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- [1] Development of novel Btk inhibitor, CB988 targering ibrutinib-resistant Btk C481S mutant[J]. CANCER RESEARCH, 2017, 77Kawahata, Wataru论文数: 0 引用数: 0 h-index: 0Asami, Tokiko论文数: 0 引用数: 0 h-index: 0Irie, Takayuki论文数: 0 引用数: 0 h-index: 0Iwata, Yasuhiro论文数: 0 引用数: 0 h-index: 0Kiyoi, Takao论文数: 0 引用数: 0 h-index: 0Sawa, Masaaki论文数: 0 引用数: 0 h-index: 0
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BLOOD ADVANCES, 2023, 7 (09) : 1929 - 1943论文数: 引用数: h-index:机构:Utro, Filippo论文数: 0 引用数: 0 h-index: 0机构: IBM Res, New York, NY 10598 USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USAWang, Qing论文数: 0 引用数: 0 h-index: 0机构: Karolinska Univ Hosp Huddinge, Karolinska Inst, Dept Lab Med Biomol & Cellular Med, SE-14186 Huddinge, Sweden Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USACha, Justin论文数: 0 引用数: 0 h-index: 0机构: Broad Inst Massachusetts Inst Technol & Harvard, Canc Program, Cambridge, MA 02142 USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USAVihinen, Mauno论文数: 0 引用数: 0 h-index: 0机构: Lund Univ, Dept Expt Med Sci, SE-22184 Lund, Sweden Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USAMartindale, Stephen论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USAZhou, Yinglu论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Harvard TH Chan Sch Publ Hlth, Dana Farber Canc Inst, Dept Data Sci, Boston, MA USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USARen, Yue论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Harvard TH Chan Sch Publ Hlth, Dana Farber Canc Inst, Dept Data Sci, Boston, MA USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USATyekucheva, Svitlana论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Harvard TH Chan Sch Publ Hlth, Dana Farber Canc Inst, Dept Data Sci, Boston, MA USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USAKim, Annette S.论文数: 0 引用数: 0 h-index: 0机构: Brigham & Womens Hosp, Dept Pathol, Boston, MA USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USAFernandes, Stacey M.论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USASaksena, Gordon论文数: 0 引用数: 0 h-index: 0机构: Broad Inst Massachusetts Inst Technol & Harvard, Canc Program, Cambridge, MA 02142 USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USARhrissorrakrai, Kahn论文数: 0 引用数: 0 h-index: 0机构: IBM Res, New York, NY 10598 USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USALevovitz, Chaya论文数: 0 引用数: 0 h-index: 0机构: IBM Res, New York, NY 10598 USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USADanysh, Brian P.论文数: 0 引用数: 0 h-index: 0机构: Broad Inst Massachusetts Inst Technol & Harvard, Canc Program, Cambridge, MA 02142 USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USASlowik, Kara论文数: 0 引用数: 0 h-index: 0机构: Broad Inst Massachusetts Inst Technol & Harvard, Canc Program, Cambridge, MA 02142 USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USAJacobs, Raquel A.论文数: 0 引用数: 0 h-index: 0机构: Broad Inst Massachusetts Inst Technol & Harvard, Canc Program, Cambridge, MA 02142 USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USADavids, Matthew S.论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA Brigham & Womens Hosp, Dept Med, Boston, MA 02115 USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USALederer, James A.论文数: 0 引用数: 0 h-index: 0机构: Brigham & Womens Hosp, Dept Surg, Boston, MA USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USAZain, Rula论文数: 0 引用数: 0 h-index: 0机构: Karolinska Univ Hosp Huddinge, Karolinska Inst, Dept Lab Med Biomol & Cellular Med, SE-14186 Huddinge, Sweden Karolinska Univ Hosp, Ctr Rare Dis, Dept Clin Genet, SE-17176 Stockholm, Sweden Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USASmith, C. I. Edvard论文数: 0 引用数: 0 h-index: 0机构: Karolinska Univ Hosp Huddinge, Karolinska Inst, Dept Lab Med Biomol & Cellular Med, SE-14186 Huddinge, Sweden Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USALeshchiner, Ignaty论文数: 0 引用数: 0 h-index: 0机构: Broad Inst Massachusetts Inst Technol & Harvard, Canc Program, Cambridge, MA 02142 USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USAParida, Laxmi论文数: 0 引用数: 0 h-index: 0机构: IBM Res, New York, NY 10598 USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USAGetz, Gad论文数: 0 引用数: 0 h-index: 0机构: Broad Inst Massachusetts Inst Technol & Harvard, Canc Program, Cambridge, MA 02142 USA Harvard Med Sch, Dept Pathol, Boston, MA USA Massachusetts Gen Hosp, Canc Ctr, Boston, MA USA Massachusetts Gen Hosp, Dept Pathol, Boston, MA USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USABrown, Jennifer R.论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA Brigham & Womens Hosp, Dept Med, Boston, MA 02115 USA Harvard Med Sch, Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA
