Quantitative prediction of histamine H1 receptor occupancy by the sedative and non-sedative antagonists in the human central nervous system based on systemic exposure and preclinical data (vol 32, pg 135, 2017)

被引：0
|
作者：
Kanamitsu, Kayoko [1 ,2 ]
Nozaki, Yoshitane [3 ]
Nagaya, Yoko [3 ]
Sugiyama, Yuichi [4 ]
Kusuhara, Hiroyuki [1 ]
机构：
[1] Univ Tokyo, Grad Sch Pharmaceut Sci, Lab Mol Pharmacokinet, Bunkyo Ku, 7-3-1 Hongo, Tokyo 1130033, Japan
[2] Otsuka Pharmaceut Co Ltd, Tokushima Res Inst, 463-10 Kagasuno,Kawauchi Cho, Tokushima, Tokushima 7710192, Japan
[3] Eisai & Co Ltd, Tsukuba Res Labs, Drug Metab & Pharmacokinet Tsukuba, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, Japan
[4] RIKEN, RIKEN Innovat Ctr, Sugiyama Lab, Res Cluster Innovat,Tsurumi Ku, 1-7-22 Suehiro Cho, Yokohama, Kanagawa 2300045, Japan
来源：
DRUG METABOLISM AND PHARMACOKINETICS | 2017年 / 32卷 / 04期
关键词：
D O I：
10.1016/j.dmpk.2017.05.003
中图分类号：
R9 [药学];
学科分类号：
1007 ;
摘要：
引用
收藏
页码：228 / 228
页数：1
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