Changing Classical Pharmacology by Exploring the Allosteric Mechanisms of Caffeine Within the Adenosine A2A-Dopamine D2 Receptor Heterotetramer

被引:0
|
作者
Ferre, Sergi [1 ]
机构
[1] NIDA, Baltimore, MD USA
关键词
D O I
暂无
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
31.2
引用
收藏
页码:S54 / S54
页数:1
相关论文
共 50 条
  • [1] Allosteric mechanisms within the adenosine A2A -dopamine D2 receptor heterotetramer
    Ferre, Sergi
    Bonaventura, Jordi
    Tomasi, Dardo
    Navarro, Gemma
    Moreno, Estefania
    Cortes, Antonio
    Lluis, Carme
    Casado, Vicent
    Volkow, Nora D.
    [J]. NEUROPHARMACOLOGY, 2016, 104 : 154 - 160
  • [2] Allosteric interactions between agonists and antagonists within the adenosine A2A receptor-dopamine D2 receptor heterotetramer
    Bonaventura, Jordi
    Navarro, Gemma
    Casado-Anguera, Veronica
    Azdad, Karima
    Rea, William
    Moreno, Estefania
    Brugarolas, Marc
    Mallol, Josefa
    Canela, Enric I.
    Lluis, Carme
    Cortes, Antoni
    Volkow, Nora D.
    Schiffmann, Serge N.
    Ferre, Sergi
    Casado, Vicent
    [J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2015, 112 (27) : E3609 - E3618
  • [3] Adenosine A2A-dopamine D2 receptor heteromers in schizophrenia
    Ciruela, F.
    Lopez-Cano, M.
    Callado, L.
    Aso, E.
    Contreras, F.
    Altafaj, X.
    Masahiko, M.
    Fernandez-Duenas, V.
    Menchon, Jose. M.
    Valle-Leon, M.
    [J]. JOURNAL OF NEUROCHEMISTRY, 2019, 150 : 179 - 179
  • [4] Heterobivalent Ligand for the Adenosine A2A-Dopamine D2 Receptor Heteromer
    Pulido, Daniel
    Casado-Anguera, Veronica
    Gomez-Autet, Marc
    Llopart, Natalia
    Moreno, Estefania
    Casajuana-Martin, Nil
    Ferre, Sergi
    Pardo, Leonardo
    Casado, Vicent
    Royo, Miriam
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 2022, 65 (01) : 616 - 632
  • [5] Unique effect of clozapine on adenosine A2A-dopamine D2 receptor heteromerization
    Valle-Leon, Marta
    Casajuana-Martin, Nil
    del Torrent, Claudia Llinas
    Argerich, Josep
    Gomez-Acero, Laura
    Sahlholm, Kristoffer
    Ferre, Sergi
    Pardo, Leonardo
    Ciruela, Francisco
    [J]. BIOMEDICINE & PHARMACOTHERAPY, 2023, 160
  • [6] Evidence for the heterotetrameric structure of the adenosine A2A-dopamine D2 receptor complex
    Casado-Anguera, Veronica
    Bonaventura, Jordi
    Moreno, Estefania
    Navarro, Gemma
    Cortes, Antoni
    Ferre, Sergi
    Casado, Vicent
    [J]. BIOCHEMICAL SOCIETY TRANSACTIONS, 2016, 44 : 595 - 600
  • [7] Decreased striatal adenosine A2A-dopamine D2 receptor heteromerization in schizophrenia
    Marta Valle-León
    Luis F. Callado
    Ester Aso
    María M. Cajiao-Manrique
    Kristoffer Sahlholm
    Marc López-Cano
    Concepció Soler
    Xavier Altafaj
    Masahiko Watanabe
    Sergi Ferré
    Víctor Fernández-Dueñas
    José M. Menchón
    Francisco Ciruela
    [J]. Neuropsychopharmacology, 2021, 46 : 665 - 672
  • [8] Behavioral control by striatal adenosine A2A-dopamine D2 receptor heteromers
    Taura, J.
    Valle-Leon, M.
    Sahlholm, K.
    Watanabe, M.
    Van Craenenbroeck, K.
    Fernandez-Duenas, V.
    Ferre, S.
    Ciruela, F.
    [J]. GENES BRAIN AND BEHAVIOR, 2018, 17 (04)
  • [9] ILLUMINATING THE ADENOSINE A2A-DOPAMINE D2 RECEPTOR OLIGOMER IN PARKINSON'S DISEASE
    Fernandez-Duenas, V
    Taura, J.
    Jacobson, K. A.
    Ferre, S.
    Ciruela, F.
    [J]. BASIC & CLINICAL PHARMACOLOGY & TOXICOLOGY, 2018, 123 : 18 - 18
  • [10] Adenosine A2A-dopamine D2 receptor-receptor interaction in neurons and astrocytes: Evidence and perspectives
    Guidolin, Diego
    Marcoli, Manuela
    Tortorella, Cinzia
    Maura, Guido
    Agnati, Luigi F.
    [J]. OLIGOMERIZATION IN HEALTH AND DISEASE: FROM ENZYMES TO G PROTEIN-COUPLED RECEPTORS, 2020, 169 : 247 - 277