One pot direct synthesis of oxazolines, benzoxazoles, and oxadiazoles from carboxylic acids using the Deoxo-Fluor reagent

被引:88
|
作者
Kangani, Cyrous O. [1 ]
Kelley, David E. [1 ]
Day, Billy W. [1 ]
机构
[1] Univ Pittsburgh, Dept Med, Pittsburgh, PA 15213 USA
基金
美国国家卫生研究院;
关键词
D O I
10.1016/j.tetlet.2006.07.032
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
A one-pot, high yield direct synthesis of various 2-substituted oxazolines, benzoxazoles, and 2-oxadiazoles from carboxylic acids using Deoxo-Fluor reagent is described. (c) 2006 Elsevier Ltd. All rights reserved.
引用
收藏
页码:6497 / 6499
页数:3
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