共 50 条
- [1] Discovery of the potent PI3K/mTOR dual inhibitor PF-04979064[J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2010, 240Cheng, Hengmiao论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA USABagrodia, Shubha论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA USABailey, Simon论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA USABaxi, Sangita M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA USAGoulet, Lance论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA USAGuo, Lisa论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA USAHoffman, Jacqui论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA USAJohnson, Ted O.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA USAJohnson, Ted W.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA USALi, Chunze论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA USALi, John论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA USALiu, Kevin论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA USALiu, Zhengyu论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA USAMarx, Matthew A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA USAPaderes, Gigi论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA USASun, Shaoxian论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA USAWalls, Marlena论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA USAWells, Peter A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA USAYang, Anle论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA USAYin, Min-Jean论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA USAZhu, Jingjiang论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA USA
- [2] Synthesis of PF-04691502, a highly potent PI3K/mTOR dual inhibitor[J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2012, 243Hoffman, Jacqui论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, Canc Chem, San Diego, CA 92121 USABailey, Simon论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, Canc Chem, San Diego, CA 92121 USACheng, Hengmiao论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, Canc Chem, San Diego, CA 92121 USAKania, Robert论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, Canc Chem, San Diego, CA 92121 USAJai, Lei论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, Canc Chem, San Diego, CA 92121 USANambu, Mitch论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, Canc Chem, San Diego, CA 92121 USANinkovich, Sacha论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, Canc Chem, San Diego, CA 92121 USAPairish, Mason论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, Canc Chem, San Diego, CA 92121 USASrirangam, Jay论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, Canc Chem, San Diego, CA 92121 USAWang, Xiaolong论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, Canc Chem, San Diego, CA 92121 USALe, Phuong论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, Canc Chem, San Diego, CA 92121 USA
- [3] Discovery of the highly potent PI3K/mTOR dual inhibitor PF-04691502 through structure based drug design[J]. MEDCHEMCOMM, 2010, 1 (02) : 139 - 144Cheng, Hengmiao论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USABagrodia, Shubha论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Oncol Res Unit, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USABailey, Simon论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USAEdwards, Martin论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USAHoffman, Jacqui论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USAHu, Qiyue论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USAKania, Robert论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USAKnighton, Daniel R.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USAMarx, Matthew A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USANinkovic, Sacha论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USASun, Shaoxian论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Oncol Res Unit, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USAZhang, Eric论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, PDM, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USA
- [4] Discovery, Optimization, and Evaluation of Potent and Highly Selective PI3Kγ-PI3Kδ Dual Inhibitors[J]. JOURNAL OF MEDICINAL CHEMISTRY, 2019, 62 (10) : 4936 - 4948Jia, Hong论文数: 0 引用数: 0 h-index: 0机构: Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaDai, Guangxiu论文数: 0 引用数: 0 h-index: 0机构: Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaSu, Weiguo论文数: 0 引用数: 0 h-index: 0机构: Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaXiao, Kun论文数: 0 引用数: 0 h-index: 0机构: Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaWeng, Jianyang论文数: 0 引用数: 0 h-index: 0机构: Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaZhang, Zhulin论文数: 0 引用数: 0 h-index: 0机构: Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaWang, Qing论文数: 0 引用数: 0 h-index: 0机构: Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaYuan, Tianhai论文数: 0 引用数: 0 h-index: 0机构: Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaShi, Fuying论文数: 0 引用数: 0 h-index: 0机构: Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaZhang, Zheng论文数: 