: 0 引用数: 0 h-index: 0机构: Univ Cambridge, Dept Biochem, Cambridge CB2 1QW, England Swinburne Univ Technol Sarawak, Fac Engn Comp & Sci, Sch Chem Engn & Sci, Sci Program, Kuching 93350, MalaysiaRahman, Taufiq论文数: 0 引用数: 0 h-index: 0机构: Univ Cambridge, Dept Pharmacol, Cambridge CB2 1PD, England Swinburne Univ Technol Sarawak, Fac Engn Comp & Sci, Sch Chem Engn & Sci, Sci Program, Kuching 93350, Malaysia
- [4] Structure-based design to improve the selectivity of kinase inhibitors in cancer therapyABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2018, 256Assadieskandar, Amin论文数: 0 引用数: 0 h-index: 0机构: Univ Southern Calif, Los Angeles, CA USA Univ Southern Calif, Los Angeles, CA USAYu, Caiyun论文数: 0 引用数: 0 h-index: 0机构: Univ Southern Calif, Los Angeles, CA USA Univ Southern Calif, Los Angeles, CA USAZhang, Chao论文数: 0 引用数: 0 h-index: 0机构: Univ Southern Calif, Dept Chem, Los Angeles, CA USA Univ Southern Calif, Los Angeles, CA USA
- [5] Fatty acid synthase (FASN) as a therapeutic target in breast cancerEXPERT OPINION ON THERAPEUTIC TARGETS, 2017, 21 (11) : 1001 - 1016Menendez, Javier A.论文数: 0 引用数: 0 h-index: 0机构: Catalan Inst Oncol, Metab & Canc Grp, ProCURE Program Canc Therapeut Resistance, Girona, Spain Girona Biomed Res Inst IDIBGI, Parc Hosp Marti i Julia, Girona 17190, Spain Catalan Inst Oncol, Metab & Canc Grp, ProCURE Program Canc Therapeut Resistance, Girona, SpainLupu, Ruth论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Dept Med & Expt Pathol, Rochester, MN USA Mayo Clin, Ctr Canc, 200 First St SW, Rochester, MN 55905 USA Catalan Inst Oncol, Metab & Canc Grp, ProCURE Program Canc Therapeut Resistance, Girona, Spain
- [6] Structure-Based Design of Bacterial Nitric Oxide Synthase InhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2015, 58 (02) : 994 - 1004Holden, Jeffrey K.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Irvine, Dept Mol Biol & Biochem, Irvine, CA 92697 USA Univ Calif Irvine, Dept Pharmaceut Sci, Irvine, CA 92697 USA Univ Calif Irvine, Dept Chem, Irvine, CA 92697 USA Univ Calif Irvine, Dept Mol Biol & Biochem, Irvine, CA 92697 USAKang, Soosung论文数: 0 引用数: 0 h-index: 0机构: Northwestern Univ, Dept Chem, Chem Life Proc Inst, Ctr Mol Innovat & Drug Discovery, Evanston, IL 60208 USA Northwestern Univ, Dept Mol Biosci, Chem Life Proc Inst, Ctr Mol Innovat & Drug Discovery, Evanston, IL 60208 USA Univ Calif Irvine, Dept Mol Biol & Biochem, Irvine, CA 92697 USAHollingsworth, Scott A.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Irvine, Dept Mol Biol & Biochem, Irvine, CA 92697 USA Univ Calif Irvine, Dept Pharmaceut Sci, Irvine, CA 92697 USA Univ Calif Irvine, Dept Chem, Irvine, CA 92697 USA Univ Calif Irvine, Dept Mol Biol & Biochem, Irvine, CA 92697 USALi, Huiying论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Irvine, Dept Mol Biol & Biochem, Irvine, CA 92697 USA Univ Calif Irvine, Dept Pharmaceut Sci, Irvine, CA 92697 USA Univ Calif Irvine, Dept Chem, Irvine, CA 92697 USA Univ Calif Irvine, Dept Mol Biol & Biochem, Irvine, CA 92697 USALim, Nathan论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Irvine, Dept Mol Biol & Biochem, Irvine, CA 92697 USA Univ Calif Irvine, Dept Pharmaceut Sci, Irvine, CA 92697 USA Univ Calif Irvine, Dept Chem, Irvine, CA 92697 USA Univ Calif Irvine, Dept Mol Biol & Biochem, Irvine, CA 92697 USAChen, Steven论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Irvine, Dept Mol Biol & Biochem, Irvine, CA 92697 USA Univ Calif Irvine, Dept Pharmaceut Sci, Irvine, CA 92697 USA Univ Calif Irvine, Dept Chem, Irvine, CA 92697 USA Univ Calif Irvine, Dept Mol Biol & Biochem, Irvine, CA 92697 USAHuang, He论文数: 0 引用数: 0 h-index: 0机构: Northwestern Univ, Dept Chem, Chem Life Proc Inst, Ctr Mol Innovat & Drug Discovery, Evanston, IL 60208 USA Northwestern Univ, Dept Mol Biosci, Chem Life Proc Inst, Ctr Mol Innovat & Drug Discovery, Evanston, IL 60208 USA Univ Calif Irvine, Dept Mol Biol & Biochem, Irvine, CA 92697 USAXue, Fengtian论文数: 0 引用数: 0 h-index: 0机构: Northwestern Univ, Dept Chem, Chem Life Proc Inst, Ctr Mol Innovat & Drug Discovery, Evanston, IL 60208 USA Northwestern Univ, Dept Mol Biosci, Chem Life Proc Inst, Ctr Mol Innovat & Drug Discovery, Evanston, IL 60208 USA Univ Calif Irvine, Dept Mol Biol & Biochem, Irvine, CA 92697 USATang, Wei论文数: 0 引用数: 0 h-index: 0机构: Northwestern Univ, Dept Chem, Chem Life Proc Inst, Ctr Mol Innovat & Drug Discovery, Evanston, IL 60208 USA Northwestern Univ, Dept Mol Biosci, Chem Life Proc Inst, Ctr Mol Innovat & Drug Discovery, Evanston, IL 60208 USA Univ Calif Irvine, Dept Mol Biol & Biochem, Irvine, CA 92697 USASilverman, Richard B.论文数: 0 引用数: 0 h-index: 0机构: Northwestern Univ, Dept Chem, Chem Life Proc Inst, Ctr Mol Innovat & Drug Discovery, Evanston, IL 60208 USA Northwestern Univ, Dept Mol Biosci, Chem Life Proc Inst, Ctr Mol Innovat & Drug Discovery, Evanston, IL 60208 USA Univ Calif Irvine, Dept Mol Biol & Biochem, Irvine, CA 92697 USAPoulos, Thomas L.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Irvine, Dept Mol Biol & Biochem, Irvine, CA 92697 USA Univ Calif Irvine, Dept Pharmaceut Sci, Irvine, CA 92697 USA Univ Calif Irvine, Dept Chem, Irvine, CA 92697 USA Univ Calif Irvine, Dept Mol Biol & Biochem, Irvine, CA 92697 USA
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