Brain localization and neurochemical effects of the histamine H3 receptor antagonist ABT-239

被引：0
|
作者：
Miller, TR [1 ]
Milicic, I [1 ]
Wang, JS [1 ]
Otte, S [1 ]
Nikkel, AL [1 ]
Bitner, RS [1 ]
Drescher, KU [1 ]
Fox, GB [1 ]
Cowart, MD [1 ]
Hancock, AA [1 ]
Esbenshade, TA [1 ]
机构：
[1] Abbott Labs, Neurosci res, GPRD, Abbott Pk, IL 60064 USA
来源：
JOURNAL OF NEUROCHEMISTRY | 2005年 / 94卷
关键词：
D O I：
暂无
中图分类号：
Q5 [生物化学]; Q7 [分子生物学];
学科分类号：
071010 ; 081704 ;
摘要：
引用
收藏
页码：82 / 82
页数：1
相关论文
共 50 条
  • [1] Effects of the histamine H3 receptor antagonist ABT-239 on cognition and nicotine-induced memory enhancement in mice
    Kruk, Marta
    Miszkiel, Joanna
    McCreary, Andrew C.
    Przegalinski, Edmund
    Filip, Malgorzata
    Biala, Grazyna
    PHARMACOLOGICAL REPORTS, 2012, 64 (06) : 1316 - 1325
  • [2] Effects of the histamine H3 receptor antagonist ABT-239 on cognition and nicotine-induced memory enhancement in mice
    Marta Kruk
    Joanna Miszkiel
    Andrew C. McCreary
    Edmund Przegaliński
    Małgorzata Filip
    Grażyna Biała
    Pharmacological Reports, 2012, 64 : 1316 - 1325
  • [3] ABT-239, A novel, selective, and potent human histamine H3 receptor antagonist with cognition enhancing properties
    Esbenshade, T
    Krueger, KM
    Miller, TR
    Branowski, J
    Kang, CH
    Yao, BB
    Witte, DG
    Pan, JB
    Carr, TL
    Fox, GB
    Faghih, R
    Black, LA
    Bennani, YL
    Sullivan, JP
    Cowart, MD
    Hancock, AA
    FASEB JOURNAL, 2004, 18 (04): : A579 - A579
  • [4] ABT-239, a potent human histamine H3 receptor antagonist with favorable drug-like properties
    Esbenshade, TA
    Wetter, JM
    Marsh, K
    Pan, L
    Bennani, YL
    Cowart, MD
    Fox, GB
    Sullivan, JP
    FASEB JOURNAL, 2005, 19 (04): : A541 - A541
  • [5] A facile and scaleable synthesis of ABT-239, a benzofuranoid H3 antagonist
    Pu, YM
    Grieme, T
    Gupta, A
    Plata, D
    Bhatia, AV
    Covart, M
    Ku, YY
    ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2005, 9 (01) : 45 - 50
  • [6] Effects of the histamine (H)3 receptor antagonist ABT-239 on acute and repeated nicotine locomotor responses in rats
    Miszkiel, Joanna
    Kruk, Marta
    McCreary, Andrew C.
    Przegalinski, Edmund
    Biala, Grazyna
    Filip, Malgorzata
    PHARMACOLOGICAL REPORTS, 2011, 63 (06) : 1553 - 1559
  • [7] Effects of the histamine (H)3 receptor antagonist ABT-239 on acute and repeated nicotine locomotor responses in rats
    Joanna Miszkiel
    Marta Kruk
    Andrew C. McCreary
    Edmund Przegaliński
    Grażyna Biała
    Małgorzata Filip
    Pharmacological Reports, 2011, 63 : 1553 - 1559
  • [8] Pharmacological properties of the S-enantiomer of the histamine H3 receptor antagonist ABT-239:: An inverse agonist with no anti-obesity effects
    Milicic, I
    Krueger, K
    Miller, T
    Witte, D
    Baranowski, J
    Carr, T
    Sharma, R
    Brunem, M
    Droz, B
    Knourek-Segel, V
    Shapiro, R
    Bush, E
    Jacobson, P
    Bennani, Y
    Cowart, M
    Esbenshade, T
    Hancock, A
    FASEB JOURNAL, 2005, 19 (04): : A95 - A95
  • [9] An efficient and convergent synthesis of the potent and selective H3 antagonist ABT-239
    Ku, YY
    Pu, YM
    Grieme, T
    Sharma, P
    Bhatia, AV
    Cowart, M
    TETRAHEDRON, 2006, 62 (18) : 4584 - 4589
  • [10] LACK OF EFFECTS BY ABT239, A HISTAMINE H3 RECEPTOR ANTAGONIST, IN HISTAMINE-DEFICIENT ANIMALS
    Blandina, P.
    Provensi, G.
    Munari, L.
    Giovannini, M. G.
    Garrison, T.
    Koenig, J. R.
    Cowart, M.
    Brioni, J.
    Passani, M. B.
    INFLAMMATION RESEARCH, 2012, 61 : S62 - S62
12345