Dihydroethanoanthracene derivatives as in vitro malarial chloroquine resistance reversal agents

被引：27
|
作者：
Millet, J
Torrentino-Madamet, M
Alibert, S
Rogier, C
Santelli-Rouvier, C
Mosnier, J
Baret, E
Barbe, J
Parzy, D
Pradines, B
机构：
[1] IMTSSA, Unite Parasitol, F-13998 Marseille, France
[2] Fac Pharm Marseille, GERCTOP, UMR CNRS 6009, Marseille, France
[3] Inst Federat Rech 48, Marseille, France
来源：
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY | 2004年 / 48卷 / 07期
关键词：
D O I：
10.1128/AAC.48.7.2753-2756.2004
中图分类号：
Q93 [微生物学];
学科分类号：
071005 ; 100705 ;
摘要：
The ability of four 9,10-dihydroethanoanthracene derivatives (BG920, BG932, BG958, and BG996), as well as verapamil and promethazine, to reverse chloroquine resistance was assessed against 24 chloroquine-resistant and 10 chloroquine-susceptible strains of Plasmodium falciparum from different countries. The 9,10-dihydroethanoanthracene derivatives clearly increase chloroquine susceptibility only in chloroquine-resistant isolates.
引用
收藏
页码：2753 / 2756
页数：4
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