- [3] PROTAC-induced BTK degradation as a novel therapy for mutated BTK C481S induced ibrutinib-resistant B-cell malignancies[J]. CELL RESEARCH, 2018, 28 (07) : 779 - 781Sun, Yonghui论文数: 0 引用数: 0 h-index: 0机构: Tsinghua Univ, Sch Pharmaceut Sci, MOE Key Lab Prot Sci, MOE Key Lab Bioorgan Phosphorus Chem & Chem Biol, Beijing 100084, Peoples R China Tsinghua Univ, Sch Pharmaceut Sci, MOE Key Lab Prot Sci, MOE Key Lab Bioorgan Phosphorus Chem & Chem Biol, Beijing 100084, Peoples R ChinaZhao, Xingwang论文数: 0 引用数: 0 h-index: 0机构: Tsinghua Univ, Beijing Key Lab Immunol Res Chron Dis, Sch Life Sci,MOE Key Lab Prot Sci, Collaborat Innovat Ctr Diag & Treatment Infect Di, Beijing 100084, Peoples R China Tsinghua Univ, Sch Pharmaceut Sci, MOE Key Lab Prot Sci, MOE Key Lab Bioorgan Phosphorus Chem & Chem Biol, Beijing 100084, Peoples R ChinaDing, Ning论文数: 0 引用数: 0 h-index: 0机构: Peking Univ, Dept Lymphoma, Key Lab Carcinogenesis & Translat Res, Minist Educ,Canc Hosp & Inst, 52 Fucheng Rd, Beijing 100142, Peoples R China Tsinghua Univ, Sch Pharmaceut Sci, MOE Key Lab Prot Sci, MOE Key Lab Bioorgan Phosphorus Chem & Chem Biol, Beijing 100084, Peoples R ChinaGao, Hongying论文数: 0 引用数: 0 h-index: 0机构: Tsinghua Univ, Sch Pharmaceut Sci, MOE Key Lab Prot Sci, MOE Key Lab Bioorgan Phosphorus Chem & Chem Biol, Beijing 100084, Peoples R China Tsinghua Univ, Beijing Key Lab Immunol Res Chron Dis, Sch Life Sci,MOE Key Lab Prot Sci, Collaborat Innovat Ctr Diag & Treatment Infect Di, Beijing 100084, Peoples R China Tsinghua Univ, Sch Pharmaceut Sci, MOE Key Lab Prot Sci, MOE Key Lab Bioorgan Phosphorus Chem & Chem Biol, Beijing 100084, Peoples R ChinaWu, Yue论文数: 0 引用数: 0 h-index: 0机构: Tsinghua Univ, Sch Pharmaceut Sci, MOE Key Lab Prot Sci, MOE Key Lab Bioorgan Phosphorus Chem & Chem Biol, Beijing 100084, Peoples R China Tsinghua Univ, Sch Pharmaceut Sci, MOE Key Lab Prot Sci, MOE Key Lab Bioorgan Phosphorus Chem & Chem Biol, Beijing 100084, Peoples R ChinaYang, Yiqing论文数: 0 引用数: 0 h-index: 0机构: Tsinghua Univ, Sch Pharmaceut Sci, MOE Key Lab Prot Sci, MOE Key Lab Bioorgan Phosphorus Chem & Chem Biol, Beijing 100084, Peoples R China Tsinghua Univ, Sch Pharmaceut Sci, MOE Key Lab Prot Sci, MOE Key Lab Bioorgan Phosphorus Chem & Chem Biol, Beijing 100084, Peoples R ChinaZhao, Meng论文数: 0 引用数: 0 h-index: 0机构: Tsinghua Univ, Beijing Key Lab Immunol Res Chron Dis, Sch Life Sci,MOE Key Lab Prot Sci, Collaborat Innovat Ctr Diag & Treatment Infect Di, Beijing 100084, Peoples R China Tsinghua Univ, Sch Pharmaceut Sci, MOE Key Lab Prot Sci, MOE Key Lab Bioorgan Phosphorus Chem & Chem Biol, Beijing 100084, Peoples R ChinaHwang, Jinseok论文数: 0 引用数: 0 h-index: 0机构: Tsinghua Univ, Beijing Key Lab Immunol Res Chron Dis, Sch Life Sci,MOE Key Lab Prot Sci, Collaborat Innovat Ctr Diag & Treatment Infect Di, Beijing 100084, Peoples R China Tsinghua Univ, Sch Pharmaceut Sci, MOE Key Lab Prot Sci, MOE Key Lab Bioorgan Phosphorus Chem & Chem Biol, Beijing 100084, Peoples R ChinaSong, Yuqin论文数: 0 引用数: 0 h-index: 0机构: Peking Univ, Dept Lymphoma, Key Lab Carcinogenesis & Translat Res, Minist Educ,Canc Hosp & Inst, 52 Fucheng Rd, Beijing 100142, Peoples R China Tsinghua Univ, Sch Pharmaceut Sci, MOE Key Lab Prot Sci, MOE Key Lab Bioorgan Phosphorus Chem & Chem Biol, Beijing 100084, Peoples R ChinaLiu, Wanli论文数: 0 引用数: 0 h-index: 0机构: Tsinghua Univ, Beijing Key Lab Immunol Res Chron Dis, Sch Life Sci,MOE Key Lab Prot Sci, Collaborat Innovat Ctr Diag & Treatment Infect Di, Beijing 100084, Peoples R China Tsinghua Univ, Sch Pharmaceut Sci, MOE Key Lab Prot Sci, MOE Key Lab Bioorgan Phosphorus Chem & Chem Biol, Beijing 100084, Peoples R ChinaRao, Yu论文数: 0 引用数: 0 h-index: 0机构: Tsinghua Univ, Sch Pharmaceut Sci, MOE Key Lab Prot Sci, MOE Key Lab Bioorgan Phosphorus Chem & Chem Biol, Beijing 100084, Peoples R China Tsinghua Univ, Sch Pharmaceut Sci, MOE Key Lab Prot Sci, MOE Key Lab Bioorgan Phosphorus Chem & Chem Biol, Beijing 100084, Peoples R China
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