0 引用数: 0 h-index: 0机构: Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaChen, Wei论文数: 0 引用数: 0 h-index: 0机构: Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaSai, Yang论文数: 0 引用数: 0 h-index: 0机构: Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaWang, Jian论文数: 0 引用数: 0 h-index: 0机构: Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaLi, Xiong论文数: 0 引用数: 0 h-index: 0机构: Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaCai, Yu论文数: 0 引用数: 0 h-index: 0机构: Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaYu, Jun论文数: 0 引用数: 0 h-index: 0机构: Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaRen, Ping论文数: 0 引用数: 0 h-index: 0机构: Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaVenable, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Janssen Pharmaceut Res & Dev, 3210 Merryfield Row, San Diego, CA 92121 USA Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaRao, Tadimeti论文数: 0 引用数: 0 h-index: 0机构: Janssen Pharmaceut Res & Dev, 3210 Merryfield Row, San Diego, CA 92121 USA Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaEdwards, James P.论文数: 0 引用数: 0 h-index: 0机构: Janssen Pharmaceut Res & Dev, 1400 McKean Rd, Spring House, PA 19477 USA Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaBembenek, Scott D.论文数: 0 引用数: 0 h-index: 0机构: Janssen Pharmaceut Res & Dev, 3210 Merryfield Row, San Diego, CA 92121 USA Hutchison MediPharma Ltd, Bldg 4,720 Cai Lun Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China
- [5] VS-5584, a Novel and Highly Selective PI3K/mTOR Kinase Inhibitor for the Treatment of Cancer[J]. MOLECULAR CANCER THERAPEUTICS, 2013, 12 (02) : 151 - 161Hart, Stefan论文数: 0 引用数: 0 h-index: 0机构: S BIO Pte Ltd, Singapore 117528, Singapore S BIO Pte Ltd, Singapore 117528, SingaporeNovotny-Diermayr, Veronica论文数: 0 引用数: 0 h-index: 0机构: S BIO Pte Ltd, Singapore 117528, Singapore S BIO Pte Ltd, Singapore 117528, SingaporeGoh, Kee Chuan论文数: 0 引用数: 0 h-index: 0机构: S BIO Pte Ltd, Singapore 117528, Singapore S BIO Pte Ltd, Singapore 117528, SingaporeWilliams, Meredith论文数: 0 引用数: 0 h-index: 0机构: S BIO Pte Ltd, Singapore 117528, Singapore S BIO Pte Ltd, Singapore 117528, SingaporeTan, Yong Cheng论文数: 0 引用数: 0 h-index: 0机构: S BIO Pte Ltd, Singapore 117528, Singapore S BIO Pte Ltd, Singapore 117528, SingaporeOng, Lai Chun论文数: 0 引用数: 0 h-index: 0机构: S BIO Pte Ltd, Singapore 117528, Singapore S BIO Pte Ltd, Singapore 117528, SingaporeCheong, Albert论文数: 0 引用数: 0 h-index: 0机构: S BIO Pte Ltd, Singapore 117528, Singapore S BIO Pte Ltd, Singapore 117528, SingaporeNg, Bee Kheng论文数: 0 引用数: 0 h-index: 0机构: S BIO Pte Ltd, Singapore 117528, Singapore S BIO Pte Ltd, Singapore 117528, SingaporeAmalini, Chithra论文数: 0 引用数: 0 h-index: 0机构: S BIO Pte Ltd, Singapore 117528, Singapore S BIO Pte Ltd, Singapore 117528, SingaporeMadan, Babita论文数: 0 引用数: 0 h-index: 0机构: S BIO Pte Ltd, Singapore 117528, Singapore S BIO Pte Ltd, Singapore 117528, SingaporeNagaraj, Harish论文数: 0 引用数: 0 h-index: 0机构: S BIO Pte Ltd, Singapore 117528, Singapore S BIO Pte Ltd, Singapore 117528, SingaporeJayaraman, Ramesh论文数: 0 引用数: 0 h-index: 0机构: S BIO Pte Ltd, Singapore 117528, Singapore S BIO Pte Ltd, Singapore 117528, SingaporePasha, Khalid M.论文数: 0 引用数: 0 h-index: 0机构: S BIO Pte Ltd, Singapore 117528, Singapore S BIO Pte Ltd, Singapore 117528, SingaporeEthirajulu, Kantharaj论文数: 0 引用数: 0 h-index: 0机构: S BIO Pte Ltd, Singapore 117528, Singapore S BIO Pte Ltd, Singapore 117528, SingaporeChng, Wee Joo论文数: 0 引用数: 0 h-index: 0机构: Natl Univ Singapore, Canc Sci Inst Singapore, Singapore 117548, Singapore Natl Univ Hlth Syst, Natl Univ Canc Inst Singapore, Dept Haematol Oncol, Singapore, Singapore S BIO Pte Ltd, Singapore 117528, SingaporeMustafa, Nurulhuda论文数: 0 引用数: 0 h-index: 0机构: Natl Univ Singapore, Canc Sci Inst Singapore, Singapore 117548, Singapore S BIO Pte Ltd, Singapore 117528, SingaporeGoh, Boon Cher论文数: 0 引用数: 0 h-index: 0机构: Natl Univ Singapore, Canc Sci Inst Singapore, Singapore 117548, Singapore S BIO Pte Ltd, Singapore 117528, SingaporeBenes, Cyril论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Massachusetts Gen Hosp, Ctr Canc, Charlestown, MA USA S BIO Pte Ltd, Singapore 117528, SingaporeMcDermott, Ultan论文数: 0 引用数: 0 h-index: 0机构: Wellcome Trust Sanger Inst, Canc Genome Project, Hinxton, England S BIO Pte Ltd, Singapore 117528, SingaporeGarnett, Mathew论文数: 0 引用数: 0 h-index: 0机构: Wellcome Trust Sanger Inst, Canc Genome Project, Hinxton, England S BIO Pte Ltd, Singapore 117528, SingaporeDymock, Brian论文数: 0 引用数: 0 h-index: 0机构: S BIO Pte Ltd, Singapore 117528, Singapore S BIO Pte Ltd, Singapore 117528, SingaporeWood, Jeanette M.论文数: 0 引用数: 0 h-index: 0机构: S BIO Pte Ltd, Singapore 117528, Singapore S BIO Pte Ltd, Singapore 117528, Singapore
