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- [1] Fragment-Based Discovery of 6-Arylindazole JAK InhibitorsACS MEDICINAL CHEMISTRY LETTERS, 2016, 7 (06): : 641 - 646Ritzen, Andreas论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, Global R&D, Drug Design, Ind Pk 55, DK-2750 Ballerup, Denmark LEO Pharma AS, Global R&D, Drug Design, Ind Pk 55, DK-2750 Ballerup, DenmarkSorensen, Morten D.论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, Global R&D, Drug Design, Ind Pk 55, DK-2750 Ballerup, Denmark LEO Pharma AS, Global R&D, Drug Design, Ind Pk 55, DK-2750 Ballerup, DenmarkDack, Kevin N.论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, Global R&D, Drug Design, Ind Pk 55, DK-2750 Ballerup, Denmark LEO Pharma AS, Global R&D, Drug Design, Ind Pk 55, DK-2750 Ballerup, DenmarkGreve, Daniel R.论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, Global R&D, Drug Design, Ind Pk 55, DK-2750 Ballerup, Denmark LEO Pharma AS, Global R&D, Drug Design, Ind Pk 55, DK-2750 Ballerup, DenmarkJerre, Anders论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, Global R&D, In Vitro Biol, Ind Pk 55, DK-2750 Ballerup, Denmark LEO Pharma AS, Global R&D, Drug Design, Ind Pk 55, DK-2750 Ballerup, DenmarkCarnerup, Martin A.论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, Global R&D, Drug Design, Ind Pk 55, DK-2750 Ballerup, Denmark LEO Pharma AS, Global R&D, Drug Design, Ind Pk 55, DK-2750 Ballerup, DenmarkRytved, Klaus A.论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, Global R&D, Skin PK & Early Safety, Ind Pk 55, DK-2750 Ballerup, Denmark LEO Pharma AS, Global R&D, Drug Design, Ind Pk 55, DK-2750 Ballerup, DenmarkBagger-Bahnsen, Jesper论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, Global R&D, Preformulat & Early Analyt Dev, Ind Pk 55, DK-2750 Ballerup, Denmark LEO Pharma AS, Global R&D, Drug Design, Ind Pk 55, DK-2750 Ballerup, Denmark
- [2] Fragment-based discovery of JAK-2 inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009, 19 (01) : 279 - 282Antonysamy, Stephen论文数: 0 引用数: 0 h-index: 0机构: SGX Pharmaceut Inc, Med Chem, San Diego, CA 92121 USA SGX Pharmaceut Inc, Med Chem, San Diego, CA 92121 USAHirst, Gavin论文数: 0 引用数: 0 h-index: 0机构: SGX Pharmaceut Inc, Med Chem, San Diego, CA 92121 USA SGX Pharmaceut Inc, Med Chem, San Diego, CA 92121 USAPark, Frances论文数: 0 引用数: 0 h-index: 0机构: SGX Pharmaceut Inc, Med Chem, San Diego, CA 92121 USA SGX Pharmaceut Inc, Med Chem, San Diego, CA 92121 USASprengeler, Paul论文数: 0 引用数: 0 h-index: 0机构: SGX Pharmaceut Inc, Med Chem, San Diego, CA 92121 USA SGX Pharmaceut Inc, Med Chem, San Diego, CA 92121 USAStappenbeck, Frank论文数: 0 引用数: 0 h-index: 0机构: SGX Pharmaceut Inc, Med Chem, San Diego, CA 92121 USA SGX Pharmaceut Inc, Med Chem, San Diego, CA 92121 USASteensma, Ruo论文数: 0 引用数: 0 h-index: 0机构: SGX Pharmaceut Inc, Med Chem, San Diego, CA 92121 USA SGX Pharmaceut Inc, Med Chem, San Diego, CA 92121 USAWilson, Mark论文数: 0 引用数: 0 h-index: 0机构: SGX Pharmaceut Inc, Med Chem, San Diego, CA 92121 USA SGX Pharmaceut Inc, Med Chem, San Diego, CA 92121 USAWong, Melissa论文数: 0 引用数: 0 h-index: 0机构: SGX Pharmaceut Inc, Med Chem, San Diego, CA 92121 USA SGX Pharmaceut Inc, Med Chem, San Diego, CA 92121 USA
- [3] Fragment-based discovery of pyrazolopyridones as JAK1 inhibitors with excellent subtype selectivityABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2018, 256Ritzen, Andreas论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, Ballerup, Denmark LEO Pharma AS, Ballerup, DenmarkVifian, Thomas论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, Ballerup, Denmark LEO Pharma AS, Ballerup, DenmarkSindet, Rikke论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, Ballerup, Denmark LEO Pharma AS, Ballerup, DenmarkHansen, Bettina论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, Ballerup, Denmark LEO Pharma AS, Ballerup, DenmarkLarsen, Mogens论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, Ballerup, Denmark