SIMPLE SYNTHETIC METHOD FOR 1-HYDROXYINDOLE AND ITS APPLICATION TO 1-HYDROXYTRYPTOPHAN DERIVATIVES1,#

被引：13

作者：

Kawasaki, Toshiya ^{[1
]}

Tabata, Mutsuko ^{[1
]}

Nakagawa, Kyoko ^{[1
]}

Kobayashi, Kensuke ^{[1
]}

Kodama, Atsushi ^{[1
]}

Kobayashi, Tetsuya ^{[1
]}

Hasegawa, Masakazu ^{[1
]}

Tanii, Keiko ^{[1
]}

Somei, Masanori ^{[1
]}

机构：

[1] Kanazawa Univ, Grad Sch Nat Sci & Technol, Fac Pharmaceut Sci, Kanazawa, Ishikawa 9201192, Japan

来源：

HETEROCYCLES | 2015年 / 90卷 / 02期

关键词：

1-Hydroxyindole; 1-Hydroxytryptophan; 1-Methoxyindole; 1-Methoxytryptophan; Oxidation; SHORT-STEP SYNTHESIS; UBER ALKALOIDE; CHEMISTRY; INDOLES; PHYTOALEXIN; AMINO; ACID;

D O I：

10.3987/COM-14-S(K)74

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Simple and general synthetic method for 1-hydroxy- and 1-methoxyindole is reported. Its application to the synthesis of various types of 1-hydroxy- and 1-methoxyindole derivatives is successful, especially for the synthesis of 1-hydroxytryptophan derivatives.

引用

页码：1038 / 1071

页数：34

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