A comparison of the in vitro effects of (±)-4-methylthioamphetamine and (±)-MDMA on 5-HT re-uptake in the brain and on vascular responses to 5-HT

被引:0
|
作者
Murphy, JEJ
Cannon, DM
Guiry, P
McCormack, P
Baird, AW
McBean, GJ
Keenan, AK
机构
[1] Univ Coll Dublin, Dept Pharmacol, Conway Inst Biomol & Biomed Res, Dublin 4, Ireland
[2] Univ Coll Dublin, Dept Biochem, Conway Inst Biomol & Biomed Res, Dublin 4, Ireland
[3] Univ Coll Dublin, Dept Chem, Dublin 4, Ireland
[4] Univ Coll Dublin, Dept Chem, Conway Inst Biomol & Biomed Res, Dublin 4, Ireland
[5] Univ Coll Dublin, Conway Inst Biomol & Biomed Res, Dept Vet Physiol & Biochem, Dublin 4, Ireland
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
35P
引用
收藏
页数:1
相关论文
共 50 条
  • [1] Effects of MDMA and related analogs on plasma 5-HT: Relevance to 5-HT transporters in blood and brain
    Yubero-Lahoz, Samanta
    Ayestas, Mario A., Jr.
    Blough, Bruce E.
    Partilla, John S.
    Rothman, Richard B.
    de la Torre, Rafael
    Baumann, Michael H.
    EUROPEAN JOURNAL OF PHARMACOLOGY, 2012, 674 (2-3) : 337 - 344
  • [2] In vitro neuronal and vascular responses to 5-HT in rats chronically exposed to MDMA
    Cannon, DM
    Keenan, AK
    Guiry, PJ
    Buon, C
    Baird, AW
    McBean, GJ
    BRITISH JOURNAL OF PHARMACOLOGY, 2001, 134 (07) : 1455 - 1460
  • [3] Ligands with dual affinity for 5-HT 1A and 5-HT re-uptake receptors for the treatment of depression.
    van Niel, MB
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2000, 220 : U571 - U571
  • [4] STEREOSELECTIVITY OF 5-HT UPTAKE AND TOPOGRAPHY OF 5-HT UPTAKE SITE
    SMITH, DF
    INTERNATIONAL JOURNAL OF NEUROSCIENCE, 1987, 32 (1-2) : 403 - 403
  • [5] Effect of repeated exposure to MDMA on the function of the 5-HT transporter as assessed by synaptosomal 5-HT uptake
    Huff, Courtney
    Bhide, Nirmal
    Schroering, Allen
    Yamamoto, Bryan K.
    Gudelsky, Gary A.
    BRAIN RESEARCH BULLETIN, 2013, 91 : 52 - 57
  • [6] EFFECTS OF TRANYLCYPROMINE ON 5-HT UPTAKE AND ITS INTERACTION WITH PCPA ON RAT-BRAIN 5-HT
    FRIEDMAN, E
    SHOPSIN, B
    GERSHON, S
    RESEARCH COMMUNICATIONS IN CHEMICAL PATHOLOGY AND PHARMACOLOGY, 1976, 15 (01): : 191 - 194
  • [7] WHICH 5-HT RECEPTORS ARE INVOLVED IN THE MODULATION OF 5-HT SYNTHESIS BY THE 5-HT UPTAKE BLOCKER, CITALOPRAM
    MORET, C
    BRILEY, M
    BRITISH JOURNAL OF PHARMACOLOGY, 1993, 108 : P96 - P96
  • [8] Genetics of the serotonin (5-HT) uptake mechanism (5-HT transporter)
    Lesch, KP
    BIOLOGICAL PSYCHIATRY, 1997, 41 : 11 - 11
  • [9] Effects of serotonin re-uptake inhibition on 5-HT in the hippocampus of 5-HT1B receptor knockout mice
    de Groote, L
    Olivier, B
    Westenberg, HGM
    MONITORING MOLECULES IN NEUROSCIENCE, 2001, : 337 - 338
  • [10] Discrepancies between the in vitro and in vivo 5-HT and norepinephrine re-uptake blocking properties of venlafaxine
    Béïque, JC
    Debonnel, G
    De Montigny, C
    Blier, P
    ADVANCES IN SEROTONIN RECEPTOR RESEARCH: MOLECULAR BIOLOGY, SIGNAL TRANSDUCTION, AND THERAPEUTICS, 1998, 861 : 290 - 291