Synthesis and bioassay of a new class of heterocycles pyrrolyl oxadiazoles/thiadiazoles/triazoles

被引：24
|
作者：
Padmavathi, V. [1 ]
Mohan, A. V. Nagendra [1 ]
Thriveni, P. [1 ]
Shazia, A. [2 ]
机构：
[1] Sri Venkateswara Univ, Dept Chem, Tirupati 517502, Andhra Pradesh, India
[2] Indian Inst Sci, Dept Mol Reprod Dev & Genet, Bangalore 560012, Karnataka, India
来源：
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | 2009年 / 44卷 / 05期
关键词：
Pyrroles; 1,3,4-Thiadiazoles; 1,3,4-Oxadiazoles; Antimicrobial activity; Cytotoxic activity; BIOLOGICAL-ACTIVITIES; OXADIAZOLES; DESIGN; DERIVATIVES; ANTAGONISTS; RECEPTOR; GROWTH; ESTER;
D O I：
10.1016/j.ejmech.2008.04.003
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
A new class of heterocycles pyrrolyl thiadiazoles, pyrrolyl oxadiazoles and pyrrolyl triazoles were prepared from arylsulfonylethenesulfonylacetic acid methyl ester and tested for their antimicrobial and cytotoxic activities. (C) 2008 Elsevier Masson SAS. All rights reserved.
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页码：2313 / 2321
页数：9
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