Synthesis, analysis and cytotoxic effects of new RGD-mimetics

被引：0
|
作者：
Balacheva, Anelia [1 ]
Dzimbova, Tatyana [1 ]
Detcheva, Roumyana [1 ]
Bruckdorfer, Thomas [2 ]
Momekov, Georgi [3 ]
Pajpanova, Tamara [1 ]
Golovinsky, Evgeny [1 ]
机构：
[1] Bulgarian Acad Sci, Inst Mol Biol Roumen Tsanev, BU-1113 Sofia, Bulgaria
[2] Iris Biotech GmbH, D-95615 Marktredwitz, Germany
[3] Med Univ Sofia, Fac Pharm, Dept Pharmacol Pharmacotherapy & Toxicol, Sofia 1000, Bulgaria
来源：
AMINO ACIDS | 2015年 / 47卷 / 08期
关键词：
D O I：
暂无
中图分类号：
Q5 [生物化学]; Q7 [分子生物学];
学科分类号：
071010 ; 081704 ;
摘要：
引用
收藏
页码：1687 / 1687
页数：1
相关论文
共 50 条
  • [1] In vitro Assessment of the Cytotoxic Effects of Novel RGD-mimetics
    Dzimbova, T.
    Georgiev, L.
    Balacheva, A.
    Iliev, I.
    Detcheva, R.
    Georgieva, M.
    Staneva, D.
    Miloshev, G.
    Pajpanova, T.
    JOURNAL OF PEPTIDE SCIENCE, 2012, 18 : S122 - S122
  • [2] New antithrombotic RGD-mimetics with high bioavailability
    Gante, J
    Juraszyk, H
    Raddatz, P
    Wurziger, H
    BernotatDanielowski, S
    Melzer, G
    Rippmann, F
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1996, 6 (20) : 2425 - 2430
  • [3] Synthesis, analysis and biological evaluation of new RGD mimetics
    Balacheva, A. A.
    Lambev, M. K.
    Pashov, I.
    Detcheva, R. L.
    Sazelova, P.
    Momekov, G. Ts.
    Kasicka, V.
    Pajpanova, T. I.
    Golovinsky, E. V.
    BULGARIAN CHEMICAL COMMUNICATIONS, 2017, 49 : 7 - 10
  • [4] Novel solid-phase synthesis of azapeptides and azapeptoides via Fmoc-strategy and its application in the synthesis of RGD-mimetics
    Gibson, C
    Goodman, SL
    Hahn, D
    Hölzemann, G
    Kessler, H
    JOURNAL OF ORGANIC CHEMISTRY, 1999, 64 (20): : 7388 - 7394
  • [5] Novel solid-phase synthesis of azapeptides and azapeptoides via Fmoc-strategy and its application in the synthesis of RGD-mimetics
    J Org Chem, 20 (7388-7394):
  • [6] RGD-mimetics (RGD-m) bind to platelets regardless of conformational change (CC) to the GPIIb/IIIa receptor.
    Heminway, SJ
    Liu, S
    Rajopadhye, M
    Cheesman, EH
    Harris, TA
    Edwards, DS
    Barrett, JA
    FASEB JOURNAL, 1999, 13 (05): : A838 - A838
  • [7] Synthesis and in vitro potency of αVβ3 receptor antagonists:: A directed approach to RGD-mimetics incorporating novel 3-substituted β-alanines.
    Brashear, K
    Coleman, PJ
    Hutchinson, JH
    Halczenko, W
    McVean, CA
    Duggan, ME
    Hartman, GD
    Hoffman, WF
    Hunt, CA
    Rodan, S
    Rodan, GA
    Leu, CT
    Prueksaritanont, T
    Fernandez-Metzler, C
    Ma, B
    Libby, L
    Merkle, K
    Stump, G
    Wallace, A
    Lynch, R
    Lynch, JJ
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2001, 221 : U46 - U46
  • [8] Synthesis and in vitro potency of αvβ3 receptor antagonists:: A library approach to RGD-mimetics incorporating novel 3-substituted β-alanines.
    McVean, CA
    Askew, BC
    Breslin, MJ
    Hunt, CA
    Leu, CT
    Meissner, RS
    Nagy, R
    Perkins, JJ
    Rodan, S
    Duggan, ME
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2001, 221 : U46 - U46
  • [9] The synthesis of alternative diketopiperazines as potential RGD mimetics
    Mihala, Nikolett
    Csampai, Antal
    Ilas, Janez
    Kikelj, Danijel
    Kiss, Robert
    Suli-Vargha, Helga
    JOURNAL OF PEPTIDE SCIENCE, 2006, 12 (10) : 663 - 669
  • [10] Synthesis and in vitro Assessment of the Cytotoxic Effects of Novel RGD Analogues and Conjugates
    Balacheva, Anelia
    Lambev, Momchil
    Detcheva, Roumyana
    Bruckdorfer, Thomas
    Paypanova, Tamara
    JOURNAL OF PEPTIDE SCIENCE, 2018, 24 : S146 - S146
12345