Evaluation of some quinoline-based hydrazone derivatives as insecticidal agents

被引：8

作者：

Yu, Xiang ^{[1
]}

Feng, Gang ^{[2
]}

Huang, Jiulin ^{[1
]}

Xu, Hui ^{[1
]}

机构：

[1] Northwest A&F Univ, Coll Sci, Res Inst Pesticidal Design & Synth, Yangling 712100, Shaanxi Provinc, Peoples R China

[2] Chinese Acad Trop Agr Sci, Environm & Plant Protect Inst, Haikou 571101, Hainan Province, Peoples R China

来源：

RSC ADVANCES | 2016年 / 6卷 / 36期

基金：

中国国家自然科学基金;

关键词：

ACTIVITY-RELATIONSHIP QSAR; SPODOPTERA-LITURA; ANTIPLASMODIAL ACTIVITY; LEPIDOPTERA-NOCTUIDAE;

D O I：

10.1039/c6ra00993j

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

In continuation of our program aimed at the discovery and development of efficient insecticidal agents, a series of quinoline-based hydrazone derivatives were synthesized and evaluated as insecticidal agents against three-day-old larvae of Spodoptera litura (Noctuidae: Lepidoptera), a polyphagous insect pest of many important crops, in vivo at 1 mg mL(-1). In particular, compounds 3c, 3e, 4g, 4h, and 6f showed potent insecticidal activity with 7 day mortality rates greater than 93%, and were comparable to that of the positive control toosendanin.

引用

页码：30405 / 30411

页数：7

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