PREDICTION OF DRUG CLEARANCE IN GENENTECH: A RETROSPECTIVE ANALYSIS OF IN VITRO IN VIVO EXTRAPOLATION METHODS AND ALLOMETRY METHODS

被引:0
|
作者
Mao, Jialin [1 ]
Chen, Yuan [1 ]
Fan, Peter [1 ]
Kenny, Jane [1 ]
Liederer, Bianca M. [1 ]
Liu, Xingrong [1 ]
Wright, Matthew [1 ]
Hop, Cornelis E. C. A. [1 ]
机构
[1] Genentech Inc, Dept Drug Metab & Pharmacokinet, San Francisco, CA 94080 USA
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
P23
引用
收藏
页码:51 / 52
页数:2
相关论文
共 50 条
  • [1] CLEARANCE PREDICTION FOR METABOLICALLY ELIMINATED COMPOUNDS: IN VITRO TO IN VIVO EXTRAPOLATION (IVIVE) OR ALLOMETRY?
    Mei, Hong
    Deshmukh, Sujal
    Gibson, Christopher
    DRUG METABOLISM REVIEWS, 2015, 47 : 51 - 51
  • [2] Prediction of metabolic drug clearance in humans:: In vitro-in vivo extrapolation vs allometric scaling
    Shiran, M. R.
    Proctor, N. J.
    Howgate, E. M.
    Rowland-Yeo, K.
    Tucker, G. T.
    Rostami-Hodjegan, A.
    XENOBIOTICA, 2006, 36 (07) : 567 - 580
  • [3] In vitro analysis of human drug glucuronidation and prediction of in vivo metabolic clearance
    Soars, MG
    Burchell, B
    Riley, RJ
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2002, 301 (01): : 382 - 390
  • [4] Impact of Plasma Protein Binding in Drug Clearance Prediction: A DataBase Analysis of Published Studies and Implications for In Vitro-In Vivo Extrapolation
    Francis, L. J.
    Houston, J. B.
    Hallifax, D.
    DRUG METABOLISM AND DISPOSITION, 2021, 49 (03) : 188 - 201
  • [5] Comparative assessment of In Vitro-In Vivo extrapolation methods used for predicting hepatic metabolic clearance of drugs
    Poulin, Patrick
    Hop, Cornelis E. C. A.
    Ho, Quynh
    Halladay, Jason S.
    Haddad, Sami
    Kenny, Jane R.
    JOURNAL OF PHARMACEUTICAL SCIENCES, 2012, 101 (11) : 4308 - 4326
  • [6] In Vitro-In Vivo Extrapolation of Metabolism- and Transporter-Mediated Drug-Drug Interactions-Overview of Basic Prediction Methods
    Yoshida, Kenta
    Zhao, Ping
    Zhang, Lei
    Abernethy, Darrell R.
    Rekic, Dinko
    Reynolds, Kellie S.
    Galetin, Aleksandra
    Huang, Shiew-Mei
    JOURNAL OF PHARMACEUTICAL SCIENCES, 2017, 106 (09) : 2209 - 2213
  • [7] Validation of Methods for in Vitro-in Vivo Extrapolation Using Hepatic Clearance Measurements in Isolated Perfused Fish Livers
    Schultz, Matthew
    Krause, Sophia
    Brinkmann, Markus
    ENVIRONMENTAL SCIENCE & TECHNOLOGY, 2022, 56 (17) : 12416 - 12423
  • [8] In vitro-in vivo extrapolation of clearance: Modeling hepatic metabolic clearance of highly bound drugs and comparative assessment with existing calculation methods
    Poulin, Patrick
    Kenny, Jane R.
    Hop, Cornelis E. C. A.
    Haddad, Sami
    JOURNAL OF PHARMACEUTICAL SCIENCES, 2012, 101 (02) : 838 - 851
  • [9] Clearance Prediction of Targeted Covalent Inhibitors by In Vitro-In Vivo Extrapolation of Hepatic and Extrahepatic Clearance Mechanisms
    Leung, Louis
    Yang, Xin
    Strelevitz, Timothy J.
    Montgomery, Justin
    Brown, Matthew F.
    Zientek, Michael A.
    Banfield, Christopher
    Gilbert, Adam M.
    Thorarensen, Atli
    Dowty, Martin E.
    DRUG METABOLISM AND DISPOSITION, 2017, 45 (01) : 1 - 7
  • [10] Integration of mechanism-based in vitro methods and quantitative in vitro-in vivo extrapolation (QIVIVE) modelling for prediction of nephrotoxicity
    Mally, A.
    Birk, B.
    DiFiore, S.
    Ellinger, B.
    Jarzina, S.
    Taverne, F.
    Kramer, N.
    TOXICOLOGY LETTERS, 2018, 295 : S27 - S27