LEO Pharma AS, Ballerup, DenmarkJepsen, Tue论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, Ballerup, Denmark LEO Pharma AS, Ballerup, DenmarkLarsen, Jens论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, Ballerup, Denmark LEO Pharma AS, Ballerup, DenmarkSeitzberg, Jimmi论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, Ballerup, Denmark LEO Pharma AS, Ballerup, DenmarkRai, Sanjay论文数: 0 引用数: 0 h-index: 0机构: GVK BIO, Hyderabad, India LEO Pharma AS, Ballerup, DenmarkNasipireddy, Venkatarathnam论文数: 0 引用数: 0 h-index: 0机构: GVK BIO, Hyderabad, India LEO Pharma AS, Ballerup, DenmarkCarnerup, Martin论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, Ballerup, Denmark LEO Pharma AS, Ballerup, DenmarkJerre, Anders论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, Ballerup, Denmark LEO Pharma AS, Ballerup, DenmarkMolck, Christina论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, Ballerup, Denmark LEO Pharma AS, Ballerup, Denmark
- [4] Fragment-Based Discovery of Pyrazolopyridones as JAK1 Inhibitors with Excellent Subtype SelectivityJOURNAL OF MEDICINAL CHEMISTRY, 2020, 63 (13) : 7008 - 7032Hansen, Bettina Borreschmidt论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, MedChem 2, DK-2750 Ballerup, Denmark LEO Pharma AS, MedChem 2, DK-2750 Ballerup, DenmarkJepsen, Tue Heesgaard论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, MedChem 2, DK-2750 Ballerup, Denmark LEO Pharma AS, MedChem 2, DK-2750 Ballerup, DenmarkLarsen, Mogens论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, MedChem 2, DK-2750 Ballerup, Denmark LEO Pharma AS, MedChem 2, DK-2750 Ballerup, DenmarkSindet, Rikke论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, MedChem 2, DK-2750 Ballerup, Denmark LEO Pharma AS, MedChem 2, DK-2750 Ballerup, DenmarkVifian, Thomas论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, MedChem 2, DK-2750 Ballerup, Denmark LEO Pharma AS, MedChem 2, DK-2750 Ballerup, DenmarkBurhardt, Mia Norreskov论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, MedChem 2, DK-2750 Ballerup, Denmark LEO Pharma AS, MedChem 2, DK-2750 Ballerup, DenmarkLarsen, Jens论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, MedChem 2, DK-2750 Ballerup, Denmark LEO Pharma AS, MedChem 2, DK-2750 Ballerup, DenmarkSeitzberg, Jimmi Gerner论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, MedChem 2, DK-2750 Ballerup, Denmark LEO Pharma AS, MedChem 2, DK-2750 Ballerup, DenmarkCarnerup, Martin A.论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, DMPK, DK-2750 Ballerup, Denmark LEO Pharma AS, MedChem 2, DK-2750 Ballerup, DenmarkJerre, Anders论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, Skin Res, DK-2750 Ballerup, Denmark LEO Pharma AS, MedChem 2, DK-2750 Ballerup, DenmarkMolck, Christina论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, Skin Res, DK-2750 Ballerup, Denmark LEO Pharma AS, MedChem 2, DK-2750 Ballerup, DenmarkLovato, Paola论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, Skin Res, DK-2750 Ballerup, Denmark LEO Pharma AS, MedChem 2, DK-2750 Ballerup, DenmarkRai, Sanjay论文数: 0 引用数: 0 h-index: 0机构: GVK Biosci Private Ltd, Med Chem, Hyderabad 500076, India LEO Pharma AS, MedChem 2, DK-2750 Ballerup, DenmarkNasipireddy, Venkatarathnam Reddy论文数: 0 引用数: 0 h-index: 0机构: GVK Biosci Private Ltd, Med Chem, Hyderabad 500076, India LEO Pharma AS, MedChem 2, DK-2750 Ballerup, DenmarkRitzen, Andreas论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, MedChem 2, DK-2750 Ballerup, Denmark LEO Pharma AS, MedChem 2, DK-2750 Ballerup, Denmark
- [5] Fragment-Based Approaches to the Discovery of Kinase InhibitorsPROTEIN KINASE INHIBITORS IN RESEARCH AND MEDICINE, 2014, 548 : 69 - 92Mortenson, Paul N.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandBerdini, Valerio论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandO'Reilly, Marc论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, England
