Synthesis and Biological Activity of Substituted 1,2,4-Triazolo[1,5-c]pyrimidine Derivatives

被引：0

作者：

Chen, Chaonan ^{[1
]}

Chen, Qiong ^{[1
]}

Yang, Guangfu ^{[1
]}

机构：

[1] Cent China Normal Univ, Coll Chem, Educ Minist, Key Lab Pesticide & Chem Biol, Wuhan 430079, Peoples R China

来源：

CHINESE JOURNAL OF ORGANIC CHEMISTRY | 2009年 / 29卷 / 02期

关键词：

1,2,4-triazolo[1,5-c]pyrimidine; synthesis; biological activity;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Sixteen novel 2-[substituted benzyloxy 7-chloro-5-methylsulfanyl-[1,2,4]-triazolo[1,5-c] pyrimidine derivatives and thirty-six novel substituted 2-phenoxy-[1,2,4]-triazolo[1,5-c]pyrimidine derivatives have been designed and synthesized using substituted 4-hydrazinopyrimidine as starting material. All synthesized compounds were confirmed by elemental analysis, MS and H-1 NMR techniques. Preliminary bioassay indicates that some of them display good herbicidal and fungicidal activities.

引用

页码：245 / 251

页数：7

共 13 条

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