Application of palladium-catalyzed amination to the synthesis of polyazamacrocycles containing 3,5-disubstituted pyridine

被引:13
|
作者
Beletskaya, IP [1 ]
Averin, AD
Ulanovskaya, OA
Fedotenko, IA
机构
[1] Moscow MV Lomonosov State Univ, Dept Chem, Moscow 119992, Russia
[2] VN Orekhovich Inst Biomed Chem, Moscow 119992, Russia
[3] Fac Sci Gabriel, LIMSAG, UMR 5633, F-21100 Dijon, France
关键词
D O I
10.1246/cl.2005.1100
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
The synthesis of a new family of nitrogen- and oxygen-containing macrocycles, which employs palladium-catalyzed amination of 3,5-dihalopyridines, is described. Synthetic approaches to cyclodimers have been elaborated via bis(pyridyl)substituted polyamines and bis(polyamino) substituted pyridines.
引用
收藏
页码:1100 / 1101
页数:2
相关论文
共 50 条
  • [1] Palladium-catalyzed amination in the synthesis of polyazamacrocycles
    I. P. Beletskaya
    A. D. Averin
    A. G. Bessmertnykh
    F. Denat
    R. Guilard
    Russian Journal of Organic Chemistry, 2010, 46 : 947 - 967
  • [2] Palladium-catalyzed amination in the synthesis of polyazamacrocycles
    Beletskaya, I. P.
    Averin, A. D.
    Bessmertnykh, A. G.
    Denat, F.
    Guilard, R.
    RUSSIAN JOURNAL OF ORGANIC CHEMISTRY, 2010, 46 (07) : 947 - 967
  • [3] Synthesis of 3,5-disubstituted piperazinones via palladium(II)-catalyzed amination
    Ferber, Benoit
    Prestat, Guillaume
    Vogel, Sophie
    Madec, David
    Poli, Giovanni
    SYNLETT, 2006, (13) : 2133 - 2135
  • [4] Palladium-catalyzed amination of 3,5-dihalopyridines - a convenient route to new polyazamacrocycles
    Averin, AD
    Ulanovskaya, OA
    Fedotenko, IA
    Borisenko, AA
    Serebryakova, MV
    Beletskaya, IP
    HELVETICA CHIMICA ACTA, 2005, 88 (07) : 1983 - 2002
  • [5] Palladium-catalyzed Amination in the synthesis of polyazamacrocycles containing a 1,3-disubstiituted benzene moiety
    Averin, Alexei D.
    Shukhaev, Anton V.
    Golub, Svetlana L.
    Buryak, Alexei K.
    Beletskaya, Irina P.
    SYNTHESIS-STUTTGART, 2007, (19): : 2995 - 3012
  • [6] Palladium-catalyzed amination in the synthesis of macrocyclic compounds containing 1,3-disubstituted adamantane fragments
    E. R. Ranyuk
    A. D. Averin
    A. K. Buryak
    E. N. Savel’ev
    B. S. Orlinson
    I. A. Novakov
    I. P. Beletskaya
    Russian Journal of Organic Chemistry, 2009, 45 : 1555 - 1566
  • [7] Palladium-catalyzed amination in the synthesis of macrocyclic compounds containing 1,3-disubstituted adamantane fragments
    Ranyuk, E. R.
    Averin, A. D.
    Buryak, A. K.
    Savel'ev, E. N.
    Orlinson, B. S.
    Novakov, I. A.
    Beletskaya, I. P.
    RUSSIAN JOURNAL OF ORGANIC CHEMISTRY, 2009, 45 (10) : 1555 - 1566
  • [8] A new access to 3,5-disubstituted piperazinones via Pd(0)-catalyzed amination
    Ferber, B
    Lemaire, S
    Mader, MM
    Prestat, G
    Poli, G
    TETRAHEDRON LETTERS, 2003, 44 (22) : 4213 - 4216
  • [9] PALLADIUM-CATALYZED AMINATION IN THE SYNTHESIS OF MACROBICYCLES INCORPORATING CYCLEN, CYCLAM AND PYRIDINE MOIETIES
    Averin, Alexei D.
    Tyutenov, Kanat S.
    Shukhaev, Anton V.
    Kobelev, Sergei M.
    Buryak, Alexei K.
    Denat, Franck
    Guilard, Roger
    Beletskaya, Irina P.
    HETEROCYCLES, 2012, 86 (02) : 1341 - 1366
  • [10] Palladium-catalyzed amination in the synthesis of macrocycles comprising cholane, polyamine and pyridine units
    Averin, Alexei D.
    Ranyuk, Elena R.
    Lukashev, Nikolai V.
    Golub, Svetlana L.
    Buryak, Alexel K.
    Beletskaya, Irina P.
    TETRAHEDRON LETTERS, 2008, 49 (07) : 1188 - 1191