- [6] Fragment-Based Drug Discovery of Phosphodiesterase InhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2018, 61 (04) : 1415 - 1424Svensson, Fredrik论文数: 0 引用数: 0 h-index: 0机构: IOTA Pharmaceut, St Johns Innovat Ctr, Cowley Rd, Cambridge CB4 0WS, England Univ Cambridge, Dept Chem, Ctr Mol Informat, Lensfield Rd, Cambridge CB2 1EW, England IOTA Pharmaceut, St Johns Innovat Ctr, Cowley Rd, Cambridge CB4 0WS, EnglandBender, Andreas论文数: 0 引用数: 0 h-index: 0机构: Univ Cambridge, Dept Chem, Ctr Mol Informat, Lensfield Rd, Cambridge CB2 1EW, England IOTA Pharmaceut, St Johns Innovat Ctr, Cowley Rd, Cambridge CB4 0WS, EnglandBailey, David论文数: 0 引用数: 0 h-index: 0机构: IOTA Pharmaceut, St Johns Innovat Ctr, Cowley Rd, Cambridge CB4 0WS, England IOTA Pharmaceut, St Johns Innovat Ctr, Cowley Rd, Cambridge CB4 0WS, England
- [7] Fragment-Based Discovery of 6-Azaindazoles As Inhibitors of Bacterial DNA LigaseACS MEDICINAL CHEMISTRY LETTERS, 2013, 4 (12): : 1208 - 1212Howard, Steven论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge CB4 0QA, England Astex Pharmaceut Inc, Cambridge CB4 0QA, EnglandAmin, Nader论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge CB4 0QA, England Astex Pharmaceut Inc, Cambridge CB4 0QA, EnglandBenowitz, Andrew B.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSrnithKline, Infect Dis TAU, Collegeville, PA 19426 USA Astex Pharmaceut Inc, Cambridge CB4 0QA, EnglandChiarparin, Elisabetta论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge CB4 0QA, England Astex Pharmaceut Inc, Cambridge CB4 0QA, EnglandCui, Haifeng论文数: 0 引用数: 0 h-index: 0机构: GlaxoSrnithKline, Infect Dis TAU, Collegeville, PA 19426 USA Astex Pharmaceut Inc, Cambridge CB4 0QA, EnglandDeng, Xiaodong论文数: 0 引用数: 0 h-index: 0机构: GlaxoSrnithKline, Infect Dis TAU, Collegeville, PA 19426 USA Astex Pharmaceut Inc, Cambridge CB4 0QA, EnglandHeightman, Tom D.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge CB4 0QA, England Astex Pharmaceut Inc, Cambridge CB4 0QA, EnglandHolmes, David J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSrnithKline, Infect Dis TAU, Collegeville, PA 19426 USA Astex Pharmaceut Inc, Cambridge CB4 0QA, EnglandHopkins, Anna论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge CB4 0QA, England Astex Pharmaceut Inc, Cambridge CB4 0QA, EnglandHuang, Jianzhong论文数: 0 引用数: 0 h-index: 0机构: GlaxoSrnithKline, Infect Dis TAU, Collegeville, PA 19426 USA Astex Pharmaceut Inc, Cambridge CB4 0QA, EnglandJin, Qi论文数: 0 引用数: 0 h-index: 0机构: GlaxoSrnithKline, Infect Dis TAU, Collegeville, PA 19426 USA Astex Pharmaceut Inc, Cambridge CB4 0QA, EnglandKreatsoulas, Constantine论文数: 0 引用数: 0 h-index: 0机构: GlaxoSrnithKline, Infect Dis TAU, Collegeville, PA 19426 USA Astex Pharmaceut Inc, Cambridge CB4 0QA, EnglandMartin, Agnes C. L.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge CB4 0QA, England Astex Pharmaceut Inc, Cambridge CB4 0QA, EnglandMassey, Frances论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge CB4 0QA, England Astex Pharmaceut Inc, Cambridge CB4 0QA, EnglandMcCloskey, Lynn论文数: 0 引用数: 0 h-index: 0机构: GlaxoSrnithKline, Infect Dis TAU, Collegeville, PA 19426 USA Astex Pharmaceut Inc, Cambridge CB4 0QA, EnglandMortenson, Paul N.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge CB4 0QA, England Astex Pharmaceut Inc, Cambridge CB4 0QA, EnglandPathuri, Puja论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge CB4 0QA, England Astex Pharmaceut Inc, Cambridge CB4 0QA, EnglandTisi, Dominic论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge CB4 0QA, England Astex Pharmaceut Inc, Cambridge CB4 0QA, EnglandWilliams, Pamela A.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge CB4 0QA, England Astex Pharmaceut Inc, Cambridge CB4 0QA, England
