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- [1] Isoquinoline Derivatives as Potent, Selective, and Orally Active CRTH2 Antagonists[J]. CHEMICAL & PHARMACEUTICAL BULLETIN, 2014, 62 (06) : 528 - 537Nishikawa-Shimono, Rie论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Med Chem Labs, Kita Ku, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Med Chem Labs, Kita Ku, Saitama 3319530, JapanSekiguchi, Yoshinori论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Med Chem Labs, Kita Ku, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Med Chem Labs, Kita Ku, Saitama 3319530, JapanKawamura, Madoka论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Med Chem Labs, Kita Ku, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Med Chem Labs, Kita Ku, Saitama 3319530, JapanWakasugi, Daisuke论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Med Chem Labs, Kita Ku, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Med Chem Labs, Kita Ku, Saitama 3319530, JapanKawanishi, Masahumi论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Mol Funct & Pharmacol Labs, Kita Ku, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Med Chem Labs, Kita Ku, Saitama 3319530, JapanWatanabe, Kazuhito论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Mol Funct & Pharmacol Labs, Kita Ku, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Med Chem Labs, Kita Ku, Saitama 3319530, JapanAsakura, Yumiko论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Mol Funct & Pharmacol Labs, Kita Ku, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Med Chem Labs, Kita Ku, Saitama 3319530, JapanTakaoka, Akiko论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Mol Funct & Pharmacol Labs, Kita Ku, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Med Chem Labs, Kita Ku, Saitama 3319530, JapanTakayama, Tetsuo论文数: 0 引用数: 0 h-index: 0机构: Taisho Pharmaceut Co Ltd, Med Chem Labs, Kita Ku, Saitama 3319530, Japan Taisho Pharmaceut Co Ltd, Med Chem Labs, Kita Ku, Saitama 3319530, Japan
- [2] Discovery of novel, potent and orally bioavailable CRTH2 antagonists[J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2011, 241Terasaka, Tadashi论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanIto, Shinji论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanZenkoh, Tatsuya论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanHayashida, Hisashi论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanMatsuda, Hiroshi论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanMiyata, Junji论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanNagata, Hiroshi论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanTakasuna, Yuji论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanKobayashi, Miki论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanTakeuchi, Makoto论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanOhta, Mitsuaki论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, Japan
- [3] Novel selective orally active CRTH2 antagonists for allergic inflammation developed from in silico derived hits[J]. JOURNAL OF MEDICINAL CHEMISTRY, 2006, 49 (23) : 6638 - 6641Ulven, Trond论文数: 0 引用数: 0 h-index: 0机构: 7TM Pharma, DK-2970 Horsholm, Denmark 7TM Pharma, DK-2970 Horsholm, DenmarkReceveur, Jean-Marie论文数: 0 引用数: 0 h-index: 0机构: 7TM Pharma, DK-2970 Horsholm, Denmark 7TM Pharma, DK-2970 Horsholm, DenmarkGrimstrup, Marie论文数: 0 引用数: 0 h-index: 0机构: 7TM Pharma, DK-2970 Horsholm, Denmark 7TM Pharma, DK-2970 Horsholm, DenmarkRist, Oystein论文数: 0 引用数: 0 h-index: 0机构: 7TM Pharma, DK-2970 Horsholm, Denmark 7TM Pharma, DK-2970 Horsholm, DenmarkFrimurer, Thomas M.论文数: 0 引用数: 0 h-index: 0机构: 7TM Pharma, DK-2970 Horsholm, Denmark 7TM Pharma, DK-2970 Horsholm, DenmarkGerlach, Lars-Ole论文数: 0 引用数: 0 h-index: 0机构: 7TM Pharma, DK-2970 Horsholm, Denmark 7TM Pharma, DK-2970 Horsholm, DenmarkMathiesen, Jesper Mosolff论文数: 0 引用数: 0 h-index: 0机构: 7TM Pharma, DK-2970 Horsholm, Denmark 7TM Pharma, DK-2970 Horsholm, DenmarkKostenis, Evi论文数: 0 引用数: 0 h-index: 0机构: 7TM Pharma, DK-2970 Horsholm, Denmark 7TM Pharma, DK-2970 Horsholm, DenmarkUller, Lena论文数: 0 引用数: 0 h-index: 0机构: 7TM Pharma, DK-2970 Horsholm, Denmark 7TM Pharma, DK-2970 Horsholm, DenmarkHogberg, Thomas论文数: 0 引用数: 0 h-index: 0机构: 7TM Pharma, DK-2970 Horsholm, Denmark 7TM Pharma, DK-2970 Horsholm, Denmark
