Rigid aminoalcohol backbone as a highly defined chiral template for the preparation of optically active tertiary α-hydroxyl acids

被引：73
|
作者：
Senanayake, CH [1 ]
Fang, K [1 ]
Grover, P [1 ]
Bakale, RP [1 ]
Vandenbossche, CP [1 ]
Wald, SA [1 ]
机构：
[1] Sepracor Inc, Chem Res & Dev, Marlborough, MA 01752 USA
来源：
TETRAHEDRON LETTERS | 1999年 / 40卷 / 05期
关键词：
D O I：
10.1016/S0040-4039(98)02587-8
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Constrained aminoalcohol derived-ketoester or amides have provided a new entry for the production of enantiopure acid 1 for (S)-oxybutynin. (C) 1999 Published by Elsevier Science Ltd. All rights reserved.
引用
收藏
页码：819 / 822
页数：4
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