Novel Selective Phosphodiesterase Type 1 Inhibitors; a Comprehensive in vitro, ex vivo and in vivo Assessment of Cardiovascular Effects

被引:0
|
作者
Laursen, M. [1 ]
Beck, L. [2 ]
Bangshaab, M. [2 ]
Christoffersen, C. T. [1 ]
Bundgaard, C. [1 ]
Mogensen, S. [2 ]
Hedegaard, E. R. [2 ]
Mow, T. [1 ]
Grunnet, M. [2 ,3 ]
Simonsen, U. [2 ]
机构
[1] Lundbeck AS, Copenhagen, Denmark
[2] Aarhus Univ, Dept Biomed Pulm & Cardiovasc Pharmacol, DK-8000 Aarhus C, Denmark
[3] Univ Copenhagen, Dept Drug Design & Pharmacol, DK-1168 Copenhagen, Denmark
关键词
D O I
暂无
中图分类号
Q4 [生理学];
学科分类号
071003 ;
摘要
引用
收藏
页码:31 / 31
页数:1
相关论文
共 50 条
  • [1] Cardiovascular effects of a novel, potent and selective phosphodiesterase 5 inhibitor, DMPPO: In vitro and in vivo characterization
    Delpy, E
    deGouville, ACL
    [J]. BRITISH JOURNAL OF PHARMACOLOGY, 1996, 118 (06) : 1377 - 1384
  • [2] The effects of bisphenols on the cardiovascular system ex vivo and in vitro
    Carazo, A.
    Tvrdy, V.
    Dias, P.
    Pourova, J.
    Jirkovsky, E.
    Moravcova, M.
    Masic, L. Peterlin
    Dolenc, M. Sollner
    Mladenka, P.
    [J]. TOXICOLOGY LETTERS, 2023, 384 : S129 - S129
  • [3] In vitro to in vivo translation of effects of phosphodiesterase inhibitors on cardiac contractility
    Liu, Xiaoqin
    Shaughnessy, Thomas
    Polakowski, Jim
    Foley, C. Michael M.
    [J]. JOURNAL OF PHARMACOLOGICAL AND TOXICOLOGICAL METHODS, 2018, 93 : 124 - 124
  • [4] Phosphodiesterase type 4 inhibitors cause proinflammatory effects in vivo
    McCluskie, Kerryn
    Klein, Uwe
    Linnevers, Chris
    Ji, Yu-hua
    Yang, Alfred
    Husfeld, Craig
    Thomas, G. Roger
    [J]. JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2006, 319 (01): : 468 - 476
  • [5] The effects of bisphenols on the cardiovascular system ex vivo and in vivo
    Tvrdy, Vaclav
    Dias, Patricia
    Nejmanova, Iveta
    Carazo, Alejandro
    Jirkovsky, Eduard
    Pourova, Jana
    Fadraersada, Jaka
    Moravcova, Monika
    Masic, Lucija Peterlin
    Dolenc, Marija Sollner
    Mladenka, Premysl
    [J]. CHEMOSPHERE, 2023, 313
  • [6] Antitumor effects of selective PRMT1 inhibitors on neuroblastoma in vitro and in vivo
    Hansen, Jeanne N.
    Lotta, Louis T.
    Eberhardt, Allison
    Zheng, Yujun George
    Ji, Sen
    Yang, Shengyong
    Schor, Nina F.
    Li, Xingguo
    [J]. CANCER RESEARCH, 2018, 78 (19)
  • [7] THE CYTOTOXICITY OF SILVERWOUND DRESSINGS: ASSESSMENT IN VITRO, EX VIVO, AND IN VIVO
    Iljas, Juvita D.
    McGovern, Jacqui
    Boonkaew, Benjawan
    Kempf, Margit
    Kimble, Roy M.
    Parker, Tony J.
    Cuttle, Leila
    [J]. WOUND REPAIR AND REGENERATION, 2016, 24 (06) : A22 - A22
  • [8] Diabetic retinopathy: a comprehensive update on in vivo, in vitro and ex vivo experimental models
    Sadikan, Muhammad Zulfiqah
    Nasir, Nurul Alimah Abdul
    Lambuk, Lidawani
    Mohamud, Rohimah
    Reshidan, Nur Hidayah
    Low, Evon
    Singar, Saiful Anuar
    Sabere, Awis Sukarni Mohmad
    Iezhitsa, Igor
    Agarwal, Renu
    [J]. BMC OPHTHALMOLOGY, 2023, 23 (01)
  • [9] Diabetic retinopathy: a comprehensive update on in vivo, in vitro and ex vivo experimental models
    Muhammad Zulfiqah Sadikan
    Nurul Alimah Abdul Nasir
    Lidawani Lambuk
    Rohimah Mohamud
    Nur Hidayah Reshidan
    Evon Low
    Saiful Anuar Singar
    Awis Sukarni Mohmad Sabere
    Igor Iezhitsa
    Renu Agarwal
    [J]. BMC Ophthalmology, 23
  • [10] The In Vitro and Ex Vivo Efficacy of Novel Arginase Inhibitors for the Treatment of Allergic Asthma
    van den Berg, M. P.
    Kurhade, S. H.
    Lunev, S.
    van Faassen, H. J.
    Bos, I. S.
    Zuidhof, A. B.
    Groves, M.
    Kema, I. P.
    Domling, A.
    Meurs, H.
    Gosens, R.
    [J]. AMERICAN JOURNAL OF RESPIRATORY AND CRITICAL CARE MEDICINE, 2018, 197