- [4] Discovery of a new class of potent, selective, and orally bioavailable CRTH2 (DP2) receptor antagonists for the treatment of allergic inflammatory diseases[J]. JOURNAL OF MEDICINAL CHEMISTRY, 2008, 51 (07) : 2227 - 2243Crosignani, Stefano论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Int SA, CH-1202 Geneva, Switzerland Merck Serono Int SA, CH-1202 Geneva, SwitzerlandPage, Patrick论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Int SA, CH-1202 Geneva, Switzerland Merck Serono Int SA, CH-1202 Geneva, SwitzerlandMissotten, Marc论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Int SA, CH-1202 Geneva, Switzerland Merck Serono Int SA, CH-1202 Geneva, SwitzerlandColovray, Veronique论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Int SA, CH-1202 Geneva, Switzerland Merck Serono Int SA, CH-1202 Geneva, SwitzerlandCleva, Christophe论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Int SA, CH-1202 Geneva, Switzerland Merck Serono Int SA, CH-1202 Geneva, SwitzerlandArrighi, Jean-Francois论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Int SA, CH-1202 Geneva, Switzerland Merck Serono Int SA, CH-1202 Geneva, SwitzerlandAtherall, John论文数: 0 引用数: 0 h-index: 0机构: BioFocus DPI, Saffron Walden CB10 1XL, Essex, England Merck Serono Int SA, CH-1202 Geneva, SwitzerlandMacritchie, Jackie论文数: 0 引用数: 0 h-index: 0机构: BioFocus DPI, Saffron Walden CB10 1XL, Essex, England Merck Serono Int SA, CH-1202 Geneva, SwitzerlandMartin, Thierry论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Int SA, CH-1202 Geneva, Switzerland Merck Serono Int SA, CH-1202 Geneva, SwitzerlandHumbert, Yves论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Int SA, CH-1202 Geneva, Switzerland Merck Serono Int SA, CH-1202 Geneva, SwitzerlandGaudet, Marilene论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Int SA, CH-1202 Geneva, Switzerland Merck Serono Int SA, CH-1202 Geneva, SwitzerlandPupowicz, Doris论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Int SA, CH-1202 Geneva, Switzerland Merck Serono Int SA, CH-1202 Geneva, SwitzerlandMaio, Maurizio论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Int SA, CH-1202 Geneva, Switzerland Merck Serono Int SA, CH-1202 Geneva, SwitzerlandPittet, Pierre-Andre论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Int SA, CH-1202 Geneva, Switzerland Merck Serono Int SA, CH-1202 Geneva, SwitzerlandGolzio, Lucia论文数: 0 引用数: 0 h-index: 0机构: Merck Serono, Ist Ric Biomed A Marxer, I-10010 Colleretto Giacosa, Italy Merck Serono Int SA, CH-1202 Geneva, SwitzerlandGiachetti, Claudio论文数: 0 引用数: 0 h-index: 0机构: Merck Serono, Ist Ric Biomed A Marxer, I-10010 Colleretto Giacosa, Italy Merck Serono Int SA, CH-1202 Geneva, SwitzerlandRocha, Cynthia论文数: 0 引用数: 0 h-index: 0机构: Merck Serono, Ist Ric Biomed A Marxer, I-10010 Colleretto Giacosa, Italy Merck Serono Int SA, CH-1202 Geneva, SwitzerlandBernardinelli, Gerald论文数: 0 引用数: 0 h-index: 0机构: Univ Geneva, Lab Xray Crystallog, CH-1211 Geneva, Switzerland Merck Serono Int SA, CH-1202 Geneva, SwitzerlandFilinchuk, Yaroslav论文数: 0 引用数: 0 h-index: 0机构: ESRF, Swiss Norwegian Beam Line, F-38043 Grenoble, France Merck Serono Int SA, CH-1202 Geneva, SwitzerlandScheer, Alexander论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Int SA, CH-1202 Geneva, Switzerland Merck Serono Int SA, CH-1202 Geneva, SwitzerlandSchwarz, Matthias K.论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Int SA, CH-1202 Geneva, Switzerland Merck Serono Int SA, CH-1202 Geneva, SwitzerlandChollet, Andre论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Int SA, CH-1202 Geneva, Switzerland Merck Serono Int SA, CH-1202 Geneva, Switzerland