- [8] Fragment-based discovery of the first known inhibitors of PHGDHABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2015, 250Fuller, Nathan论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Chem Innovat Ctr, Somerville, MA USA AstraZeneca, Chem Innovat Ctr, Somerville, MA USA
- [9] Fragment-based discovery of focal adhesion kinase inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2013, 23 (19) : 5401 - 5409Graedler, Ulrich论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Res, Merck KGaA, D-64293 Darmstadt, Germany Merck Serono Res, Merck KGaA, D-64293 Darmstadt, GermanyBomke, Joerg论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Res, Merck KGaA, D-64293 Darmstadt, Germany Merck Serono Res, Merck KGaA, D-64293 Darmstadt, GermanyMusil, Djordje论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Res, Merck KGaA, D-64293 Darmstadt, Germany Merck Serono Res, Merck KGaA, D-64293 Darmstadt, GermanyDresing, Verena论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Res, Merck KGaA, D-64293 Darmstadt, Germany Merck Serono Res, Merck KGaA, D-64293 Darmstadt, GermanyLehmann, Martin论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Res, Merck KGaA, D-64293 Darmstadt, Germany Merck Serono Res, Merck KGaA, D-64293 Darmstadt, GermanyHoelzemann, Guenter论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Res, Merck KGaA, D-64293 Darmstadt, Germany Merck Serono Res, Merck KGaA, D-64293 Darmstadt, GermanyGreiner, Hartmut论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Res, Merck KGaA, D-64293 Darmstadt, Germany Merck Serono Res, Merck KGaA, D-64293 Darmstadt, GermanyEsdar, Christina论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Res, Merck KGaA, D-64293 Darmstadt, Germany Merck Serono Res, Merck KGaA, D-64293 Darmstadt, GermanyKrier, Mireille论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Res, Merck KGaA, D-64293 Darmstadt, Germany Merck Serono Res, Merck KGaA, D-64293 Darmstadt, GermanyHeinrich, Timo论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Res, Merck KGaA, D-64293 Darmstadt, Germany Merck Serono Res, Merck KGaA, D-64293 Darmstadt, Germany
- [10] Discovery of KATII inhibitors via a fragment-based approachABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2016, 251Han, Ying论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USAStachura, Sylwia论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, LVL, Princeton, NJ USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USAMcClure, Andrea论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USACavallaro, Cullen论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, LVL, Princeton, NJ USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USAAllard, Christopher论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USARajamani, Ramkumar论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, LVL, Princeton, NJ USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USAYong, Wei论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, LVL, Princeton, NJ USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USALewis, Hal论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, LVL, Princeton, NJ USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USAMuckelbauer, Jodi论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, LVL, Princeton, NJ USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USALoughney, Deborah论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, LVL, Princeton, NJ USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USAMetzler, William论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, LVL, Princeton, NJ USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USANirschl, David论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, LVL, Princeton, NJ USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USAWeller, Harold论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, LVL, Princeton, NJ USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USAGerritz, Sam论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USA