Synthesis and herbicidal activities of pentylchrysanthemacyl thiourea pyrimidine derivatives and related fuse ring compounds

被引：0

作者：

Xue, SJ ^{[1
]}

Duan, LP ^{[1
]}

Ke, SY ^{[1
]}

Zhu, JM ^{[1
]}

机构：

[1] Shanghai Normal Univ, Coll Life & Environm Sci, Shanghai 200234, Peoples R China

来源：

CHINESE JOURNAL OF ORGANIC CHEMISTRY | 2004年 / 24卷 / 06期

关键词：

pentylchrysanthem acid; acylthiourea; substituted-2-amino-pyrimidine; 2H-1,2,4-thiadiazolo[2,3-alpha]-pyrimidine; synthesis; herbicidal activity;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Five N-[3-methyl-2-(4-chlorophenyl)butyryl]-N'-(2-pyrimidinyl)thioureas (3) have been synthesized. Compounds 4 were obtained by oxidizing cyclization. of compounds 3 in the presence of bromine in chloroform. The structures of 3 and 4 were confirmed by 111, H-1 NMR and elemental analysis. The preliminary biological tests indicate that compound 3a has excellent herbicidal activity.

引用

页码：686 / 690

页数：5

共 14 条

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