- [5] Discovery of Potent, Selective, and Orally Bioavailable Alkynylphenoxyacetic Acid CRTH2 (DP2) Receptor Antagonists for the Treatment of Allergic Inflammatory Diseases[J]. JOURNAL OF MEDICINAL CHEMISTRY, 2011, 54 (20) : 7299 - 7317Crosignani, Stefano论文数: 0 引用数: 0 h-index: 0机构: Merck Serono SA, CH-1202 Geneva, Switzerland Merck Serono SA, CH-1202 Geneva, SwitzerlandPretre, Adeline论文数: 0 引用数: 0 h-index: 0机构: Merck Serono SA, CH-1202 Geneva, Switzerland Merck Serono SA, CH-1202 Geneva, SwitzerlandJorand-Lebrun, Catherine论文数: 0 引用数: 0 h-index: 0机构: Merck Serono SA, CH-1202 Geneva, Switzerland Merck Serono SA, CH-1202 Geneva, SwitzerlandFraboulet, Gaele论文数: 0 引用数: 0 h-index: 0机构: Merck Serono SA, CH-1202 Geneva, Switzerland Merck Serono SA, CH-1202 Geneva, SwitzerlandSeenisamy, Jeyaprakashnarayanan论文数: 0 引用数: 0 h-index: 0机构: Syngene Int Ltd, Bangalore 560099, Karnataka, India Merck Serono SA, CH-1202 Geneva, SwitzerlandAugustine, John Kallikat论文数: 0 引用数: 0 h-index: 0机构: Syngene Int Ltd, Bangalore 560099, Karnataka, India Merck Serono SA, CH-1202 Geneva, SwitzerlandMissotten, Marc论文数: 0 引用数: 0 h-index: 0机构: Merck Serono SA, CH-1202 Geneva, Switzerland Merck Serono SA, CH-1202 Geneva, SwitzerlandHumbert, Yves论文数: 0 引用数: 0 h-index: 0机构: Merck Serono SA, CH-1202 Geneva, Switzerland Merck Serono SA, CH-1202 Geneva, SwitzerlandCleva, Christophe论文数: 0 引用数: 0 h-index: 0机构: Merck Serono SA, CH-1202 Geneva, Switzerland Merck Serono SA, CH-1202 Geneva, SwitzerlandAbla, Nada论文数: 0 引用数: 0 h-index: 0机构: Merck Serono SA, CH-1202 Geneva, Switzerland Merck Serono SA, CH-1202 Geneva, SwitzerlandDaff, Hamina论文数: 0 引用数: 0 h-index: 0机构: Merck Serono SA, CH-1202 Geneva, Switzerland Merck Serono SA, CH-1202 Geneva, SwitzerlandSchott, Olivier论文数: 0 引用数: 0 h-index: 0机构: Merck Serono SA, CH-1202 Geneva, Switzerland Merck Serono SA, CH-1202 Geneva, SwitzerlandSchneider, Manfred论文数: 0 引用数: 0 h-index: 0机构: Merck Serono SA, CH-1202 Geneva, Switzerland Merck Serono SA, CH-1202 Geneva, SwitzerlandBurgat-Charvillon, Fabienne论文数: 0 引用数: 0 h-index: 0机构: Merck Serono SA, CH-1202 Geneva, Switzerland Merck Serono SA, CH-1202 Geneva, SwitzerlandRivron, Delphine论文数: 0 引用数: 0 h-index: 0机构: Merck Serono SA, CH-1202 Geneva, Switzerland Merck Serono SA, CH-1202 Geneva, SwitzerlandHamernig, Ingrid论文数: 0 引用数: 0 h-index: 0机构: Merck Serono SA, CH-1202 Geneva, Switzerland Merck Serono SA, CH-1202 Geneva, SwitzerlandArrighi, Jean-Francois论文数: 0 引用数: 0 h-index: 0机构: Merck Serono SA, CH-1202 Geneva, Switzerland Merck Serono SA, CH-1202 Geneva, SwitzerlandGaudet, Marilene论文数: 0 引用数: 0 h-index: 0机构: Merck Serono SA, CH-1202 Geneva, Switzerland Merck Serono SA, CH-1202 Geneva, SwitzerlandZimmerli, Simone C.论文数: 0 引用数: 0 h-index: 0机构: Merck Serono SA, CH-1202 Geneva, Switzerland Merck Serono SA, CH-1202 Geneva, SwitzerlandJuillard, Pierre论文数: 0 引用数: 0 h-index: 0机构: Merck Serono SA, CH-1202 Geneva, Switzerland Merck Serono SA, CH-1202 Geneva, SwitzerlandJohnson, Zoe论文数: 0 引用数: 0 h-index: 0机构: Merck Serono SA, CH-1202 Geneva, Switzerland Merck Serono SA, CH-1202 Geneva, Switzerland
- [6] Azaindoles as potent CRTH2 receptor antagonists[J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 21 (02) : 841 - 845Simard, Daniel论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, CanadaLeblanc, Yves论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, CanadaBerthelette, Carl论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, CanadaZaghdane, M. Helmi论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, CanadaMolinaro, Carmela论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, CanadaWang, Zhaoyin论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, CanadaGallant, Michel论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, CanadaLau, Stephen论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, CanadaThao, Trinh论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, CanadaHamel, Martine论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, CanadaStocco, Rino论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, CanadaSawyer, Nicole论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, CanadaSillaots, Susan论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, CanadaGervais, Francois论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, CanadaHoule, Robert论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, CanadaLevesque, Jean-Francois论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada
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