Synthesis and characterization of phosphonic acid-substituted amino acids as excitatory amino acid receptor antagonists

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作者
Ornstein, PL
Arnold, MB
Allen, NK
Schoepp, DD
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O61 [无机化学];
学科分类号
070301 ; 081704 ;
摘要
Decahydroisoquinoline-3-carboxylic acids, substituted at C-6 with an acidic moiety such as a phosphonic, sulfonic or carboxylic acid or tetrazole, were prepared as antagonists of excitatory amino acid (EAA) receptors.
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页码:309 / 312
页数:4
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