Tripeptide methylketones: Synthesis and antiplasmin activity

被引：0
|
作者：
MiduraNowaczek, K [1 ]
Bruzgo, I [1 ]
RoszkowskaJakimiec, W [1 ]
Worowski, K [1 ]
机构：
[1] AKAD MED BIALYMSTOKU,ZAKLAD ANALIZY INSTRUMENTALNEJ,PL-15230 BIALYSTOK,POLAND
来源：
FARMACO | 1997年 / 52卷 / 01期
关键词：
D O I：
暂无
中图分类号：
R9 [药学];
学科分类号：
1007 ;
摘要：
A series of tripeptide methylketones with C-terminal lysine was obtained via Dakin-West method and tested for their antiplasmin activity with the use of antifibrinolytic and antiamidolytic tests. The tripeptide methylketones has been found to inhibit plasmin, however with much lower potency than respective aldehydes.
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收藏
页码：35 / 37
页数：3
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