- [6] Discovery of GSK2126458, a Highly Potent Inhibitor of PI3K and the Mammalian Target of Rapamycin[J]. ACS MEDICINAL CHEMISTRY LETTERS, 2010, 1 (01): : 39 - 43Knight, Steven D.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USAAdams, Nicholas D.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USABurgess, JoeIle L.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USAChaudhari, Amita M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USADarcy, Michael G.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USADonatelli, Carla A.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USALuengo, Juan I.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USANewlander, Ken A.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USAParrish, Cynthia A.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USARidgers, Lance H.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USASarpong, Martha A.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USASchmidt, Stanley J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USAVan Aller, Glenn S.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USACarson, Jeffrey D.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USADiamond, Melody A.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USAElkins, Patricia A.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USAGardiner, Christine M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USAGarver, Eric论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USAGilbert, Seth A.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USAGontarek, Richard R.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USAJackson, Jeffrey R.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USAKershner, Kevin L.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USALuo, Lusong论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USARaha, Kaushik论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USASherk, Christian S.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USASung, Chiu-Mei论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USASutton, David论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USATummino, Peter J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USAWegrzyn, Ronald J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USAAuger, Kurt R.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USADhanak, Dashyant论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Collegeville, PA 19426 USA GlaxoSmithKline Inc, Collegeville, PA 19426 USA
- [7] Discovery of a Potent, Selective, and Orally Available PI3Kδ Inhibitor for the Treatment of Inflammatory Diseases[J]. ACS MEDICINAL CHEMISTRY LETTERS, 2017, 8 (01): : 118 - 123Erra, Montse论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Med Chem & Screening, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainTaltavull, Joan论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Med Chem & Screening, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainGreco, Angelique论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Med Chem & Screening, Barcelona 08980, Spain Pharmaxis Ltd, 20 Rodborough Rd, Frenchs Forest, NSW 2086, Australia Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainJavier Bernal, Francisco论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Med Chem & Screening, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainFrancisco Caturla, Juan论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Med Chem & Screening, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainGracia, Jordi论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Med Chem & Screening, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainDominguez, Maria论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Pharmacokinet & Metab, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainSabate, Mar论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Pharmacokinet & Metab, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainParis, Stephane论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Med Chem & Screening, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainSoria, Salome论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Med Chem & Screening, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainHernandez, Begona论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Med Chem & Screening, Barcelona 08980, Spain Fundacio ACE, Marques Sentmenat,57, Barcelona 08029, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainArmengol, Clara论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainCabedo, Judit论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Syst Biol, Barcelona 08980, Spain Almirall R&D, Resp Therapeut Area, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainBravo, Monica论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Resp Therapeut Area, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainCalama, Elena论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Resp Therapeut Area, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainMiralpeix, Montserrat论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Resp Therapeut Area, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainLehner, Martin D.论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Resp Therapeut Area, Barcelona 08980, Spain Bionor SE, Kerschensteinerstr 11-15, D-92318 Neumarkt, Germany Almirall R&D, Med Chem & Screening, Barcelona 08980, Spain
