An efficient synthesis of novel spirodeoxoartemisinin with 2-pyrazoline ring

被引：4
|
作者：
Jung, M
Lee, S
机构：
[1] Department of Chemistry, Yonsei University, Seoul
来源：
HETEROCYCLES | 1997年 / 45卷 / 10期
关键词：
D O I：
10.3987/COM-97-7913
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Water-soluble, novel spirodeoxoartemisinin (10a) with 2-pyrazoline ring at C-11 was prepared from artemisinic acid (3) in four steps.
引用
收藏
页码：1907 / 1912
页数：6
相关论文
共 50 条
  • [1] Synthesis and Characterization of a Novel 2-Pyrazoline
    Singh, Pramod
    Negi, Jagmohan S.
    Pant, Geeta Joshi Nee
    Rawat, Mohan S. M.
    Budakoti, Asha
    MOLBANK, 2009, (03)
  • [2] Efficient asymmetric synthesis of a functionalized Δ2-pyrazoline
    Poupardin, O
    Greck, C
    Genet, JP
    TETRAHEDRON LETTERS, 2000, 41 (45) : 8795 - 8797
  • [3] Novel Analogues of 2-Pyrazoline: Synthesis, Characterization, and Antimycobacterial Evaluation
    Ozdemir, Ahmet
    Turan-Zitouni, Guelhan
    Kaplancikli, Zafer Asim
    TURKISH JOURNAL OF CHEMISTRY, 2008, 32 (05) : 529 - 538
  • [4] Design and synthesis of novel 2-pyrazoline analogues and their hMAO inhibitory activities
    Ucar, G.
    Evranos-Aksoz, B.
    Yabanoglu-Ciftci, S.
    Yelekci, K.
    FEBS JOURNAL, 2015, 282 : 299 - 299
  • [5] Design, Synthesis and hMAO Inhibitory Screening of Novel 2-Pyrazoline Analogues
    Evranos-Aksoz, Begum
    Ucar, Gulberk
    Yelekci, Kemal
    COMBINATORIAL CHEMISTRY & HIGH THROUGHPUT SCREENING, 2017, 20 (06) : 510 - 521
  • [6] Synthesis, antitubercular, anticonvulsant and antiinflammatory activities of some novel 2-pyrazoline derivatives
    Valarmathy, J.
    Joshua, L. Samuel
    Kumar, K. L. Senthil
    Kasabe, Amit J.
    ORIENTAL JOURNAL OF CHEMISTRY, 2010, 26 (03) : 1049 - 1054
  • [7] Synthesis and biological evaluation of some novel 2-mercaptobenzothiazoles carrying 2-pyrazoline
    Azam, Md Afzal
    Suresh, Bhojraj
    JOURNAL OF SCIENTIFIC & INDUSTRIAL RESEARCH, 2012, 71 (02): : 113 - 119
  • [8] Synthesis of some acylated 2-pyrazoline and chalcone derivatives
    Demet Coşkun
    Misir Ahmedzade
    Research on Chemical Intermediates, 2014, 40 : 1193 - 1199
  • [9] Novel 2-pyrazoline derivatives as potential anticonvulsant agents
    Shradha Bhandari
    Avinash C. Tripathi
    Shailendra K. Saraf
    Medicinal Chemistry Research, 2013, 22 : 5290 - 5296
  • [10] Synthesis of some acylated 2-pyrazoline and chalcone derivatives
    Coskun, Demet
    Ahmedzade, Misir
    RESEARCH ON CHEMICAL INTERMEDIATES, 2014, 40 (03) : 1193 - 1199
12345