- [8] Discovery of the Highly Potent PI3K/mTOR Dual Inhibitor PF-04979064 through Structure-Based Drug Design[J]. ACS MEDICINAL CHEMISTRY LETTERS, 2013, 4 (01): : 91 - 97Cheng, Hengmiao论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USALi, Chunze论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, PDM, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USABailey, Simon论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USABaxi, Sangita M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Oncol Res Unit, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USAGoulet, Lance论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, PDM, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USAGuo, Lisa论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USAHoffman, Jacqui论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USAJiang, Ying论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, PDM, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USAJohnson, Theodore Otto论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USAJohnson, Ted W.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USAKnighton, Daniel R.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USALi, John论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Oncol Res Unit, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USALiu, Kevin K. -C.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USALiu, Zhengyu论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USAMarx, Matthew A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USAWalls, Marlena论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Oncol Res Unit, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USAWells, Peter A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Oncol Res Unit, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USAYin, Min-Jean论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Oncol Res Unit, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USAZhu, Jinjiang论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USAZientek, Michael论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, La Jolla Labs, PDM, San Diego, CA 92121 USA Pfizer Worldwide Res & Dev, La Jolla Labs, Canc Chem, San Diego, CA 92121 USA
- [9] Antitumor Efficacy of PKI-587, a Highly Potent Dual PI3K/mTOR Kinase Inhibitor[J]. CLINICAL CANCER RESEARCH, 2011, 17 (10) : 3193 - 3203Mallon, Robert论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Oncol, Pearl River, NY 10965 USA Pfizer, Dept Oncol, Pearl River, NY 10965 USAFeldberg, Larry R.论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Oncol, Pearl River, NY 10965 USA Pfizer, Dept Oncol, Pearl River, NY 10965 USALucas, Judy论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Oncol, Pearl River, NY 10965 USA Pfizer, Dept Oncol, Pearl River, NY 10965 USAChaudhary, Inder论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Drug Safety & Metab, Pearl River, NY 10965 USA Pfizer, Dept Oncol, Pearl River, NY 10965 USADehnhardt, Christoph论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Discovery Med Chem, Pearl River, NY 10965 USA Pfizer, Dept Oncol, Pearl River, NY 10965 USADelos Santos, Efren论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Discovery Med Chem, Pearl River, NY 10965 USA Pfizer, Dept Oncol, Pearl River, NY 10965 USAChen, Zecheng论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Discovery Med Chem, Pearl River, NY 10965 USA Pfizer, Dept Oncol, Pearl River, NY 10965 USAdos Santos, Osvaldo论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Discovery Med Chem, Pearl River, NY 10965 USA Pfizer, Dept Oncol, Pearl River, NY 10965 USAAyral-Kaloustian, Semiramis论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Discovery Med Chem, Pearl River, NY 10965 USA Pfizer, Dept Oncol, Pearl River, NY 10965 USAVenkatesan, Aranapakam论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Discovery Med Chem, Pearl River, NY 10965 USA Pfizer, Dept Oncol, Pearl River, NY 10965 USAHollander, Irwin论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Oncol, Pearl River, NY 10965 USA Pfizer, Dept Oncol, Pearl River, NY 10965 USA
- [10] Discovery of novel and potent PARP/PI3K dual inhibitors for the treatment of cancer[J]. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 217Wu, Zhengyang论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Dept Med Chem, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaBai, Ying论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaJin, Jiaming论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Dept Med Chem, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaJiang, Teng论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Dept Med Chem, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaShen, Hui论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Dept Med Chem, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaJu, Qiurong论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Dept Med Chem, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaZhu, Qihua论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Dept Med Chem, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaXu, Yungen论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Dept Med Chem, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China